Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Adenosine receptor A3 (Homo sapiens (Human)) | BDBM50100418 ((1S,2R,3S,4R,5S)-4-(6-(3-iodobenzylamino)-2-chloro...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Ability to displace specific radioligand [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cells | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 (Homo sapiens (Human)) | BDBM50088428 ((1R,2R,3S,4R,5S)-4-[2-Chloro-6-(3-iodo-benzylamino...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 2.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Displacement of [125I]AB-MECA from human Adenosine A3 receptor expressed in CHO cells expressed as Ki | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 (Homo sapiens (Human)) | BDBM50100423 ((1S,2R,3S,4R,5S)-2,3-Dihydroxy-4-[6-(3-iodo-benzyl...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 2.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Ability to displace specific radioligand [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cells | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 (Homo sapiens (Human)) | BDBM50088425 ((1R,2R,3S,4R,5S)-1-Hydroxymethyl-4-[6-(3-iodo-benz...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 4.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Displacement of [125I]AB-MECA from human Adenosine A3 receptor expressed in CHO cells | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1 (Rattus norvegicus (rat)) | BDBM50088424 ((1R,2R,3S,4R,5S)-4-(6-Cyclopentylamino-purin-9-yl)...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 5.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Ability to displace specific radioligand [3H]R-PIA binding at Adenosine A1 receptor in rat brain membrane | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 (Homo sapiens (Human)) | BDBM50100416 ((1S,2R,3S,4R,5S)-4-(2-Chloro-6-methylamino-purin-9...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 6.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Ability to displace specific radioligand [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cells | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1 (Rattus norvegicus (rat)) | BDBM50088423 ((1R,2R,3S,4R,5S)-4-(2-Chloro-6-cyclopentylamino-pu...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 8.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Ability to displace specific radioligand [3H]R-PIA binding at Adenosine A1 receptor in rat brain membrane | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 (Homo sapiens (Human)) | BDBM50100425 ((1R,2R,3S,4R,5S)-4-(2-Chloro-6-methylamino-purin-9...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 23 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Ability to displace specific radioligand [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cells | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 (Homo sapiens (Human)) | BDBM50100419 ((1S,2R,3S,4R,5S)-4-(6-Amino-purin-9-yl)-2,3-dihydr...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Ability to displace specific radioligand [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cells | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1 (Rattus norvegicus (rat)) | BDBM50100419 ((1S,2R,3S,4R,5S)-4-(6-Amino-purin-9-yl)-2,3-dihydr...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 32 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Ability to displace specific radioligand [3H]R-PIA binding at Adenosine A1 receptor in rat brain membrane | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1 (Rattus norvegicus (rat)) | BDBM50100423 ((1S,2R,3S,4R,5S)-2,3-Dihydroxy-4-[6-(3-iodo-benzyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 53 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Ability to displace specific radioligand [3H]R-PIA binding at Adenosine A1 receptor in rat brain membrane | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1 (Rattus norvegicus (rat)) | BDBM50088425 ((1R,2R,3S,4R,5S)-1-Hydroxymethyl-4-[6-(3-iodo-benz...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 69 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Ability to displace specific radioligand [3H]R-PIA binding at Adenosine A1 receptor in rat brain membrane | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1 (Rattus norvegicus (rat)) | BDBM50100418 ((1S,2R,3S,4R,5S)-4-(6-(3-iodobenzylamino)-2-chloro...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 84 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Ability to displace specific radioligand [3H]R-PIA binding at Adenosine A1 receptor in rat brain membrane | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 (Homo sapiens (Human)) | BDBM50100420 ((1R,2R,3S,4R,5S)-4-(6-Amino-2-chloro-purin-9-yl)-1...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 85 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Ability to displace specific radioligand [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cells | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A2a (Rattus norvegicus (rat)) | BDBM50100419 ((1S,2R,3S,4R,5S)-4-(6-Amino-purin-9-yl)-2,3-dihydr...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Displacement of [3H]-CGS- 21680 from Adenosine A2A receptor in rat brain membrane | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1 (Rattus norvegicus (rat)) | BDBM50088428 ((1R,2R,3S,4R,5S)-4-[2-Chloro-6-(3-iodo-benzylamino...