Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248583 (US9434711, 496) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.183 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica, N.V. US Patent | Assay Description For patch clamp experiments, HEK293 cells are stably transfected with canine TRPM8 and cultured in DMEM supplemented with 10% fetal bovine serum, 100... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM50036555 (CHEMBL3353610 | US9434711, 497) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 0.400 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248583 (US9434711, 496) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.554 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica, N.V. US Patent | Assay Description For patch clamp experiments, HEK293 cells are stably transfected with canine TRPM8 and cultured in DMEM supplemented with 10% fetal bovine serum, 100... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248370 (US9434711, 227) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.600 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248576 (US9434711, 489) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.600 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248599 (US9434711, 518) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.700 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248838 (US9434711, 808) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.700 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248426 (US9434711, 292) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.800 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248583 (US9434711, 496) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.800 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248580 (US9434711, 493) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.800 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248480 (US9434711, 361) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.800 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM50426573 (CHEMBL2324349 | US9434711, 306) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 0.800 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248581 (US9434711, 494) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.900 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248789 (US9434711, 755) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.900 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248389 (US9434711, 249) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.900 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248613 (US9434711, 535) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248607 (US9434711, 526) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248458 (US9434711, 335) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248578 (US9434711, 491) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248840 (US9434711, 810) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248577 (US9434711, 490) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248575 (US9434711, 488) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248414 (US9434711, 278) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248361 (US9434711, 218) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248367 (US9434711, 224) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM50426573 (CHEMBL2324349 | US9434711, 306) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 1.10 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Pharmaceutica, N.V. US Patent | Assay Description For patch clamp experiments, HEK293 cells are stably transfected with canine TRPM8 and cultured in DMEM supplemented with 10% fetal bovine serum, 100... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248363 (US9434711, 220) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.20 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248808 (US9434711, 774) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.30 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248415 (US9434711, 279) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.30 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248790 (US9434711, 756) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.40 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential cation channel subfamily M member 8 (Homo sapiens (Human)) | BDBM248583 (US9434711, 496) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.40 | n/a | n/a | n/a | n/a | n/a | 25 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description For functional expression of TRPM8, the full-length cDNA encoding human and rat TRPM8 are subcloned into pCI-NEO mammalian expression vectors. The ex... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248356 (US9434711, 213) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.40 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248809 (US9434711, 775) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.60 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248365 (US9434711, 222) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.70 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248640 (US9434711, 566) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.80 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248622 (US9434711, 544) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.80 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential cation channel subfamily M member 8 (Rattus norvegicus (Rat)) | BDBM248583 (US9434711, 496) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.80 | n/a | n/a | n/a | n/a | n/a | 25 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description For functional expression of TRPM8, the full-length cDNA encoding human and rat TRPM8 are subcloned into pCI-NEO mammalian expression vectors. The ex... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248662 (US9434711, 592) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.80 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248428 (US9434711, 294) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.80 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248623 (US9434711, 545) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.90 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248564 (US9434711, 475) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248549 (US9434711, 453) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248369 (US9434711, 226) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248574 (US9434711, 487) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248538 (US9434711, 439) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248598 (US9434711, 517) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248746 (US9434711, 698) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248758 (US9434711, 711) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248605 (US9434711, 524) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transient receptor potential M8 protein (Canis lupus familiaris (Dog)) | BDBM248602 (US9434711, 521) | PDB KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | 37 |
Janssen Pharmaceutica, N.V. US Patent | Assay Description The functional activity of compounds of the formula (I) was determined by measuring changes in intracellular calcium concentration using a Ca2+-sensi... | US Patent US9434711 (2016) BindingDB Entry DOI: 10.7270/Q2H41QB6 | |||||||||||
More data for this Ligand-Target Pair |
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