Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Platelet-activating factor acetylhydrolase (Homo sapiens (Human)) | BDBM50097709 (CHEMBL351434 | {5-[1-[(Dodecyl-methyl-carbamoyl)-m...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 533 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Pharmaceuticals Curated by ChEMBL | Assay Description Concentration required for inhibition ofLipoprotein associated phospholipase A2 in rat at dose 2 micromol/kg/h | Bioorg Med Chem Lett 11: 701-4 (2001) BindingDB Entry DOI: 10.7270/Q27W6BF0 | |||||||||||
More data for this Ligand-Target Pair |