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Patent code US9688695

Compile Data Set for Download or QSAR

Found 384 hits of Enzyme Inhibition Constant Data   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM175987
PNG
(US10047103, 20 | US9688695, 20)
Show SMILES COc1nn2cc(nc2s1)-c1cc2c(OCc3csc(n3)C3CCCCC3)cc(OC)cc2o1
Show InChI InChI=1S/C24H24N4O4S2/c1-29-16-8-19(31-12-15-13-33-22(25-15)14-6-4-3-5-7-14)17-10-21(32-20(17)9-16)18-11-28-23(26-18)34-24(27-28)30-2/h8-11,13-14H,3-7,12H2,1-2H3
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n/an/an/an/a 1.10n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM175991
PNG
(US10047103, 24 | US9688695, 24)
Show SMILES COc1nn2cc(nc2s1)-c1cc2c(OCc3csc(n3)-c3ccc(F)cc3F)cc(OC)cc2o1
Show InChI InChI=1S/C24H16F2N4O4S2/c1-31-14-6-19(33-10-13-11-35-22(27-13)15-4-3-12(25)5-17(15)26)16-8-21(34-20(16)7-14)18-9-30-23(28-18)36-24(29-30)32-2/h3-9,11H,10H2,1-2H3
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n/an/an/an/a 1.10n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176009
PNG
(US10047103, 42 | US9688695, 42)
Show SMILES COc1nn2cc(nc2s1)-c1cc2c(OCc3nc(sc3C(C)C)-c3ccc(cc3)C(=O)N(C)C)cc(OC)cc2o1
Show InChI InChI=1S/C30H29N5O5S2/c1-16(2)26-22(31-27(41-26)17-7-9-18(10-8-17)28(36)34(3)4)15-39-23-11-19(37-5)12-24-20(23)13-25(40-24)21-14-35-29(32-21)42-30(33-35)38-6/h7-14,16H,15H2,1-6H3
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n/an/an/an/a 2.5n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176017
PNG
(US10047103, 50 | US9688695, 50)
Show SMILES COc1nn2cc(nc2s1)-c1cc2c(OCc3csc(CC(C)C)n3)cc(OC)cc2o1
Show InChI InChI=1S/C22H22N4O4S2/c1-12(2)5-20-23-13(11-31-20)10-29-17-6-14(27-3)7-18-15(17)8-19(30-18)16-9-26-21(24-16)32-22(25-26)28-4/h6-9,11-12H,5,10H2,1-4H3
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n/an/an/an/a 0.210n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176018
PNG
(US10047103, 51 | US9688695, 51)
Show SMILES COc1nn2cc(nc2s1)-c1cc2c(OCc3csc(n3)N3C[C@H](C)O[C@H](C)C3)cc(OC)cc2o1 |r|
Show InChI InChI=1S/C24H25N5O5S2/c1-13-8-28(9-14(2)33-13)22-25-15(12-35-22)11-32-19-5-16(30-3)6-20-17(19)7-21(34-20)18-10-29-23(26-18)36-24(27-29)31-4/h5-7,10,12-14H,8-9,11H2,1-4H3/t13-,14+
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n/an/an/an/a 0.260n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176029
PNG
(US10047103, 62 | US9688695, 62)
Show SMILES COc1nn2cc(nc2s1)-c1cc2c(OCc3csc(n3)-c3cccc(OC(C)=O)c3)cc(OC)cc2o1
Show InChI InChI=1S/C26H20N4O6S2/c1-14(31)35-17-6-4-5-15(7-17)24-27-16(13-37-24)12-34-21-8-18(32-2)9-22-19(21)10-23(36-22)20-11-30-25(28-20)38-26(29-30)33-3/h4-11,13H,12H2,1-3H3
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n/an/an/an/a 0.480n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176032
PNG
