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| Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM5446 (CHEMBL553 | ERLOTINIB HYDROCHLORIDE | Erlotinib | ...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet  | Purchase CHEMBL DrugBank MCE MMDB PC cid PC sid PDB UniChem Patents Similars | DrugBank MMDB PDB US Patent | n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | 25 |
PHARMAXYN LABORATORIES LTD. US Patent | Assay Description The kinase activity of EGFR was detected according to time-resolved fluorescence detection technology to evaluate automatic phosphorylation levels. T... | US Patent US9409845 (2016) BindingDB Entry DOI: 10.7270/Q25M64MC | |||||||||||
| More data for this Ligand-Target Pair |  3D Structure (crystal) | ||||||||||||
| Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM50424964 (CHEMBL2316151 | US9409845, Table 1, Compound 12: (...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 430 | n/a | n/a | n/a | n/a | n/a | 25 |
PHARMAXYN LABORATORIES LTD. US Patent | Assay Description The kinase activity of EGFR was detected according to time-resolved fluorescence detection technology to evaluate automatic phosphorylation levels. T... | US Patent US9409845 (2016) BindingDB Entry DOI: 10.7270/Q25M64MC | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM50424973 (CHEMBL2316142 | US9409845, Table 1, Compound 3: (2...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 1.54E+3 | n/a | n/a | n/a | n/a | n/a | 25 |
PHARMAXYN LABORATORIES LTD. US Patent | Assay Description The kinase activity of EGFR was detected according to time-resolved fluorescence detection technology to evaluate automatic phosphorylation levels. T... | US Patent US9409845 (2016) BindingDB Entry DOI: 10.7270/Q25M64MC | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM50424975 (CHEMBL2316140 | US9409845, Table 1, Compound 1: (2...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 1.68E+3 | n/a | n/a | n/a | n/a | n/a | 25 |
PHARMAXYN LABORATORIES LTD. US Patent | Assay Description The kinase activity of EGFR was detected according to time-resolved fluorescence detection technology to evaluate automatic phosphorylation levels. T... | US Patent US9409845 (2016) BindingDB Entry DOI: 10.7270/Q25M64MC | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM50424957 (CHEMBL2316158 | US9409845, Table 1, Compound 19: (...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | US Patent | n/a | n/a | 1.96E+3 | n/a | n/a | n/a | n/a | n/a | 25 |
PHARMAXYN LABORATORIES LTD. US Patent | Assay Description The kinase activity of EGFR was detected according to time-resolved fluorescence detection technology to evaluate automatic phosphorylation levels. T... | US Patent US9409845 (2016) BindingDB Entry DOI: 10.7270/Q25M64MC | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM50424958 (CHEMBL2316157 | US9409845, Table 1, Compound 18: (...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 2.08E+3 | n/a | n/a | n/a | n/a | n/a | 25 |
PHARMAXYN LABORATORIES LTD. US Patent | Assay Description The kinase activity of EGFR was detected according to time-resolved fluorescence detection technology to evaluate automatic phosphorylation levels. T... | US Patent US9409845 (2016) BindingDB Entry DOI: 10.7270/Q25M64MC | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM50424972 (CHEMBL2316143 | US9409845, Table 1, Compound 4: (2...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 2.17E+3 | n/a | n/a | n/a | n/a | n/a | 25 |
PHARMAXYN LABORATORIES LTD. US Patent | Assay Description The kinase activity of EGFR was detected according to time-resolved fluorescence detection technology to evaluate automatic phosphorylation levels. T... | US Patent US9409845 (2016) BindingDB Entry DOI: 10.7270/Q25M64MC | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM50424974 (CHEMBL2316141 | US9409845, Table 1, Compound 2: (2...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 2.27E+3 | n/a | n/a | n/a | n/a | n/a | 25 |
PHARMAXYN LABORATORIES LTD. US Patent | Assay Description The kinase activity of EGFR was detected according to time-resolved fluorescence detection technology to evaluate automatic phosphorylation levels. T... | US Patent US9409845 (2016) BindingDB Entry DOI: 10.7270/Q25M64MC | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM50424961 (CHEMBL2316154 | US9409845, Table 1, Compound 15: (...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 3.98E+3 | n/a | n/a | n/a | n/a | n/a | 25 |
PHARMAXYN LABORATORIES LTD. US Patent | Assay Description The kinase activity of EGFR was detected according to time-resolved fluorescence detection technology to evaluate automatic phosphorylation levels. T... | US Patent US9409845 (2016) BindingDB Entry DOI: 10.7270/Q25M64MC | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM50424962 (CHEMBL2316153 | US9409845, Table 1, Compound 14: (...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 4.66E+3 | n/a | n/a | n/a | n/a | n/a | 25 |
PHARMAXYN LABORATORIES LTD. US Patent | Assay Description The kinase activity of EGFR was detected according to time-resolved fluorescence detection technology to evaluate automatic phosphorylation levels. T... | US Patent US9409845 (2016) BindingDB Entry DOI: 10.7270/Q25M64MC | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM50424956 (CHEMBL2316159 | US9409845, Table 1, Compound 20: (...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | US Patent | n/a | n/a | 4.81E+3 | n/a | n/a | n/a | n/a | n/a | 25 |
