Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
P2Y purinoceptor 12 (Homo sapiens (Human)) | BDBM50101892 (2-(7-Ethoxy-4-hydroxy-2,2-dioxo-2H-2lambda*6*,9-di...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | n/a |
COR Therapeutics, Inc. Curated by ChEMBL | Assay Description Ability to displace [3H]-2-MeS-ADP from human Purinergic receptor P2Y12 | Bioorg Med Chem Lett 11: 1805-8 (2001) BindingDB Entry DOI: 10.7270/Q2VT1RC2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2Y purinoceptor 12 (Homo sapiens (Human)) | BDBM50101892 (2-(7-Ethoxy-4-hydroxy-2,2-dioxo-2H-2lambda*6*,9-di...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 170 | n/a | n/a | n/a | n/a | n/a | n/a |
COR Therapeutics, Inc. Curated by ChEMBL | Assay Description Ability to displace [3H]-2-MeS-ADP from human Purinergic receptor P2Y12 | Bioorg Med Chem Lett 11: 1805-8 (2001) BindingDB Entry DOI: 10.7270/Q2VT1RC2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2Y purinoceptor 12 (Homo sapiens (Human)) | BDBM50101903 (CHEMBL50806 | N-(6-Ethoxy-benzothiazol-2-yl)-2-(6-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | 170 | n/a | n/a | n/a | n/a | n/a | n/a |
COR Therapeutics, Inc. Curated by ChEMBL | Assay Description Ability to displace [3H]-2-MeS-ADP from human Purinergic receptor P2Y12 | Bioorg Med Chem Lett 11: 1805-8 (2001) BindingDB Entry DOI: 10.7270/Q2VT1RC2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2Y purinoceptor 12 (Homo sapiens (Human)) | BDBM50101894 (2-(4-Hydroxy-7-methoxy-2,2-dioxo-2H-2lambda*6*,9-d...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 800 | n/a | n/a | n/a | n/a | n/a | n/a |
COR Therapeutics, Inc. Curated by ChEMBL | Assay Description Ability to displace [3H]-2-MeS-ADP from human Purinergic receptor P2Y12 | Bioorg Med Chem Lett 11: 1805-8 (2001) BindingDB Entry DOI: 10.7270/Q2VT1RC2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2Y purinoceptor 12 (Homo sapiens (Human)) | BDBM50101898 (2-(4-Hydroxy-7-methanesulfonyl-2,2-dioxo-2H-2lambd...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
COR Therapeutics, Inc. Curated by ChEMBL | Assay Description Ability to displace [3H]-2-MeS-ADP from human Purinergic receptor P2Y12 | Bioorg Med Chem Lett 11: 1805-8 (2001) BindingDB Entry DOI: 10.7270/Q2VT1RC2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2Y purinoceptor 12 (Homo sapiens (Human)) | BDBM50101896 (3-[2-(6-Ethoxycarbonyl-benzothiazol-2-ylsulfamoyl)...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
COR Therapeutics, Inc. Curated by ChEMBL | Assay Description Ability to displace [3H]-2-MeS-ADP from human Purinergic receptor P2Y12 | Bioorg Med Chem Lett 11: 1805-8 (2001) BindingDB Entry DOI: 10.7270/Q2VT1RC2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2Y purinoceptor 12 (Homo sapiens (Human)) | BDBM50101890 (2-(4-Hydroxy-2,2-dioxo-2H-2lambda*6*,9-dithia-1,4a...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
COR Therapeutics, Inc. Curated by ChEMBL | Assay Description Ability to displace [3H]-2-MeS-ADP from human Purinergic receptor P2Y12 | Bioorg Med Chem Lett 11: 1805-8 (2001) BindingDB Entry DOI: 10.7270/Q2VT1RC2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2Y purinoceptor 12 (Homo sapiens (Human)) | BDBM50101893 (2-(4-Hydroxy-7-methyl-2,2-dioxo-2H-2lambda*6*,9-di...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
COR Therapeutics, Inc. Curated by ChEMBL | Assay Description Ability to displace [3H]-2-MeS-ADP from human Purinergic receptor P2Y12 | Bioorg Med Chem Lett 11: 1805-8 (2001) BindingDB Entry DOI: 10.7270/Q2VT1RC2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2Y purinoceptor 12 (Homo sapiens (Human)) | BDBM50101895 (2-(7-Chloro-4-hydroxy-2,2-dioxo-2H-2lambda*6*,9-di...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 3.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
