Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Histamine H4 receptor (Homo sapiens (Human)) | BDBM227453 (US9333199, S-NORKETOTIFEN (SNORK)) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
BRIDGE PHARMA, INC. US Patent | Assay Description The specific binding of the radioactive ligand to the receptor was defined as the difference between total binding and nonspecific binding, determine... | US Patent US9333199 (2016) BindingDB Entry DOI: 10.7270/Q2639NMV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H4 receptor (Homo sapiens (Human)) | BDBM181150 (US9138431, R-NORKETOTIFEN (RNORK) | US9138431, RS-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | US Patent | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
BRIDGE PHARMA, INC. US Patent | Assay Description The specific binding of the radioactive ligand to the receptor was defined as the difference between total binding and nonspecific binding, determine... | US Patent US9333199 (2016) BindingDB Entry DOI: 10.7270/Q2639NMV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H4 receptor (Homo sapiens (Human)) | BDBM227454 (US9333199, R-NORKETOTIFEN (RNORK)) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 2.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
BRIDGE PHARMA, INC. US Patent | Assay Description The specific binding of the radioactive ligand to the receptor was defined as the difference between total binding and nonspecific binding, determine... | US Patent US9333199 (2016) BindingDB Entry DOI: 10.7270/Q2639NMV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H4 receptor (Homo sapiens (Human)) | BDBM50017674 ((2-Benzhydryloxy-ethyl)-dimethyl-amine | 2-(benzhy...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | US Patent | 1.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
BRIDGE PHARMA, INC. US Patent | Assay Description The specific binding of the radioactive ligand to the receptor was defined as the difference between total binding and nonspecific binding, determine... | US Patent US9333199 (2016) BindingDB Entry DOI: 10.7270/Q2639NMV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H4 receptor (Homo sapiens (Human)) | BDBM50073179 (8-Chloro-11-piperidin-4-ylidene-6,11-dihydro-5H-be...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid PDB UniChem Patents Similars | US Patent | 1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
BRIDGE PHARMA, INC. US Patent | Assay Description The specific binding of the radioactive ligand to the receptor was defined as the difference between total binding and nonspecific binding, determine... | US Patent US9333199 (2016) BindingDB Entry DOI: 10.7270/Q2639NMV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H4 receptor (Homo sapiens (Human)) | BDBM94597 ((Z)-2-butenedioate;10-(1-methyl-4-piperidinylidene...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase DrugBank MCE PC cid PC sid UniChem Similars | US Patent | 2.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
BRIDGE PHARMA, INC. US Patent | Assay Description The specific binding of the radioactive ligand to the receptor was defined as the difference between total binding and nonspecific binding, determine... | US Patent US9333199 (2016) BindingDB Entry DOI: 10.7270/Q2639NMV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Homo sapiens (Human)) | BDBM94597 ((Z)-2-butenedioate;10-(1-methyl-4-piperidinylidene...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase DrugBank MCE PC cid PC sid UniChem Similars | DrugBank US Patent | n/a | n/a | 2.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
BRIDGE PHARMA, INC. US Patent | Assay Description The specific binding of the radioactive ligand to the receptor was defined as the difference between total binding and nonspecific binding, determine... | US Patent US9333199 (2016) BindingDB Entry DOI: 10.7270/Q2639NMV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Homo sapiens (Human)) | BDBM181150 (US9138431, R-NORKETOTIFEN (RNORK) | US9138431, RS-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 1.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
BRIDGE PHARMA, INC. US Patent | Assay Description The specific binding of the radioactive ligand to the receptor was defined as the difference between total binding and nonspecific binding, determine... | US Patent US9333199 (2016) BindingDB Entry DOI: 10.7270/Q2639NMV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Homo sapiens (Human)) | BDBM50073179 (8-Chloro-11-piperidin-4-ylidene-6,11-dihydro-5H-be...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid PDB UniChem Patents Similars | DrugBank US Patent | n/a | n/a | 1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
BRIDGE PHARMA, INC. US Patent | Assay Description The specific binding of the radioactive ligand to the receptor was defined as the difference between total binding and nonspecific binding, determine... | US Patent US9333199 (2016) BindingDB Entry DOI: 10.7270/Q2639NMV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Homo sapiens (Human)) | BDBM227454 (US9333199, R-NORKETOTIFEN (RNORK)) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
BRIDGE PHARMA, INC. US Patent | Assay Description The specific binding of the radioactive ligand to the receptor was defined as the difference between total binding and nonspecific binding, determine... | US Patent US9333199 (2016) BindingDB Entry DOI: 10.7270/Q2639NMV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Homo sapiens (Human)) | BDBM227453 (US9333199, S-NORKETOTIFEN (SNORK)) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
BRIDGE PHARMA, INC. US Patent | Assay Description The specific binding of the radioactive ligand to the receptor was defined as the difference between total binding and nonspecific binding, determine... | US Patent US9333199 (2016) BindingDB Entry DOI: 10.7270/Q2639NMV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Homo sapiens (Human)) | BDBM50017674 ((2-Benzhydryloxy-ethyl)-dimethyl-amine | 2-(benzhy...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | DrugBank US Patent | n/a | n/a | 8.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
BRIDGE PHARMA, INC. US Patent | Assay Description The specific binding of the radioactive ligand to the receptor was defined as the difference between total binding and nonspecific binding, determine... | US Patent US9333199 (2016) BindingDB Entry DOI: 10.7270/Q2639NMV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Homo sapiens (Human)) | BDBM22876 (CHEMBL998 | Claritin | Loratadine | Sch 29851 | US...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid UniChem Patents Similars | DrugBank US Patent | n/a | n/a | 1.50E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
BRIDGE PHARMA, INC. US Patent | Assay Description The specific binding of the radioactive ligand to the receptor was defined as the difference between total binding and nonspecific binding, determine... | US Patent US9333199 (2016) BindingDB Entry DOI: 10.7270/Q2639NMV | |||||||||||
More data for this Ligand-Target Pair |