Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Glucose-1-phosphate thymidylyltransferase (293/293 = 100%)† (Pseudomonas aeruginosa) | BDBM93091 (Analogue of 1a, 8k) | PDB MMDB KEGG UniProtKB/TrEMBL B.MOAD DrugBank GoogleScholar AffyNet | MMDB PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | 205 | n/a | n/a | n/a | n/a | n/a | n/a |
University of St. Andrews | Assay Description Inhibition assay using glucose-1-phosphate thymidylyltransferase (RmlA). | ACS Chem Biol 8: 387-96 (2013) Article DOI: 10.1021/cb300426u BindingDB Entry DOI: 10.7270/Q26D5RMP | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) |