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 141 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Ability to displace specific radioligand [3H]R-PIA binding at Adenosine A1 receptor in rat brain membrane | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 (Homo sapiens (Human)) | BDBM50088424 ((1R,2R,3S,4R,5S)-4-(6-Cyclopentylamino-purin-9-yl)...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 170 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Ability to displace specific radioligand [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cells | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1 (Rattus norvegicus (rat)) | BDBM50100420 ((1R,2R,3S,4R,5S)-4-(6-Amino-2-chloro-purin-9-yl)-1...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 273 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Ability to displace specific radioligand [3H]R-PIA binding at Adenosine A1 receptor in rat brain membrane | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 (Homo sapiens (Human)) | BDBM50088427 ((1R,2R,3S,4R,5S)-4-(6-Amino-purin-9-yl)-1-hydroxym...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 404 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Displacement of [125I]AB-MECA from human Adenosine A3 receptor expressed in CHO cells in absence of adenosine deaminase | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 (Homo sapiens (Human)) | BDBM50088423 ((1R,2R,3S,4R,5S)-4-(2-Chloro-6-cyclopentylamino-pu...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 466 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Displacement of [125I]AB-MECA from human Adenosine A3 receptor expressed in CHO cells | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A2a (Rattus norvegicus (rat)) | BDBM50100423 ((1S,2R,3S,4R,5S)-2,3-Dihydroxy-4-[6-(3-iodo-benzyl...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 548 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Ability to displace specific radioligand [3H]-CGS- 21680 binding at A2A receptors (rA2A) in rat brain membrane | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A2a (Rattus norvegicus (rat)) | BDBM50088425 ((1R,2R,3S,4R,5S)-1-Hydroxymethyl-4-[6-(3-iodo-benz...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 601 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Ability to displace specific radioligand [3H]-CGS- 21680 binding at A2A receptors (rA2A) in rat brain membrane | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A2a (Rattus norvegicus (rat)) | BDBM50088428 ((1R,2R,3S,4R,5S)-4-[2-Chloro-6-(3-iodo-benzylamino...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 732 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Ability to displace specific radioligand [3H]-CGS- 21680 binding at A2A receptors (rA2A) in rat brain membrane | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1 (Rattus norvegicus (rat)) | BDBM50100416 ((1S,2R,3S,4R,5S)-4-(2-Chloro-6-methylamino-purin-9...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 805 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Ability to displace specific radioligand [3H]R-PIA binding at Adenosine A1 receptor in rat brain membrane | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1 (Rattus norvegicus (rat)) | BDBM50100425 ((1R,2R,3S,4R,5S)-4-(2-Chloro-6-methylamino-purin-9...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 884 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Ability to displace specific radioligand [3H]R-PIA binding at Adenosine A1 receptor in rat brain membrane | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 (Homo sapiens (Human)) | BDBM50100421 ((1R,2S,4S,5S)-4-[2-Chloro-6-(3-iodo-benzylamino)-p...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 912 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Ability to displace specific radioligand [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cells | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 (Homo sapiens (Human)) | BDBM50100417 ((1R,2S,4S,5S)-4-(2-Chloro-6-cyclopentylamino-purin...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.09E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Ability to displace specific radioligand [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cells | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1 (Rattus norvegicus (rat)) | BDBM50100424 ((1R,2R,3S,4R,5S)-1-Hydroxymethyl-4-(6-methylamino-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.47E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Ability to displace specific radioligand [3H]R-PIA binding at Adenosine A1 receptor in rat brain membrane | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A2a (Rattus norvegicus (rat)) | BDBM50100418 ((1S,2R,3S,4R,5S)-4-(6-(3-iodobenzylamino)-2-chloro...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.66E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Ability to displace specific radioligand [3H]-CGS- 21680 binding at A2A receptors (rA2A) in rat brain membrane | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1 (Rattus norvegicus (rat)) | BDBM50088427 ((1R,2R,3S,4R,5S)-4-(6-Amino-purin-9-yl)-1-hydroxym...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.68E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Ability to displace specific radioligand [3H]R-PIA binding at Adenosine A1 receptor in rat brain membrane | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A2a (Rattus norvegicus (rat)) | BDBM50100420 ((1R,2R,3S,4R,5S)-4-(6-Amino-2-chloro-purin-9-yl)-1...