Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9606 ((2R,3S,4S,5R)-1,6-bis[(2-fluorophenyl)methoxy]-2,5...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9605 ((2R,3S,4S,5R)-1,6-bis[(2,6-difluorophenyl)methoxy]...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 330 | n/a | n/a | n/a | n/a | n/a | n/a |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9594 ((2R,3S,4S,5R)-2,5-bis(benzyloxy)-1,6-bis[(2,6-difl...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 330 | n/a | n/a | n/a | n/a | n/a | n/a |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9593 ((2R,3S,4S,5R)-2,5-bis(benzyloxy)-1,6-bis[(2-fluoro...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 600 | n/a | n/a | n/a | n/a | n/a | n/a |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9576 ((2R,3S,4S,5R)-1,6-bis(benzyloxy)-2,5-bis[(4-fluoro...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 700 | n/a | n/a | n/a | n/a | 4.7 | 30 |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9604 ((2R,3S,4S,5R)-1,6-bis[(2-fluorophenyl)methoxy]-2,5...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 800 | n/a | n/a | n/a | n/a | n/a | n/a |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9603 ((2R,3S,4S,5R)-2,5-bis(benzyloxy)-1,6-bis({[4-(hydr...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9592 ((2R,3S,4S,5R)-2,5-bis(benzyloxy)-1,6-bis[(3-fluoro...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9574 ((2R,3S,4S,5R)-1,2,5,6-tetrakis[(4-fluorophenyl)met...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.60E+3 | n/a | n/a | n/a | n/a | 4.7 | 30 |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9579 ((2R,3S,4S,5R)-1,6-bis(benzyloxy)-2,5-bis[(3-fluoro...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9577 ((2R,3S,4S,5R)-1,6-bis(benzyloxy)-2,5-bis[(4-chloro...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a | 4.7 | 30 |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9601 (tetra-O-benzyl-d-mannitol deriv. 1ee) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9578 ((2R,3S,4S,5R)-1,6-bis(benzyloxy)-2,5-bis[(4-bromop...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.10E+3 | n/a | n/a | n/a | n/a | 4.7 | 30 |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9571 ((2R,3S,4S,5R)-1,2,5,6-tetrakis(benzyloxy)hexane-3,...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 2.40E+3 | n/a | n/a | n/a | n/a | 4.7 | 30 |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9591 ((2R,3S,4S,5R)-2,5-bis(benzyloxy)-1,6-bis[(4-fluoro...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9582 ((2R,3S,4S,5R)-1,6-bis(benzyloxy)-2,5-bis[(2,4-difl...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9599 ((2R,3S,4S,5R)-2,5-bis(benzyloxy)-1,6-bis[(4-methyl...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9575 (4-({[(2R,3S,4S,5R)-1,5,6-tris[(4-cyanophenyl)metho...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 3.10E+3 | n/a | n/a | n/a | n/a | 4.7 | 30 |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9580 ((2R,3S,4S,5R)-1,6-bis(benzyloxy)-2,5-bis[(2-fluoro...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 3.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9584 ((2R,3S,4S,5R)-1,6-bis(benzyloxy)-2,5-bis[(4-methyl...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9595 ((2R,3S,4S,5R)-2,5-bis(benzyloxy)-1,6-bis[(2,4-difl...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9600 (4-({[(2R,3S,4S,5R)-2,5-bis(benzyloxy)-6-[(4-cyanop...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 4.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9598 ((2R,3S,4S,5R)-2,5-bis(benzyloxy)-1,6-bis({[4-(trif...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9602 (4-({[(2R,3S,4S,5R)-2,5-bis(benzyloxy)-6-[(4-carbox...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9597 ((2R,3S,4S,5R)-2,5-bis(benzyloxy)-1,6-bis[(4-chloro...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9585 (4-({[(2R,3S,4S,5R)-1,6-bis(benzyloxy)-5-[(4-cyanop...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 5.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9573 ((2R,3S,4S,5R)-1,2,5,6-tetrakis({[4-(trifluoromethy...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 6.00E+3 | n/a | n/a | n/a | n/a | 4.7 | 30 |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9596 ((2R,3S,4S,5R)-2,5-bis(benzyloxy)-1,6-bis[(4-bromop...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 6.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9581 ((2R,3S,4S,5R)-1,6-bis(benzyloxy)-2,5-bis[(2,6-difl...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9572 ((2R,3S,4S,5R)-1,2,5,6-tetrakis[(4-methylphenyl)met...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 7.00E+3 | n/a | n/a | n/a | n/a | 4.7 | 30 |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9586 (tetra-O-benzyl-d-mannitol deriv. 1p) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 8.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9588 ((2R,3S,4S,5R)-1,6-bis(benzyloxy)-2,5-bis({[4-(hydr...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9583 ((2R,3S,4S,5R)-1,6-bis(benzyloxy)-2,5-bis({[4-(trif...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9590 (4-({[(2R,3S,4S,5R)-1,6-bis(benzyloxy)-5-[(4-carbam...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9587 (4-({[(2R,3S,4S,5R)-1,6-bis(benzyloxy)-5-[(4-carbox...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9589 ((2R,3S,4S,5R)-2,5-bis({[4-(aminomethyl)phenyl]meth...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9569 ((2R,3S,4S,5R)-2,5-bis(benzyloxy)-1,6-diphenylhexan...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | 4.7 | 30 |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9568 ((2R,3S,4S,5R)-2,5-bis(benzyloxy)-1,6-diphenoxyhexa...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | 4.7 | 30 |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9567 ((2R,3R,4S,5R)-1,2,5,6-tetrakis(benzyloxy)hexane-3,...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | 4.7 | 30 |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9566 ((2R,3S,4S,5S)-1,2,5,6-tetrakis(benzyloxy)hexane-3,...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | 4.7 | 30 |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9565 ((2R,3R,4S,5S)-1,2,5,6-tetrakis(benzyloxy)hexane-3,...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | 4.7 | 30 |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9564 ((2S,3R,4R,5S)-1,2,5,6-tetrakis(benzyloxy)hexane-3,...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | 4.7 | 30 |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dimer of Gag-Pol polyprotein [501-599] (Human immunodeficiency virus type 1) | BDBM9570 ((2R,3S,5S)-1,2,5,6-tetrakis(benzyloxy)hexan-3-ol |...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | 4.7 | 30 |
Pharmacor Inc | Assay Description HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-Ser-Gln-Asn-Tyr-Pr... | Bioorg Med Chem Lett 13: 3601-5 (2003) Article DOI: 10.1016/s0960-894x(03)00677-2 BindingDB Entry DOI: 10.7270/Q27H1GSF | |||||||||||
More data for this Ligand-Target Pair |