(US10047103, 65 | US9688695, 65)
Show SMILES COc1nn2cc(nc2s1)-c1cc2c(OCc3csc(n3)-c3cccc(c3)C(=O)N(C)C)cc(OC)cc2o1
Show InChI InChI=1S/C27H23N5O5S2/c1-31(2)25(33)16-7-5-6-15(8-16)24-28-17(14-38-24)13-36-21-9-18(34-3)10-22-19(21)11-23(37-22)20-12-32-26(29-20)39-27(30-32)35-4/h5-12,14H,13H2,1-4H3
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BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176033
PNG
(US10047103, 66 | US9688695, 66)
Show SMILES COc1nn2cc(nc2s1)-c1cc2c(OCc3nc(sc3C)-c3ccc(cc3)C(=O)N(C)C)cc(OC)cc2o1
Show InChI InChI=1S/C28H25N5O5S2/c1-15-21(29-25(39-15)16-6-8-17(9-7-16)26(34)32(2)3)14-37-22-10-18(35-4)11-23-19(22)12-24(38-23)20-13-33-27(30-20)40-28(31-33)36-5/h6-13H,14H2,1-5H3
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n/an/an/an/a 0.75n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176036
PNG
(US10047103, 69 | US9688695, 69)
Show SMILES COc1nn2cc(nc2s1)-c1cc2c(OCc3csc(n3)-c3ccc(CO)cc3)cc(OC)cc2o1
Show InChI InChI=1S/C25H20N4O5S2/c1-31-17-7-20(33-12-16-13-35-23(26-16)15-5-3-14(11-30)4-6-15)18-9-22(34-21(18)8-17)19-10-29-24(27-19)36-25(28-29)32-2/h3-10,13,30H,11-12H2,1-2H3
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n/an/an/an/a 0.230n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176041
PNG
(US10047103, 74 | US9688695, 74)
Show SMILES COc1nn2cc(nc2s1)-c1cc2c(OCc3csc(n3)-c3ccc(C)nc3)cc(OC)cc2o1
Show InChI InChI=1S/C24H19N5O4S2/c1-13-4-5-14(9-25-13)22-26-15(12-34-22)11-32-19-6-16(30-2)7-20-17(19)8-21(33-20)18-10-29-23(27-18)35-24(28-29)31-3/h4-10,12H,11H2,1-3H3
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BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176072
PNG
(US10047103, 105 | US9688695, 105)
Show SMILES CCc1sc(nc1COc1cc(OC)cc2oc(cc12)-c1cn2nc(OC)sc2n1)N1CCOCC1
Show InChI InChI=1S/C24H25N5O5S2/c1-4-21-17(26-22(35-21)28-5-7-32-8-6-28)13-33-18-9-14(30-2)10-19-15(18)11-20(34-19)16-12-29-23(25-16)36-24(27-29)31-3/h9-12H,4-8,13H2,1-3H3
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n/an/an/an/a 0.320n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176088
PNG
(US10047103, 121 | US9688695, 121)
Show SMILES COc1nn2cc(nc2s1)-c1cc2c(OCc3csc(n3)C3(O)CC(C)OC(C)C3)cc(OC)cc2o1
Show InChI InChI=1S/C25H26N4O6S2/c1-13-8-25(30,9-14(2)34-13)22-26-15(12-36-22)11-33-19-5-16(31-3)6-20-17(19)7-21(35-20)18-10-29-23(27-18)37-24(28-29)32-4/h5-7,10,12-14,30H,8-9,11H2,1-4H3
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n/an/an/an/a 0.270n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176089
PNG
(US10047103, 122 | US9688695, 122)
Show SMILES COc1nn2cc(nc2s1)-c1cc2c(OCc3csc(n3)C3(F)CC(C)OC(C)C3)cc(OC)cc2o1
Show InChI InChI=1S/C25H25FN4O5S2/c1-13-8-25(26,9-14(2)34-13)22-27-15(12-36-22)11-33-19-5-16(31-3)6-20-17(19)7-21(35-20)18-10-30-23(28-18)37-24(29-30)32-4/h5-7,10,12-14H,8-9,11H2,1-4H3
