Affinity Data by PubMed id=12723950

PubMed code 12723950

Found 2 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Adenosine receptor A1 (Homo sapiens (Human))	BDBM50127510 (CHEMBL54461 \| [2-Amino-5-bromo-4-(3-trifluoromethy...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	6.36E+3	n/a	n/a	n/a	n/a
Deakin University Curated by ChEMBL					Assay Description Effective dose as dissociation of [3H]-N6-cyclohexyladenosine ([3H]-CHA) from CHO-K1 membrane after treatment with allosteric enhancer and (R)-PIA				J Med Chem 46: 1870-7 (2003) Article DOI: 10.1021/jm020295m BindingDB Entry DOI: 10.7270/Q2FJ2G5Z
Deakin University Curated by ChEMBL					More data for this Ligand-Target Pair
Adenosine receptor A1 (Homo sapiens (Human))	BDBM50080550 ((2-Amino-4,5-dimethyl-thiophen-3-yl)-(3-trifluorom...) Show SMILES Cc1sc(N)c(C(=O)c2cccc(c2)C(F)(F)F)c1C Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Patents	Article PubMed	n/a	n/a	n/a	n/a	8.40E+3	n/a	n/a	n/a	n/a
Deakin University Curated by ChEMBL					Assay Description Effective dose as dissociation of [3H]-N6-cyclohexyladenosine ([3H]-CHA) from CHO-K1 membrane after treatment with allosteric enhancer and (R)-PIA				J Med Chem 46: 1870-7 (2003) Article DOI: 10.1021/jm020295m BindingDB Entry DOI: 10.7270/Q2FJ2G5Z
Deakin University Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%