Affinity Data by PubMed id=12014953

PubMed code 12014953

Found 3 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human))	BDBM50113255 (5-[2-(5-Nitro-furan-2-yl)-vinyl]-furan-2-carboxyli...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem	PubMed	n/a	n/a	1.26E+5	n/a	n/a	n/a	n/a	n/a	n/a
Daiichi Pharmaceutical Co., Ltd. Curated by ChEMBL					Assay Description Inhibition of Beta-adrenergic receptor kinase 1				J Med Chem 45: 2150-9 (2002) BindingDB Entry DOI: 10.7270/Q2Q81CCR
Daiichi Pharmaceutical Co., Ltd. Curated by ChEMBL					More data for this Ligand-Target Pair
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human))	BDBM50113256 (2-[5-Amino-3-(3,4-dihydroxy-5-hydroxymethyl-tetrah...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	PubMed	n/a	n/a	5.57E+5	n/a	n/a	n/a	n/a	n/a	n/a
Daiichi Pharmaceutical Co., Ltd. Curated by ChEMBL					Assay Description Inhibition of Beta-adrenergic receptor kinase 1				J Med Chem 45: 2150-9 (2002) BindingDB Entry DOI: 10.7270/Q2Q81CCR
Daiichi Pharmaceutical Co., Ltd. Curated by ChEMBL					More data for this Ligand-Target Pair
Beta-adrenergic receptor kinase 1 (Homo sapiens (Human))	BDBM50113257 (3-tert-Butyl-2-propionyl-2H-indeno[1,2-c]pyrazol-4...) Show SMILES CCC(=O)n1nc2-c3ccccc3C(=O)c2c1C(C)(C)C Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem	PubMed	n/a	n/a	5.63E+5	n/a	n/a	n/a	n/a	n/a	n/a
Daiichi Pharmaceutical Co., Ltd. Curated by ChEMBL					Assay Description Inhibition of Beta-adrenergic receptor kinase 1				J Med Chem 45: 2150-9 (2002) BindingDB Entry DOI: 10.7270/Q2Q81CCR
Daiichi Pharmaceutical Co., Ltd. Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%