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BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176104
PNG
(US10047103, 137 | US9688695, 137)
Show SMILES COc1nn2cc(nc2s1)-c1cc2c(OCc3csc(n3)C(O)(c3ccccc3)C(F)(F)F)cc(OC)cc2o1
Show InChI InChI=1S/C26H19F3N4O5S2/c1-35-16-8-19(17-10-21(38-20(17)9-16)18-11-33-23(31-18)40-24(32-33)36-2)37-12-15-13-39-22(30-15)25(34,26(27,28)29)14-6-4-3-5-7-14/h3-11,13,34H,12H2,1-2H3
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BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176110
PNG
(US10047103, 143 | US9688695, 143)
Show SMILES COc1nn2cc(nc2s1)-c1cc2c(OCc3csc(n3)C(C)(O)C(F)(F)F)cc(OC)cc2o1
Show InChI InChI=1S/C21H17F3N4O5S2/c1-20(29,21(22,23)24)17-25-10(9-34-17)8-32-14-4-11(30-2)5-15-12(14)6-16(33-15)13-7-28-18(26-13)35-19(27-28)31-3/h4-7,9,29H,8H2,1-3H3
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BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176117
PNG
(US10047103, 150 | US9688695, 150)
Show SMILES COc1nn2cc(nc2s1)-c1cc2c(OCc3csc(n3)C3(O)CCC(CC3)C(O)=O)cc(OC)cc2o1 |(-12.26,-1.72,;-11.49,-.38,;-9.89,-.38,;-8.99,.86,;-7.52,.38,;-6.06,.86,;-5.15,-.38,;-6.06,-1.63,;-7.52,-1.15,;-8.99,-1.63,;-3.7,-.38,;-2.79,.86,;-1.33,.38,;.01,1.15,;.01,2.7,;1.34,3.47,;2.67,2.7,;2.67,1.15,;4.14,.68,;5.04,1.93,;4.14,3.17,;6.77,1.94,;6,.61,;7.54,.61,;9.08,.61,;9.85,1.94,;9.08,3.27,;7.54,3.27,;11.39,1.94,;12.26,.43,;12.16,3.27,;1.34,.38,;1.34,-1.15,;2.67,-1.93,;2.67,-3.47,;.01,-1.93,;-1.33,-1.15,;-2.79,-1.63,)|
Show InChI InChI=1S/C25H24N4O7S2/c1-33-15-7-18(35-11-14-12-37-22(26-14)25(32)5-3-13(4-6-25)21(30)31)16-9-20(36-19(16)8-15)17-10-29-23(27-17)38-24(28-29)34-2/h7-10,12-13,32H,3-6,11H2,1-2H3,(H,30,31)
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BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176123
PNG
(US10047103, 156 | US9688695, 156)
Show SMILES COc1nn2cc(nc2s1)-c1cc2c(OCc3csc(n3)C3(CCOCC3)c3ccccc3F)cc(OC)cc2o1
Show InChI InChI=1S/C29H25FN4O5S2/c1-35-18-11-23(19-13-25(39-24(19)12-18)22-14-34-27(32-22)41-28(33-34)36-2)38-15-17-16-40-26(31-17)29(7-9-37-10-8-29)20-5-3-4-6-21(20)30/h3-6,11-14,16H,7-10,15H2,1-2H3
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BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176131
PNG
(US10047103, 164 | US9688695, 164)
Show SMILES COc1nn2cc(nc2s1)-c1cc2c(OCc3csc(n3)C3(CCOC3)c3ccc(C)cc3)cc(OC)cc2o1
Show InChI InChI=1S/C29H26N4O5S2/c1-17-4-6-18(7-5-17)29(8-9-36-16-29)26-30-19(15-39-26)14-37-23-10-20(34-2)11-24-21(23)12-25(38-24)22-13-33-27(31-22)40-28(32-33)35-3/h4-7,10-13,15H,8-9,14,16H2,1-3H3
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n/an/an/an/a 1.30n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176146
PNG
(US10047103, 179 | US9605024, Example 36 | US968869...)
