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| Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM50365262 ((+)-JQ1 | (S)-JQ1 (1) | CHEMBL1957266 | JQ1 | US10...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet  | Purchase CHEMBL MCE MMDB PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 44 | n/a | n/a | n/a | n/a | 7.5 | 25 |
Dana-Farber Cancer Institute, Inc. US Patent | Assay Description Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150 mM ... | US Patent US9695172 (2017) BindingDB Entry DOI: 10.7270/Q2JD4TX8 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain testis-specific protein (Homo sapiens (Human)) | BDBM50365262 ((+)-JQ1 | (S)-JQ1 (1) | CHEMBL1957266 | JQ1 | US10...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 147 | n/a | n/a | n/a | n/a | 7.5 | 25 |
Dana-Farber Cancer Institute, Inc. US Patent | Assay Description Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150 mM ... | US Patent US9695172 (2017) BindingDB Entry DOI: 10.7270/Q2JD4TX8 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM106150 (US9695172, 3) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 1.37E+3 | n/a | n/a | n/a | n/a | 7.5 | 25 |
Dana-Farber Cancer Institute, Inc. US Patent | Assay Description Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150 mM ... | US Patent US9695172 (2017) BindingDB Entry DOI: 10.7270/Q2JD4TX8 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM106153 (US9695172, 2-227) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 2.14E+3 | n/a | n/a | n/a | n/a | 7.5 | 25 |
Dana-Farber Cancer Institute, Inc. US Patent | Assay Description Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150 mM ... | US Patent US9695172 (2017) BindingDB Entry DOI: 10.7270/Q2JD4TX8 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM106152 (US9695172, 2-221) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 2.99E+3 | n/a | n/a | n/a | n/a | 7.5 | 25 |
Dana-Farber Cancer Institute, Inc. US Patent | Assay Description Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150 mM ... | US Patent US9695172 (2017) BindingDB Entry DOI: 10.7270/Q2JD4TX8 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain testis-specific protein (Homo sapiens (Human)) | BDBM106150 (US9695172, 3) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 3.68E+3 | n/a | n/a | n/a | n/a | 7.5 | 25 |
Dana-Farber Cancer Institute, Inc. US Patent | Assay Description Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150 mM ... | US Patent US9695172 (2017) BindingDB Entry DOI: 10.7270/Q2JD4TX8 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain testis-specific protein (Homo sapiens (Human)) | BDBM106153 (US9695172, 2-227) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 5.41E+3 | n/a | n/a | n/a | n/a | 7.5 | 25 |
Dana-Farber Cancer Institute, Inc. US Patent | Assay Description Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150 mM ... | US Patent US9695172 (2017) BindingDB Entry DOI: 10.7270/Q2JD4TX8 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain testis-specific protein (Homo sapiens (Human)) | BDBM106152 (US9695172, 2-221) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 5.66E+3 | n/a | n/a | n/a | n/a | 7.5 | 25 |
Dana-Farber Cancer Institute, Inc. US Patent | Assay Description Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150 mM ... | US Patent US9695172 (2017) BindingDB Entry DOI: 10.7270/Q2JD4TX8 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Leucine-rich repeat serine/threonine-protein kinase 2 (Homo sapiens (Human)) | BDBM106150 (US9695172, 3) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | 7.5 | 25 |
Dana-Farber Cancer Institute, Inc. US Patent | Assay Description Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150 mM ... | US Patent US9695172 (2017) BindingDB Entry DOI: 10.7270/Q2JD4TX8 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Aurora kinase B (Homo sapiens (Human)) | BDBM106152 (US9695172, 2-221) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | 7.5 | 25 |
Dana-Farber Cancer Institute, Inc. US Patent | Assay Description Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150 mM ... | US Patent US9695172 (2017) BindingDB Entry DOI: 10.7270/Q2JD4TX8 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Aurora kinase C (Homo sapiens (Human)) | BDBM106152 (US9695172, 2-221) | PDB NCI pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | 7.5 | 25 |
Dana-Farber Cancer Institute, Inc. US Patent | Assay Description Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150 mM ... | US Patent US9695172 (2017) BindingDB Entry DOI: 10.7270/Q2JD4TX8 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Leucine-rich repeat serine/threonine-protein kinase 2 (Homo sapiens (Human)) | BDBM106153 (US9695172, 2-227) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | 7.5 | 25 |
Dana-Farber Cancer Institute, Inc. US Patent | Assay Description Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150 mM ... | US Patent US9695172 (2017) BindingDB Entry DOI: 10.7270/Q2JD4TX8 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Aurora kinase A (Homo sapiens (Human)) | BDBM106152 (US9695172, 2-221) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | 7.5 | 25 |
Dana-Farber Cancer Institute, Inc. US Patent | Assay Description Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150 mM ... | US Patent US9695172 (2017) BindingDB Entry DOI: 10.7270/Q2JD4TX8 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain-containing protein 4 (Homo sapiens (Human)) | BDBM50355500 (CHEMBL1908394 | US9695172, GSK461364) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | 7.5 | 25 |
Dana-Farber Cancer Institute, Inc. US Patent | Assay Description Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150 mM ... | US Patent US9695172 (2017) BindingDB Entry DOI: 10.7270/Q2JD4TX8 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Bromodomain testis-specific protein (Homo sapiens (Human)) | BDBM50355500 (CHEMBL1908394 | US9695172, GSK461364) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | 7.5 | 25 |
Dana-Farber Cancer Institute, Inc. US Patent | Assay Description Assays were performed with minor modifications from the manufacturer's protocol (PerkinElmer, USA). All reagents were diluted in 50 mM HEPES, 150 mM ... | US Patent US9695172 (2017) BindingDB Entry DOI: 10.7270/Q2JD4TX8 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