COR Therapeutics, Inc. Curated by ChEMBL | Assay Description Ability to displace [3H]-2-MeS-ADP from human Purinergic receptor P2Y12 | Bioorg Med Chem Lett 11: 1805-8 (2001) BindingDB Entry DOI: 10.7270/Q2VT1RC2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2Y purinoceptor 12 (Homo sapiens (Human)) | BDBM50101900 (2-(4-Hydroxy-7-nitro-2,2-dioxo-2H-2lambda*6*,9-dit...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 3.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
COR Therapeutics, Inc. Curated by ChEMBL | Assay Description Ability to displace [3H]-2-MeS-ADP from human Purinergic receptor P2Y12 | Bioorg Med Chem Lett 11: 1805-8 (2001) BindingDB Entry DOI: 10.7270/Q2VT1RC2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2Y purinoceptor 12 (Homo sapiens (Human)) | BDBM50101897 (2-(7-Fluoro-4-hydroxy-2,2-dioxo-2H-2lambda*6*,9-di...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 3.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
COR Therapeutics, Inc. Curated by ChEMBL | Assay Description Ability to displace [3H]-2-MeS-ADP from human Purinergic receptor P2Y12 | Bioorg Med Chem Lett 11: 1805-8 (2001) BindingDB Entry DOI: 10.7270/Q2VT1RC2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2Y purinoceptor 12 (Homo sapiens (Human)) | BDBM50101899 (2-(4-Hydroxy-2,2-dioxo-7-phenoxy-2H-2lambda*6*,9-d...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
COR Therapeutics, Inc. Curated by ChEMBL | Assay Description Ability to displace [3H]-2-MeS-ADP from human Purinergic receptor P2Y12 | Bioorg Med Chem Lett 11: 1805-8 (2001) BindingDB Entry DOI: 10.7270/Q2VT1RC2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2Y purinoceptor 12 (Homo sapiens (Human)) | BDBM50101902 (2-(4-Hydroxy-2,2-dioxo-7-phenyl-2H-2lambda*6*,9-di...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
COR Therapeutics, Inc. Curated by ChEMBL | Assay Description Ability to displace [3H]-2-MeS-ADP from human Purinergic receptor P2Y12 | Bioorg Med Chem Lett 11: 1805-8 (2001) BindingDB Entry DOI: 10.7270/Q2VT1RC2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2Y purinoceptor 12 (Homo sapiens (Human)) | BDBM50101891 (5-Methoxy-2,2-dioxo-2H-2lambda*6*,9-dithia-1,4a-di...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 7.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
COR Therapeutics, Inc. Curated by ChEMBL | Assay Description Ability to displace [3H]-2-MeS-ADP from human Purinergic receptor P2Y12 | Bioorg Med Chem Lett 11: 1805-8 (2001) BindingDB Entry DOI: 10.7270/Q2VT1RC2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2Y purinoceptor 12 (Homo sapiens (Human)) | BDBM50101901 (2,2-Dioxo-7-trifluoromethoxy-2H-2lambda*6*,9-dithi...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >1.20E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
COR Therapeutics, Inc. Curated by ChEMBL | Assay Description Ability to displace [3H]-2-MeS-ADP from human Purinergic receptor P2Y12 | Bioorg Med Chem Lett 11: 1805-8 (2001) BindingDB Entry DOI: 10.7270/Q2VT1RC2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2Y purinoceptor 12 (Homo sapiens (Human)) | BDBM50101889 (2-(7-Cyclohexyl-4-hydroxy-2,2-dioxo-2H-2lambda*6*,...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >1.20E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
COR Therapeutics, Inc. Curated by ChEMBL | Assay Description Ability to displace [3H]-2-MeS-ADP from human Purinergic receptor P2Y12 | Bioorg Med Chem Lett 11: 1805-8 (2001) BindingDB Entry DOI: 10.7270/Q2VT1RC2 | |||||||||||
More data for this Ligand-Target Pair |