Show SMILES COc1nn2cc(nc2s1)-c1cc2c(OCc3csc(n3)-c3ccccc3)cc(F)cc2o1
Show InChI InChI=1S/C23H15FN4O3S2/c1-29-23-27-28-10-17(26-22(28)33-23)20-9-16-18(7-14(24)8-19(16)31-20)30-11-15-12-32-21(25-15)13-5-3-2-4-6-13/h2-10,12H,11H2,1H3
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n/an/an/an/a 1n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176149
PNG
(US10047103, 182 | US9688695, 182)
Show SMILES COc1nn2cc(nc2s1)-c1cc2c(OCc3csc(n3)-c3ccc(cc3)C(=O)N(C)C(C)(C)C)cc(F)cc2o1
Show InChI InChI=1S/C29H26FN5O4S2/c1-29(2,3)34(4)26(36)17-8-6-16(7-9-17)25-31-19(15-40-25)14-38-22-10-18(30)11-23-20(22)12-24(39-23)21-13-35-27(32-21)41-28(33-35)37-5/h6-13,15H,14H2,1-5H3
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n/an/an/an/a 0.300n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176165
PNG
(US10047103, 198 | US9688695, 198)
Show SMILES COc1cc(OCc2csc(n2)C2(O)CC(C)OC(C)C2)c2cc(oc2c1)-c1cn2nc(sc2n1)[C@H](C)F |r|
Show InChI InChI=1S/C26H27FN4O5S2/c1-13-8-26(32,9-14(2)35-13)24-28-16(12-37-24)11-34-20-5-17(33-4)6-21-18(20)7-22(36-21)19-10-31-25(29-19)38-23(30-31)15(3)27/h5-7,10,12-15,32H,8-9,11H2,1-4H3/t13?,14?,15-,26?/m0/s1
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n/an/an/an/a 0.420n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176175
PNG
(US10047103, 208 | US9688695, 208)
Show SMILES COc1cc(OCc2csc(n2)-c2ccc(cc2)C(F)(F)F)c2cc(oc2c1)-c1cn2nc(C)ccc2n1
Show InChI InChI=1S/C27H19F3N4O3S/c1-15-3-8-25-32-21(12-34(25)33-15)24-11-20-22(9-19(35-2)10-23(20)37-24)36-13-18-14-38-26(31-18)16-4-6-17(7-5-16)27(28,29)30/h3-12,14H,13H2,1-2H3
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n/an/an/an/a 0.820n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176191
PNG
(US10047103, 224 | US9688695, 224)
Show SMILES COc1cc(OCc2csc(n2)-c2ccc(cc2)C#N)c2cc(oc2c1)-c1cn2nc(C)ccc2n1
Show InChI InChI=1S/C27H19N5O3S/c1-16-3-8-26-30-22(13-32(26)31-16)25-11-21-23(9-20(33-2)10-24(21)35-25)34-14-19-15-36-27(29-19)18-6-4-17(12-28)5-7-18/h3-11,13,15H,14H2,1-2H3
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n/an/an/an/a 0.75n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176194
PNG
(US10047103, 227 | US9688695, 227)
Show SMILES COc1cc(OCc2nc(sc2C)-c2ccnc(F)c2)c2cc(oc2c1)-c1cn2nc(C)ccc2n1
Show InChI InChI=1S/C26H20FN5O3S/c1-14-4-5-25-29-19(12-32(25)31-14)23-11-18-21(9-17(33-3)10-22(18)35-23)34-13-20-15(2)36-26(30-20)16-6-7-28-24(27)8-16/h4-12H,13H2,1-3H3
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n/an/an/an/a 0.310n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176203
PNG
(US10047103, 236 | US9688695, 236)
Show SMILES COc1cc(OCc2csc(n2)N2CCN(CC2)S(C)(=O)=O)c2cc(oc2c1)-c1cn2nc(C)ccc2n1
Show InChI InChI=1S/C25H26N6O5S2/c1-16-4-5-24-27-20(13-31(24)28-16)23-12-19-21(10-18(34-2)11-22(19)36-23)35-14-17-15-37-25(26-17)29-6-8-30(9-7-29)38(3,32)33/h4-5,10-13,15H,6-9,14H2,1-3H3
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n/an/an/an/a 1.90n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176209
PNG
(US10047103, 242 | US9688695, 242)
Show SMILES COc1cc(OCc2csc(n2)C2(CCOCC2)c2ccc(C)cc2)c2cc(oc2c1)-c1cn2nc(C)ccc2n1
Show InChI InChI=1S/C32H30N4O4S/c1-20-4-7-22(8-5-20)32(10-12-38-13-11-32)31-33-23(19-41-31)18-39-27-14-24(37-3)15-28-25(27)16-29(40-28)26-17-36-30(34-26)9-6-21(2)35-36/h4-9,14-17,19H,10-13,18H2,1-3H3
