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| Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50121977 (2-(3,4-Dimethoxy-phenyl)-5-[2-(3,4-dimethoxy-pheny...) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet  | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 300 | n/a | n/a | n/a | n/a | n/a | n/a |
Dr. Margarete Fischer-Bosch-Institute of Clinical Pharmacology Curated by ChEMBL | Assay Description TP_TRANSPORTER: inhibition of Digoxin transepithelial transport (basal to apical) (Digoxin: 5 uM) in Caco-2 cells | J Pharmacol Exp Ther 293: 376-82 (2000) BindingDB Entry DOI: 10.7270/Q2RB75VT | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50420214 (CHEMBL2074918) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Dr. Margarete Fischer-Bosch-Institute of Clinical Pharmacology Curated by ChEMBL | Assay Description TP_TRANSPORTER: inhibition of Digoxin transepithelial transport (basal to apical) (Digoxin: 5 uM) in Caco-2 cells | J Pharmacol Exp Ther 293: 376-82 (2000) BindingDB Entry DOI: 10.7270/Q2RB75VT | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
