Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50117898 (2-(2-Dimethylamino-ethoxy)-fluoren-9-one oxime | C...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Schering Plough Research Institute Curated by ChEMBL | Assay Description In vitro binding affinity for Histamine H3 receptor | Bioorg Med Chem Lett 12: 2643-6 (2002) BindingDB Entry DOI: 10.7270/Q26Q1WMX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50117887 (2-(2-Piperidin-1-yl-ethoxy)-fluoren-9-one oxime | ...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 45 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Schering Plough Research Institute Curated by ChEMBL | Assay Description In vitro binding affinity against Histamine H3 receptor | Bioorg Med Chem Lett 12: 2643-6 (2002) BindingDB Entry DOI: 10.7270/Q26Q1WMX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50117891 (2-(3-Dimethylamino-propoxy)-fluoren-9-one oxime | ...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 48 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Schering Plough Research Institute Curated by ChEMBL | Assay Description In vitro binding affinity for Histamine H3 receptor | Bioorg Med Chem Lett 12: 2643-6 (2002) BindingDB Entry DOI: 10.7270/Q26Q1WMX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50117887 (2-(2-Piperidin-1-yl-ethoxy)-fluoren-9-one oxime | ...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 65 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Schering Plough Research Institute Curated by ChEMBL | Assay Description In vitro binding affinity for Histamine H3 receptor | Bioorg Med Chem Lett 12: 2643-6 (2002) BindingDB Entry DOI: 10.7270/Q26Q1WMX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50117888 (2-(2-Pyrrolidin-1-yl-ethoxy)-fluoren-9-one oxime |...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 65 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Schering Plough Research Institute Curated by ChEMBL | Assay Description In vitro binding affinity for Histamine H3 receptor | Bioorg Med Chem Lett 12: 2643-6 (2002) BindingDB Entry DOI: 10.7270/Q26Q1WMX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50117890 (2-(1-Methyl-azepan-3-yloxy)-fluoren-9-one oxime | ...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 110 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Schering Plough Research Institute Curated by ChEMBL | Assay Description In vitro binding affinity for Histamine H3 receptor | Bioorg Med Chem Lett 12: 2643-6 (2002) BindingDB Entry DOI: 10.7270/Q26Q1WMX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50117889 (2-(2-Piperidin-1-yl-ethoxy)-9H-fluoren-9-ol | CHEM...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 190 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Schering Plough Research Institute Curated by ChEMBL | Assay Description In vitro binding affinity for Histamine H3 receptor | Bioorg Med Chem Lett 12: 2643-6 (2002) BindingDB Entry DOI: 10.7270/Q26Q1WMX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50117897 (2-[2-(1-Methyl-pyrrolidin-2-yl)-ethoxy]-fluoren-9-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 310 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Schering Plough Research Institute Curated by ChEMBL | Assay Description In vitro binding affinity for Histamine H3 receptor | Bioorg Med Chem Lett 12: 2643-6 (2002) BindingDB Entry DOI: 10.7270/Q26Q1WMX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50117893 (2-(2-Morpholin-4-yl-ethoxy)-fluoren-9-one oxime | ...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 325 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Schering Plough Research Institute Curated by ChEMBL | Assay Description In vitro binding affinity for Histamine H3 receptor | Bioorg Med Chem Lett 12: 2643-6 (2002) BindingDB Entry DOI: 10.7270/Q26Q1WMX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50117896 (CHEMBL89623 | [2-(2-Piperidin-1-yl-ethoxy)-9H-fluo...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 570 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Schering Plough Research Institute Curated by ChEMBL | Assay Description In vitro binding affinity for Histamine H3 receptor | Bioorg Med Chem Lett 12: 2643-6 (2002) BindingDB Entry DOI: 10.7270/Q26Q1WMX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50117892 (CHEMBL92558 | Dimethyl-[2-(2-piperidin-1-yl-ethoxy...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 650 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Schering Plough Research Institute Curated by ChEMBL | Assay Description In vitro binding affinity for Histamine H3 receptor | Bioorg Med Chem Lett 12: 2643-6 (2002) BindingDB Entry DOI: 10.7270/Q26Q1WMX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50117894 (2-(1-Methyl-piperidin-3-ylmethoxy)-fluoren-9-one o...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 920 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The Schering Plough Research Institute Curated by ChEMBL | Assay Description In vitro binding affinity for Histamine H3 receptor | Bioorg Med Chem Lett 12: 2643-6 (2002) BindingDB Entry DOI: 10.7270/Q26Q1WMX | |||||||||||
More data for this Ligand-Target Pair |