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n/an/an/an/a 0.590n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176211
PNG
(US10047103, 244 | US9688695, 244)
Show SMILES COc1cc(OCc2csc(NCCN3CCOCC3)n2)c2cc(oc2c1)-c1cn2nc(C)ccc2n1
Show InChI InChI=1S/C26H28N6O4S/c1-17-3-4-25-29-21(14-32(25)30-17)24-13-20-22(11-19(33-2)12-23(20)36-24)35-15-18-16-37-26(28-18)27-5-6-31-7-9-34-10-8-31/h3-4,11-14,16H,5-10,15H2,1-2H3,(H,27,28)
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n/an/an/an/a 909n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176213
PNG
(US10047103, 246 | US9688695, 246)
Show SMILES COCCN(CCOC)c1nc(COc2cc(OC)cc3oc(cc23)-c2cn3nc(C)ccc3n2)cs1
Show InChI InChI=1S/C26H29N5O5S/c1-17-5-6-25-28-21(14-31(25)29-17)24-13-20-22(11-19(34-4)12-23(20)36-24)35-15-18-16-37-26(27-18)30(7-9-32-2)8-10-33-3/h5-6,11-14,16H,7-10,15H2,1-4H3
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n/an/an/an/a 1.40n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176218
PNG
(US10047103, 251 | US9688695, 251)
Show SMILES COCCNc1nc(COc2cc(OC)cc3oc(cc23)-c2cn3nc(C)ccc3n2)cs1
Show InChI InChI=1S/C23H23N5O4S/c1-14-4-5-22-26-18(11-28(22)27-14)21-10-17-19(8-16(30-3)9-20(17)32-21)31-12-15-13-33-23(25-15)24-6-7-29-2/h4-5,8-11,13H,6-7,12H2,1-3H3,(H,24,25)
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n/an/an/an/a 11n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176232
PNG
(US10047103, 265 | US9688695, 265)
Show SMILES COc1cc(OCc2csc(Nc3cc(F)ccc3F)n2)c2cc(oc2c1)-c1cn2nc(C)ccc2n1
Show InChI InChI=1S/C26H19F2N5O3S/c1-14-3-6-25-30-21(11-33(25)32-14)24-10-18-22(8-17(34-2)9-23(18)36-24)35-12-16-13-37-26(29-16)31-20-7-15(27)4-5-19(20)28/h3-11,13H,12H2,1-2H3,(H,29,31)
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n/an/an/an/a 48n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176234
PNG
(US10047103, 267 | US9688695, 267)
Show SMILES COc1cc(OCc2csc(Nc3cccc(C)c3)n2)c2cc(oc2c1)-c1cn2nc(C)ccc2n1
Show InChI InChI=1S/C27H23N5O3S/c1-16-5-4-6-18(9-16)28-27-29-19(15-36-27)14-34-23-10-20(33-3)11-24-21(23)12-25(35-24)22-13-32-26(30-22)8-7-17(2)31-32/h4-13,15H,14H2,1-3H3,(H,28,29)
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n/an/an/an/a 4.20n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176238
PNG
(US10047103, 271 | US9688695, 271)
Show SMILES CCC1CCN(CC1)c1nc(COc2cc(OC)cc3oc(cc23)-c2cn3nc(C)ccc3n2)cs1
Show InChI InChI=1S/C27H29N5O3S/c1-4-18-7-9-31(10-8-18)27-28-19(16-36-27)15-34-23-11-20(33-3)12-24-21(23)13-25(35-24)22-14-32-26(29-22)6-5-17(2)30-32/h5-6,11-14,16,18H,4,7-10,15H2,1-3H3
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n/an/an/an/a 1.30n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176242
PNG
(US10047103, 275 | US9688695, 275)
Show SMILES COc1cc(OCc2csc(n2)N2CCC[C@H]2C)c2cc(oc2c1)-c1cn2nc(C)ccc2n1 |r|
Show InChI InChI=1S/C25H25N5O3S/c1-15-6-7-24-27-20(12-30(24)28-15)23-11-19-21(9-18(31-3)10-22(19)33-23)32-13-17-14-34-25(26-17)29-8-4-5-16(29)2/h6-7,9-12,14,16H,4-5,8,13H2,1-3H3/t16-/m1/s1
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n/an/an/an/a 4.20n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176248
PNG
(US10047103, 281 | US9688695, 281)
Show SMILES COc1cc(OCc2csc(Nc3ccc4scnc4c3)n2)c2cc(oc2c1)-c1cn2nc(C)ccc2n1
