Affinity Data by PubMed id=11906293

PubMed code 11906293

Found 7 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Peroxisome proliferator-activated receptor gamma/Retinoic acid receptor RXR-alpha (Homo sapiens (Human))	BDBM50111009 (5-{3-[4-(5-Methyl-2-phenyl-oxazol-4-ylmethoxy)-phe...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	n/a	n/a	119	n/a	n/a	n/a	n/a
Takeda Chemical Industries, Ltd. Curated by ChEMBL					Assay Description Transcriptional activation in COS cells expressing PPAR gamma and RXR alpha				J Med Chem 45: 1518-34 (2002) BindingDB Entry DOI: 10.7270/Q2SJ1JXC
Takeda Chemical Industries, Ltd. Curated by ChEMBL					More data for this Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma/Retinoic acid receptor RXR-alpha (Homo sapiens (Human))	BDBM50111008 (5-{3-[4-(5-Methyl-2-phenyl-thiazol-4-ylmethoxy)-ph...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	PubMed	n/a	n/a	n/a	n/a	813	n/a	n/a	n/a	n/a
Takeda Chemical Industries, Ltd. Curated by ChEMBL					Assay Description Transcriptional activation in COS cells expressing PPAR gamma and RXR alpha				J Med Chem 45: 1518-34 (2002) BindingDB Entry DOI: 10.7270/Q2SJ1JXC
Takeda Chemical Industries, Ltd. Curated by ChEMBL					More data for this Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma/Retinoic acid receptor RXR-alpha (Homo sapiens (Human))	BDBM50111008 (5-{3-[4-(5-Methyl-2-phenyl-thiazol-4-ylmethoxy)-ph...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	PubMed	n/a	n/a	n/a	n/a	269	n/a	n/a	n/a	n/a
Takeda Chemical Industries, Ltd. Curated by ChEMBL					Assay Description Transcriptional activation in COS cells expressing PPAR gamma and RXR alpha				J Med Chem 45: 1518-34 (2002) BindingDB Entry DOI: 10.7270/Q2SJ1JXC
Takeda Chemical Industries, Ltd. Curated by ChEMBL					More data for this Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma/Retinoic acid receptor RXR-alpha (Homo sapiens (Human))	BDBM50111007 (5-{3-[6-(5-Methyl-2-phenyl-oxazol-4-ylmethoxy)-pyr...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	n/a	n/a	16.5	n/a	n/a	n/a	n/a
Takeda Chemical Industries, Ltd. Curated by ChEMBL					Assay Description Transcriptional activation in COS cells expressing PPAR gamma and RXR alpha				J Med Chem 45: 1518-34 (2002) BindingDB Entry DOI: 10.7270/Q2SJ1JXC
Takeda Chemical Industries, Ltd. Curated by ChEMBL					More data for this Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma/Retinoic acid receptor RXR-alpha (Homo sapiens (Human))	BDBM50049240 ((+-)-5-((4-(2-(5-ethyl-2-pyridinyl)ethoxy)phenyl)m...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	PubMed	n/a	n/a	n/a	n/a	490	n/a	n/a	n/a	n/a
Takeda Chemical Industries, Ltd. Curated by ChEMBL					Assay Description Transcriptional activation in COS cells expressing PPAR gamma and RXR alpha; values in the parentheses indicates 95% confidence interval				J Med Chem 45: 1518-34 (2002) BindingDB Entry DOI: 10.7270/Q2SJ1JXC
Takeda Chemical Industries, Ltd. Curated by ChEMBL					More data for this Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma/Retinoic acid receptor RXR-alpha (Homo sapiens (Human))	BDBM50111006 (5-{3-[4-(2-Furan-2-yl-5-methyl-oxazol-4-ylmethoxy)...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	PubMed	n/a	n/a	n/a	n/a	8.87	n/a	n/a	n/a	n/a
Takeda Chemical Industries, Ltd. Curated by ChEMBL					Assay Description Transcriptional activation in COS cells expressing PPAR gamma and RXR alpha				J Med Chem 45: 1518-34 (2002) BindingDB Entry DOI: 10.7270/Q2SJ1JXC
Takeda Chemical Industries, Ltd. Curated by ChEMBL					More data for this Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma/Retinoic acid receptor RXR-alpha (Homo sapiens (Human))	BDBM50111010 (5-{3-[4-(5-Methyl-2-naphthalen-2-yl-oxazol-4-ylmet...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt antibodypedia antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	n/a	n/a	29.3	n/a	n/a	n/a	n/a
Takeda Chemical Industries, Ltd. Curated by ChEMBL					Assay Description Transcriptional activation in COS cells expressing PPAR gamma and RXR alpha				J Med Chem 45: 1518-34 (2002) BindingDB Entry DOI: 10.7270/Q2SJ1JXC
Takeda Chemical Industries, Ltd. Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%