Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
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Bifunctional epoxide hydrolase 2 (555/555 = 100%)† (Homo sapiens (Human)) | BDBM50002344 (CHEMBL3233607) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | PDB Article PubMed | n/a | n/a | 2.90E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Astellas Pharma Inc. Curated by ChEMBL | Assay Description Inhibition of human full-length C-terminal His6-tagged sEH expressed in Escherichia coli BL21(DE3) cells using PHOME as substrate incubated with enzy... | Bioorg Med Chem 22: 2427-34 (2014) Article DOI: 10.1016/j.bmc.2014.03.001 BindingDB Entry DOI: 10.7270/Q2NV9KRF | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) |