Show InChI InChI=1S/C27H20N6O3S2/c1-15-3-6-26-31-21(11-33(26)32-15)24-10-19-22(8-18(34-2)9-23(19)36-24)35-12-17-13-37-27(30-17)29-16-4-5-25-20(7-16)28-14-38-25/h3-11,13-14H,12H2,1-2H3,(H,29,30)
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BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176262
PNG
(US10047103, 295 | US9688695, 295)
Show SMILES COc1nn2cc(nc2s1)-c1cc2c(OCc3csc(n3)-c3ccc(cc3)C(=O)NC3COC3)cc(OC)cc2o1
Show InChI InChI=1S/C28H23N5O6S2/c1-35-19-7-22(20-9-24(39-23(20)8-19)21-10-33-27(31-21)41-28(32-33)36-2)38-13-18-14-40-26(30-18)16-5-3-15(4-6-16)25(34)29-17-11-37-12-17/h3-10,14,17H,11-13H2,1-2H3,(H,29,34)
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n/an/an/an/a 92n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176264
PNG
(US10047103, 297 | US9688695, 297)
Show SMILES COc1nn2cc(nc2s1)-c1cc2c(OCc3csc(n3)-c3ccc(cc3)C(=O)N(C)C(C)(C)C)cc(OC)cc2o1
Show InChI InChI=1S/C30H29N5O5S2/c1-30(2,3)34(4)27(36)18-9-7-17(8-10-18)26-31-19(16-41-26)15-39-23-11-20(37-5)12-24-21(23)13-25(40-24)22-14-35-28(32-22)42-29(33-35)38-6/h7-14,16H,15H2,1-6H3
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BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176269
PNG
(US10047103, 302 | US9688695, 302)
Show SMILES COc1nn2cc(nc2s1)-c1cc2c(OCc3csc(n3)-c3ccc(cc3)C(=O)N3CCC(C)CC3)cc(OC)cc2o1
Show InChI InChI=1S/C31H29N5O5S2/c1-18-8-10-35(11-9-18)29(37)20-6-4-19(5-7-20)28-32-21(17-42-28)16-40-25-12-22(38-2)13-26-23(25)14-27(41-26)24-15-36-30(33-24)43-31(34-36)39-3/h4-7,12-15,17-18H,8-11,16H2,1-3H3
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n/an/an/an/a 0.440n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176270
PNG
(US10047103, 303 | US9688695, 303)
Show SMILES COc1nn2cc(nc2s1)-c1cc2c(OCc3csc(n3)-c3ccc(cc3)C(=O)N3CCCCCC3)cc(OC)cc2o1
Show InChI InChI=1S/C31H29N5O5S2/c1-38-22-13-25(23-15-27(41-26(23)14-22)24-16-36-30(33-24)43-31(34-36)39-2)40-17-21-18-42-28(32-21)19-7-9-20(10-8-19)29(37)35-11-5-3-4-6-12-35/h7-10,13-16,18H,3-6,11-12,17H2,1-2H3
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n/an/an/an/a 0.850n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176276
PNG
(US10047103, 309 | US9688695, 309)
Show SMILES CCCN(CC)C(=O)c1ccc(cc1)-c1nc(COc2cc(OC)cc3oc(cc23)-c2cn3nc(OC)sc3n2)cs1
Show InChI InChI=1S/C30H29N5O5S2/c1-5-11-34(6-2)28(36)19-9-7-18(8-10-19)27-31-20(17-41-27)16-39-24-12-21(37-3)13-25-22(24)14-26(40-25)23-15-35-29(32-23)42-30(33-35)38-4/h7-10,12-15,17H,5-6,11,16H2,1-4H3
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n/an/an/an/a 0.540n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176280
PNG
(US10047103, 313 | US9688695, 313)
Show SMILES CCCN(C(C)C1CC1)C(=O)c1ccc(cc1)-c1nc(COc2cc(OC)cc3oc(cc23)-c2cn3nc(OC)sc3n2)cs1
Show InChI InChI=1S/C33H33N5O5S2/c1-5-12-37(19(2)20-6-7-20)31(39)22-10-8-21(9-11-22)30-34-23(18-44-30)17-42-27-13-24(40-3)14-28-25(27)15-29(43-28)26-16-38-32(35-26)45-33(36-38)41-4/h8-11,13-16,18-20H,5-7,12,17H2,1-4H3
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n/an/an/an/a 0.430n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, HEK293 EBNA PAR4 clone 20664.1J cells were plated 24 hrs. prior to experiment in 384 well, Poly-D-Lysine coated, black, clear bottom plates ...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM175969
PNG
(US10047103, 2 | US9605024, Example 2 | US9688695, ...)
