Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Metabotropic glutamate receptor 1 (Homo sapiens (Human)) | BDBM17657 ((2S)-2-aminopentanedioic acid | (S)-Glu | D-Glutam...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | PubMed | n/a | n/a | n/a | n/a | 1.05E+3 | n/a | n/a | n/a | n/a |
CNRS Curated by ChEMBL | Assay Description Effect of compound on Metabotropic glutamate receptor 1 expressed in HEK 293 cells was determined by measuring IP production relative to glutamate | Bioorg Med Chem Lett 10: 129-33 (2000) BindingDB Entry DOI: 10.7270/Q2P84CFG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 1 (Homo sapiens (Human)) | BDBM50084962 ((2S,3S,4S)-2-Amino-3,4-dihydroxy-pentanedioic acid...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | n/a | 2.57E+5 | n/a | n/a | n/a | n/a |
CNRS Curated by ChEMBL | Assay Description Effect of compound on Metabotropic glutamate receptor 1 expressed in HEK 293 cells was determined by measuring IP production relative to glutamate | Bioorg Med Chem Lett 10: 129-33 (2000) BindingDB Entry DOI: 10.7270/Q2P84CFG | |||||||||||
More data for this Ligand-Target Pair |