PHARMAXYN LABORATORIES LTD. US Patent | Assay Description The kinase activity of EGFR was detected according to time-resolved fluorescence detection technology to evaluate automatic phosphorylation levels. T... | US Patent US9409845 (2016) BindingDB Entry DOI: 10.7270/Q25M64MC | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM50424960 (CHEMBL2316155 | US9409845, Table 1, Compound 16: (...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 5.37E+3 | n/a | n/a | n/a | n/a | n/a | 25 |
PHARMAXYN LABORATORIES LTD. US Patent | Assay Description The kinase activity of EGFR was detected according to time-resolved fluorescence detection technology to evaluate automatic phosphorylation levels. T... | US Patent US9409845 (2016) BindingDB Entry DOI: 10.7270/Q25M64MC | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM50424968 (CHEMBL2316147 | US9409845, Table 1, Compound 8: (2...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 5.69E+3 | n/a | n/a | n/a | n/a | n/a | 25 |
PHARMAXYN LABORATORIES LTD. US Patent | Assay Description The kinase activity of EGFR was detected according to time-resolved fluorescence detection technology to evaluate automatic phosphorylation levels. T... | US Patent US9409845 (2016) BindingDB Entry DOI: 10.7270/Q25M64MC | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM50424965 (CHEMBL2316150 | US9409845, Table 1, Compound 11: (...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 6.13E+3 | n/a | n/a | n/a | n/a | n/a | 25 |
PHARMAXYN LABORATORIES LTD. US Patent | Assay Description The kinase activity of EGFR was detected according to time-resolved fluorescence detection technology to evaluate automatic phosphorylation levels. T... | US Patent US9409845 (2016) BindingDB Entry DOI: 10.7270/Q25M64MC | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM50424970 (CHEMBL2316145 | US9409845, Table 1, Compound 6: (2...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 6.85E+3 | n/a | n/a | n/a | n/a | n/a | 25 |
PHARMAXYN LABORATORIES LTD. US Patent | Assay Description The kinase activity of EGFR was detected according to time-resolved fluorescence detection technology to evaluate automatic phosphorylation levels. T... | US Patent US9409845 (2016) BindingDB Entry DOI: 10.7270/Q25M64MC | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM50424969 (CHEMBL2316146 | US9409845, Table 1, Compound 7: (2...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 7.12E+3 | n/a | n/a | n/a | n/a | n/a | 25 |
PHARMAXYN LABORATORIES LTD. US Patent | Assay Description The kinase activity of EGFR was detected according to time-resolved fluorescence detection technology to evaluate automatic phosphorylation levels. T... | US Patent US9409845 (2016) BindingDB Entry DOI: 10.7270/Q25M64MC | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM50424966 (CHEMBL2316149 | US9409845, Table 1, Compound 10: (...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 7.52E+3 | n/a | n/a | n/a | n/a | n/a | 25 |
PHARMAXYN LABORATORIES LTD. US Patent | Assay Description The kinase activity of EGFR was detected according to time-resolved fluorescence detection technology to evaluate automatic phosphorylation levels. T... | US Patent US9409845 (2016) BindingDB Entry DOI: 10.7270/Q25M64MC | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM50424971 (CHEMBL2316144 | US9409845, Table 1, Compound 5: (2...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 8.08E+3 | n/a | n/a | n/a | n/a | n/a | 25 |
PHARMAXYN LABORATORIES LTD. US Patent | Assay Description The kinase activity of EGFR was detected according to time-resolved fluorescence detection technology to evaluate automatic phosphorylation levels. T... | US Patent US9409845 (2016) BindingDB Entry DOI: 10.7270/Q25M64MC | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM50140172 (CHEBI:3962 | CHEMBL140 | Curcumin | US9409845, Tab...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | US Patent | n/a | n/a | 8.65E+3 | n/a | n/a | n/a | n/a | n/a | 25 |
PHARMAXYN LABORATORIES LTD. US Patent | Assay Description The kinase activity of EGFR was detected according to time-resolved fluorescence detection technology to evaluate automatic phosphorylation levels. T... | US Patent US9409845 (2016) BindingDB Entry DOI: 10.7270/Q25M64MC | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM50424967 (CHEMBL2316148 | US9409845, Table 1, Compound 9: (2...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 1.53E+4 | n/a | n/a | n/a | n/a | n/a | 25 |
PHARMAXYN LABORATORIES LTD. US Patent | Assay Description The kinase activity of EGFR was detected according to time-resolved fluorescence detection technology to evaluate automatic phosphorylation levels. T... | US Patent US9409845 (2016) BindingDB Entry DOI: 10.7270/Q25M64MC | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM239058 (US9409845, Table 1, Compound 17: (2E,6E)-2-di-(3,5...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.87E+4 | n/a | n/a | n/a | n/a | n/a | 25 |
PHARMAXYN LABORATORIES LTD. US Patent | Assay Description The kinase activity of EGFR was detected according to time-resolved fluorescence detection technology to evaluate automatic phosphorylation levels. T... | US Patent US9409845 (2016) BindingDB Entry DOI: 10.7270/Q25M64MC | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM50424963 (CHEMBL2316152 | US9409845, Table 1, Compound 13: (...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 2.09E+4 | n/a | n/a | n/a | n/a | n/a | 25 |
PHARMAXYN LABORATORIES LTD. US Patent | Assay Description The kinase activity of EGFR was detected according to time-resolved fluorescence detection technology to evaluate automatic phosphorylation levels. T... | US Patent US9409845 (2016) BindingDB Entry DOI: 10.7270/Q25M64MC | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