Show SMILES COc1nn2cc(nc2s1)-c1cc2c(OCc3csc(n3)C(F)(F)F)cc(OC)cc2o1
Show InChI InChI=1S/C19H13F3N4O4S2/c1-27-10-3-13(29-7-9-8-31-16(23-9)19(20,21)22)11-5-15(30-14(11)4-10)12-6-26-17(24-12)32-18(25-26)28-2/h3-6,8H,7H2,1-2H3
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n/an/an/an/a 49n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, PRP or washed platelet suspension (100 μl) was pre-incubated for 5 minutes at room temperature with varying concentrations of compounds...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM175970
PNG
(US10047103, 3 | US9605024, Example 3 | US9688695, ...)
Show SMILES COc1nn2cc(nc2s1)-c1cc2c(OCc3csc(n3)-c3ccccc3)cc(OC)cc2o1
Show InChI InChI=1S/C24H18N4O4S2/c1-29-16-8-19(31-12-15-13-33-22(25-15)14-6-4-3-5-7-14)17-10-21(32-20(17)9-16)18-11-28-23(26-18)34-24(27-28)30-2/h3-11,13H,12H2,1-2H3
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n/an/an/an/a 4.70n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, PRP or washed platelet suspension (100 μl) was pre-incubated for 5 minutes at room temperature with varying concentrations of compounds...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM175985
PNG
(US10047103, 18 | US9605024, Example 18 | US9688695...)
Show SMILES COc1nn2cc(nc2s1)-c1cc2c(OCc3csc(n3)-c3ccc(OC)cc3)cc(OC)cc2o1
Show InChI InChI=1S/C25H20N4O5S2/c1-30-16-6-4-14(5-7-16)23-26-15(13-35-23)12-33-20-8-17(31-2)9-21-18(20)10-22(34-21)19-11-29-24(27-19)36-25(28-29)32-3/h4-11,13H,12H2,1-3H3
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n/an/an/an/a 3.60n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, PRP or washed platelet suspension (100 μl) was pre-incubated for 5 minutes at room temperature with varying concentrations of compounds...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM175995
PNG
(US10047103, 75 | US9605024, Example 28 | US9688695...)