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.91E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Displacement of [3H]-CGS- 21680 from Adenosine A2A receptor in rat brain membrane | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 (Homo sapiens (Human)) | BDBM50100422 ((1R,2S,4S,5S)-4-(6-Cyclopentylamino-purin-9-yl)-1-...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 2.88E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Ability to displace specific radioligand [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cells | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A2a (Rattus norvegicus (rat)) | BDBM50088423 ((1R,2R,3S,4R,5S)-4-(2-Chloro-6-cyclopentylamino-pu...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 3.39E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Ability to displace specific radioligand [3H]-CGS- 21680 binding at A2A receptors (rA2A) in rat brain membrane | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1 (Rattus norvegicus (rat)) | BDBM50100417 ((1R,2S,4S,5S)-4-(2-Chloro-6-cyclopentylamino-purin...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 3.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Ability to displace specific radioligand [3H]R-PIA binding at Adenosine A1 receptor in rat brain membrane | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1 (Rattus norvegicus (rat)) | BDBM50100422 ((1R,2S,4S,5S)-4-(6-Cyclopentylamino-purin-9-yl)-1-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 5.11E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Ability to displace specific radioligand [3H]R-PIA binding at Adenosine A1 receptor in rat brain membrane | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A2a (Rattus norvegicus (rat)) | BDBM50088424 ((1R,2R,3S,4R,5S)-4-(6-Cyclopentylamino-purin-9-yl)...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 6.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Ability to displace specific radioligand [3H]-CGS- 21680 binding at A2A receptors (rA2A) in rat brain membrane | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1 (Rattus norvegicus (rat)) | BDBM50100421 ((1R,2S,4S,5S)-4-[2-Chloro-6-(3-iodo-benzylamino)-p...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 8.73E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Ability to displace specific radioligand [3H]R-PIA binding at Adenosine A1 receptor in rat brain membrane | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A2a (Homo sapiens (Human)) | BDBM50088427 ((1R,2R,3S,4R,5S)-4-(6-Amino-purin-9-yl)-1-hydroxym...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 2.25E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Displacement of [3H]-CGS- 21680 from A2A receptor in human brain membrane | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A2a (Rattus norvegicus (rat)) | BDBM50100421 ((1R,2S,4S,5S)-4-[2-Chloro-6-(3-iodo-benzylamino)-p...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 2.54E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Ability to displace specific radioligand [3H]-CGS- 21680 binding at A2A receptors (rA2A) in rat brain membrane | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 (Homo sapiens (Human)) | BDBM21220 ((2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Similars | PubMed | n/a | n/a | n/a | n/a | 3.03E+5 | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Agonist efficacy as effective concentration to stimulate binding of [35S]GTP-gamma-S, by activation of human A3AR receptor | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 (Homo sapiens (Human)) | BDBM50100423 ((1S,2R,3S,4R,5S)-2,3-Dihydroxy-4-[6-(3-iodo-benzyl...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | n/a | 6.80E+3 | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Agonist efficacy as effective concentration to stimulate binding of [35S]GTP-gamma-S, by activation of human A3AR receptor | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 (Homo sapiens (Human)) | BDBM50100418 ((1S,2R,3S,4R,5S)-4-(6-(3-iodobenzylamino)-2-chloro...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | n/a | 5.25E+3 | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Agonist efficacy as effective concentration to stimulate binding of [35S]GTP-gamma-S, by activation of human A3AR receptor | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1 (Homo sapiens (Human)) | BDBM50100417 ((1R,2S,4S,5S)-4-(2-Chloro-6-cyclopentylamino-purin...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | n/a | 2.28E+3 | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Agonist efficacy as effective concentration to stimulate binding of [35S]GTP-gamma-S, at human Adenosine A1 receptor | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1 (Homo sapiens (Human)) | BDBM50100422 ((1R,2S,4S,5S)-4-(6-Cyclopentylamino-purin-9-yl)-1-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | n/a | 2.89E+3 | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Agonist efficacy as effective concentration to stimulate binding of [35S]GTP-gamma-S, at human A1 adenosine receptor | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A3 (Homo sapiens (Human)) | BDBM50100416 ((1S,2R,3S,4R,5S)-4-(2-Chloro-6-methylamino-purin-9...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | n/a | 2.55E+4 | n/a | n/a | n/a | n/a |
NIDDK Curated by ChEMBL | Assay Description Agonist efficacy as effective concentration to stimulate binding of [35S]GTP-gamma-S, by activation of human A3AR receptor | Bioorg Med Chem Lett 11: 1333-7 (2001) BindingDB Entry DOI: 10.7270/Q2445N1F | |||||||||||
More data for this Ligand-Target Pair |