Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
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Enoyl-[acyl-carrier-protein] reductase [NADH] (260/260 = 100%)† (Francisella tularensis subsp. tularensis (strain S...) | BDBM50392117 (CHEMBL1945507) | PDB MMDB KEGG UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MMDB PC cid PC sid PDB UniChem Similars | PDB Article PubMed | 360 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Illinois at Chicago Curated by ChEMBL | Assay Description Competitive inhibition of Francisella tularensis subsp. tularensis SCHU4 N-terminal His-tagged FabI expressed in Escherichia coli BL21(DE3) using cro... | J Med Chem 55: 5933-41 (2012) Article DOI: 10.1021/jm300489v BindingDB Entry DOI: 10.7270/Q2S46T27 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) |