Show SMILES COc1nn2cc(nc2s1)-c1cc2c(OCc3csc(n3)-c3ccncc3)cc(OC)cc2o1
Show InChI InChI=1S/C23H17N5O4S2/c1-29-15-7-18(31-11-14-12-33-21(25-14)13-3-5-24-6-4-13)16-9-20(32-19(16)8-15)17-10-28-22(26-17)34-23(27-28)30-2/h3-10,12H,11H2,1-2H3
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n/an/an/an/a 2.90n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, PRP or washed platelet suspension (100 μl) was pre-incubated for 5 minutes at room temperature with varying concentrations of compounds...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176015
PNG
(US10047103, 48 | US9688695, 48)
Show SMILES COc1nn2cc(nc2s1)-c1cc2c(OCc3nc(sc3C)-c3ccc(cc3)C(=O)N(C)CC#N)cc(OC)cc2o1
Show InChI InChI=1S/C29H24N6O5S2/c1-16-22(31-26(41-16)17-5-7-18(8-6-17)27(36)34(2)10-9-30)15-39-23-11-19(37-3)12-24-20(23)13-25(40-24)21-14-35-28(32-21)42-29(33-35)38-4/h5-8,11-14H,10,15H2,1-4H3
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n/an/an/an/a 1.20n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, PRP or washed platelet suspension (100 μl) was pre-incubated for 5 minutes at room temperature with varying concentrations of compounds...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176034
PNG
(US10047103, 67 | US9688695, 67)
Show SMILES COc1nn2cc(nc2s1)-c1cc2c(OCc3csc(n3)-c3ccnc(F)c3)cc(OC)cc2o1
Show InChI InChI=1S/C23H16FN5O4S2/c1-30-14-6-17(32-10-13-11-34-21(26-13)12-3-4-25-20(24)5-12)15-8-19(33-18(15)7-14)16-9-29-22(27-16)35-23(28-29)31-2/h3-9,11H,10H2,1-2H3
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n/an/an/an/a 2.20n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, PRP or washed platelet suspension (100 μl) was pre-incubated for 5 minutes at room temperature with varying concentrations of compounds...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176088
PNG
(US10047103, 121 | US9688695, 121)
Show SMILES COc1nn2cc(nc2s1)-c1cc2c(OCc3csc(n3)C3(O)CC(C)OC(C)C3)cc(OC)cc2o1
Show InChI InChI=1S/C25H26N4O6S2/c1-13-8-25(30,9-14(2)34-13)22-26-15(12-36-22)11-33-19-5-16(31-3)6-20-17(19)7-21(35-20)18-10-29-23(27-18)37-24(28-29)32-4/h5-7,10,12-14,30H,8-9,11H2,1-4H3
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n/an/an/an/a 27n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, PRP or washed platelet suspension (100 μl) was pre-incubated for 5 minutes at room temperature with varying concentrations of compounds...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176106
PNG
(US10047103, 139 | US9688695, 139)
Show SMILES CCC(F)(c1nc(COc2cc(OC)cc3oc(cc23)-c2cn3nc(OC)sc3n2)cs1)C(F)(F)F
Show InChI InChI=1S/C22H18F4N4O4S2/c1-4-21(23,22(24,25)26)18-27-11(10-35-18)9-33-15-5-12(31-2)6-16-13(15)7-17(34-16)14-8-30-19(28-14)36-20(29-30)32-3/h5-8,10H,4,9H2,1-3H3
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n/an/an/an/a 26n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, PRP or washed platelet suspension (100 μl) was pre-incubated for 5 minutes at room temperature with varying concentrations of compounds...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176176
PNG
(US10047103, 209 | US9688695, 209)
Show SMILES COc1cc(OCc2csc(n2)-c2ccc(Cl)cc2)c2cc(oc2c1)-c1cn2nc(C)ccc2n1
Show InChI InChI=1S/C26H19ClN4O3S/c1-15-3-8-25-29-21(12-31(25)30-15)24-11-20-22(9-19(32-2)10-23(20)34-24)33-13-18-14-35-26(28-18)16-4-6-17(27)7-5-16/h3-12,14H,13H2,1-2H3
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n/an/an/an/a 23n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, PRP or washed platelet suspension (100 μl) was pre-incubated for 5 minutes at room temperature with varying concentrations of compounds...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
Proteinase-activated receptor 4


(Homo sapiens (Human))		BDBM176211
PNG
(US10047103, 244 | US9688695, 244)
Show SMILES COc1cc(OCc2csc(NCCN3CCOCC3)n2)c2cc(oc2c1)-c1cn2nc(C)ccc2n1
Show InChI InChI=1S/C26H28N6O4S/c1-17-3-4-25-29-21(14-32(25)30-17)24-13-20-22(11-19(33-2)12-23(20)36-24)35-15-18-16-37-26(28-18)27-5-6-31-7-9-34-10-8-31/h3-4,11-14,16H,5-10,15H2,1-2H3,(H,27,28)
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n/an/an/an/a>3.00E+3n/an/an/a25



BRISTOL-MYERS SQUIBB COMPANY

US Patent


Assay Description
Briefly, PRP or washed platelet suspension (100 μl) was pre-incubated for 5 minutes at room temperature with varying concentrations of compounds...

US Patent US9688695 (2017)


BindingDB Entry DOI: 10.7270/Q28K777N
More data for this
Ligand-Target Pair
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* indicates data uncertainty>20%