Affinity Data by PubMed id=10514288

PubMed code 10514288

Found 12 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
B2 bradykinin receptor (Homo sapiens (Human))	BDBM50403371 (Firazyr \| HOE-140 \| ICATIBANT) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Similars	PubMed	0.0640	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£s Montpellier I et II Curated by ChEMBL					Assay Description Binding affinity against human cloned Bradykinin receptor B2 expressed in CHO cells using [3H]-bradykinin as radioligand				J Med Chem 42: 4185-92 (1999) BindingDB Entry DOI: 10.7270/Q25Q4WTF
Universit£s Montpellier I et II Curated by ChEMBL					More data for this Ligand-Target Pair
B2 bradykinin receptor (RAT)	BDBM50403371 (Firazyr \| HOE-140 \| ICATIBANT) Show SMILES Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	Purchase KEGG PC cid PC sid UniChem Similars	PubMed	0.0770	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£s Montpellier I et II Curated by ChEMBL					Assay Description Binding affinity against rat bradykinin B2 receptors expressed in CHO cells using [3H]bradykinin as radioligand				J Med Chem 42: 4185-92 (1999) BindingDB Entry DOI: 10.7270/Q25Q4WTF
Universit£s Montpellier I et II Curated by ChEMBL					More data for this Ligand-Target Pair
B2 bradykinin receptor (RAT)	BDBM50049949 ((BK) H-Arg-Pro-Pro-Gly-Phe-Ser-Pro-Phe-Arg-OH \| (b...) Show SMILES Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	PubMed	0.460	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£s Montpellier I et II Curated by ChEMBL					Assay Description Binding affinity against rat Bradykinin receptor B2 expressed in CHO cells using [3H]-bradykinin as radioligand				J Med Chem 42: 4185-92 (1999) BindingDB Entry DOI: 10.7270/Q25Q4WTF
Universit£s Montpellier I et II Curated by ChEMBL					More data for this Ligand-Target Pair
B2 bradykinin receptor (Homo sapiens (Human))	BDBM50049949 ((BK) H-Arg-Pro-Pro-Gly-Phe-Ser-Pro-Phe-Arg-OH \| (b...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	PubMed	0.650	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£s Montpellier I et II Curated by ChEMBL					Assay Description Binding affinity against human cloned Bradykinin receptor B2 expressed in CHO cells using [3H]-bradykinin as radioligand				J Med Chem 42: 4185-92 (1999) BindingDB Entry DOI: 10.7270/Q25Q4WTF
Universit£s Montpellier I et II Curated by ChEMBL					More data for this Ligand-Target Pair
B2 bradykinin receptor (Homo sapiens (Human))	BDBM50408748 (CHEMBL2112698) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL KEGG PC cid PC sid UniChem Similars	PubMed	0.700	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£s Montpellier I et II Curated by ChEMBL					Assay Description Binding affinity against human cloned Bradykinin receptor B2 expressed in CHO cells using [3H]-bradykinin as radioligand				J Med Chem 42: 4185-92 (1999) BindingDB Entry DOI: 10.7270/Q25Q4WTF
Universit£s Montpellier I et II Curated by ChEMBL					More data for this Ligand-Target Pair
B2 bradykinin receptor (RAT)	BDBM50408748 (CHEMBL2112698) Show SMILES Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL KEGG PC cid PC sid UniChem Similars	PubMed	6	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£s Montpellier I et II Curated by ChEMBL					Assay Description Binding affinity against rat bradykinin B2 receptors expressed in CHO cells using [3H]bradykinin as radioligand				J Med Chem 42: 4185-92 (1999) BindingDB Entry DOI: 10.7270/Q25Q4WTF
Universit£s Montpellier I et II Curated by ChEMBL					More data for this Ligand-Target Pair
B2 bradykinin receptor (Homo sapiens (Human))	BDBM50081653 (CHEMBL413386 \| [2-[2-(3-Amino-4-oxo-3,4-dihydro-2H...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	13	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£s Montpellier I et II Curated by ChEMBL					Assay Description Binding affinity against human cloned Bradykinin receptor B2 expressed in CHO cells using [3H]-bradykinin as radioligand				J Med Chem 42: 4185-92 (1999) BindingDB Entry DOI: 10.7270/Q25Q4WTF
Universit£s Montpellier I et II Curated by ChEMBL					More data for this Ligand-Target Pair
B2 bradykinin receptor (Homo sapiens (Human))	BDBM50081652 ((RMP-7)H-Arg-Pro-Hyp-Gly-Ser-Pro-4-Me-Tyr(CH2NH2)-...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL KEGG PC cid PC sid UniChem Similars	PubMed	19	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£s Montpellier I et II Curated by ChEMBL					Assay Description Binding affinity against human cloned Bradykinin receptor B2 expressed in CHO cells using [3H]-bradykinin as radioligand				J Med Chem 42: 4185-92 (1999) BindingDB Entry DOI: 10.7270/Q25Q4WTF
Universit£s Montpellier I et II Curated by ChEMBL					More data for this Ligand-Target Pair
B2 bradykinin receptor (Homo sapiens (Human))	BDBM50408749 (CHEMBL2111889) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL KEGG PC cid PC sid UniChem Similars	PubMed	162	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£s Montpellier I et II Curated by ChEMBL					Assay Description Binding affinity against human cloned Bradykinin receptor B2 expressed in CHO cells using [3H]-bradykinin as radioligand				J Med Chem 42: 4185-92 (1999) BindingDB Entry DOI: 10.7270/Q25Q4WTF
Universit£s Montpellier I et II Curated by ChEMBL					More data for this Ligand-Target Pair
B1 bradykinin receptor (Homo sapiens (Human))	BDBM50408749 (CHEMBL2111889) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL KEGG PC cid PC sid UniChem Similars	PubMed	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£s Montpellier I et II Curated by ChEMBL					Assay Description Binding affinity against human cloned Bradykinin receptor B1 expressed in CHO cells using [3H]-bradykinin as radioligand				J Med Chem 42: 4185-92 (1999) BindingDB Entry DOI: 10.7270/Q25Q4WTF
Universit£s Montpellier I et II Curated by ChEMBL					More data for this Ligand-Target Pair
B1 bradykinin receptor (Homo sapiens (Human))	BDBM50081653 (CHEMBL413386 \| [2-[2-(3-Amino-4-oxo-3,4-dihydro-2H...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£s Montpellier I et II Curated by ChEMBL					Assay Description Binding affinity against human cloned Bradykinin receptor B1 expressed in CHO cells using [3H]-bradykinin as radioligand				J Med Chem 42: 4185-92 (1999) BindingDB Entry DOI: 10.7270/Q25Q4WTF
Universit£s Montpellier I et II Curated by ChEMBL					More data for this Ligand-Target Pair
B1 bradykinin receptor (Homo sapiens (Human))	BDBM50408748 (CHEMBL2112698) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL KEGG PC cid PC sid UniChem Similars	PubMed	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£s Montpellier I et II Curated by ChEMBL					Assay Description Binding affinity against human cloned Bradykinin receptor B1 expressed in CHO cells using [3H]-bradykinin as radioligand				J Med Chem 42: 4185-92 (1999) BindingDB Entry DOI: 10.7270/Q25Q4WTF
Universit£s Montpellier I et II Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%