Search and Browse
Download
Enter Data
| Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| D(2) dopamine receptor (Homo sapiens (Human)) | BDBM50185473 (4-(3-(4-chlorophenyl)-3-hydroxy-8-aza-bicyclo[3.2....) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet  | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 0.309 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A & M University Curated by ChEMBL | Assay Description Cataleptogenic effect against cloned human Dopamine receptor D2 in male Sprague-Dawley rats in a bar test | Bioorg Med Chem Lett 13: 3779-82 (2003) BindingDB Entry DOI: 10.7270/Q2BK1BQH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| D(2) dopamine receptor (Homo sapiens (Human)) | BDBM50185473 (4-(3-(4-chlorophenyl)-3-hydroxy-8-aza-bicyclo[3.2....) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 0.310 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A & M University Curated by ChEMBL | Assay Description In vitro ability to inhibit the binding of [3H]-spiperone to cloned human Dopamine receptor D2 using apomorphine induced climbing test in male Swiss ... | Bioorg Med Chem Lett 13: 3779-82 (2003) BindingDB Entry DOI: 10.7270/Q2BK1BQH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| D(3) dopamine receptor (Homo sapiens (Human)) | BDBM50185473 (4-(3-(4-chlorophenyl)-3-hydroxy-8-aza-bicyclo[3.2....) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 0.708 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A & M University Curated by ChEMBL | Assay Description Cataleptogenic effect against cloned human Dopamine receptor D3 in male Sprague-Dawley rats in a bar test | Bioorg Med Chem Lett 13: 3779-82 (2003) BindingDB Entry DOI: 10.7270/Q2BK1BQH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| D(3) dopamine receptor (Homo sapiens (Human)) | BDBM50185473 (4-(3-(4-chlorophenyl)-3-hydroxy-8-aza-bicyclo[3.2....) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 0.710 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A & M University Curated by ChEMBL | Assay Description In vitro ability to inhibit the binding of [3H]-7-OH-DPAT to cloned human Dopamine receptor D3 using apomorphine induced climbing test in male Swiss ... | Bioorg Med Chem Lett 13: 3779-82 (2003) BindingDB Entry DOI: 10.7270/Q2BK1BQH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| D(2) dopamine receptor (Homo sapiens (Human)) | BDBM21398 (4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid PDB UniChem Patents Similars | DrugBank PubMed | 0.890 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A & M University Curated by ChEMBL | Assay Description In vitro ability to inhibit the binding of [3H]spiperone to cloned human Dopamine receptor D2 using apomorphine induced climbing test in male Swiss m... | Bioorg Med Chem Lett 13: 3779-82 (2003) BindingDB Entry DOI: 10.7270/Q2BK1BQH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| D(2) dopamine receptor (Homo sapiens (Human)) | BDBM21398 (4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid PDB UniChem Patents Similars | DrugBank PubMed | 0.891 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A & M University Curated by ChEMBL | Assay Description In vitro ability to inhibit the binding of [3H]-spiperone to cloned human Dopamine receptor D2 using apomorphine induced climbing test in male Swiss ... | Bioorg Med Chem Lett 13: 3779-82 (2003) BindingDB Entry DOI: 10.7270/Q2BK1BQH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| D(3) dopamine receptor (Homo sapiens (Human)) | BDBM21398 (4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid PDB UniChem Patents Similars | PubMed | 4.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A & M University Curated by ChEMBL | Assay Description In vitro ability to inhibit the binding of [3H]-7-OH-DPAT to cloned human Dopamine receptor D3 using apomorphine induced climbing test in male Swiss ... | Bioorg Med Chem Lett 13: 3779-82 (2003) BindingDB Entry DOI: 10.7270/Q2BK1BQH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| D(3) dopamine receptor (Homo sapiens (Human)) | BDBM21398 (4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid PDB UniChem Patents Similars | PubMed | 4.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A & M University Curated by ChEMBL | Assay Description Cataleptogenic effect against cloned human Dopamine receptor D3 in male Sprague-Dawley rats in a bar test | Bioorg Med Chem Lett 13: 3779-82 (2003) BindingDB Entry DOI: 10.7270/Q2BK1BQH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| D(4) dopamine receptor (Homo sapiens (Human)) | BDBM21398 (4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid PDB UniChem Patents Similars | PubMed | 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A & M University Curated by ChEMBL | Assay Description In vitro ability to inhibit the binding of [3H]-spiperone to cloned human dopamine receptor D4 using apomorphine induced climbing test in male Swiss ... | Bioorg Med Chem Lett 13: 3779-82 (2003) BindingDB Entry DOI: 10.7270/Q2BK1BQH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| D(4) dopamine receptor (Homo sapiens (Human)) | BDBM21398 (4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid PDB UniChem Patents Similars | PubMed | 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A & M University Curated by ChEMBL | Assay Description Cataleptogenic effect against cloned human dopamine receptor D4 in male Sprague-Dawley rats in a bar test | Bioorg Med Chem Lett 13: 3779-82 (2003) BindingDB Entry DOI: 10.7270/Q2BK1BQH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| D(4) dopamine receptor (Homo sapiens (Human)) | BDBM50185473 (4-(3-(4-chlorophenyl)-3-hydroxy-8-aza-bicyclo[3.2....) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 12 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A & M University Curated by ChEMBL | Assay Description In vitro ability to inhibit the binding of [3H]-spiperone to cloned human dopamine receptor D4 using apomorphine induced climbing test in male Swiss ... | Bioorg Med Chem Lett 13: 3779-82 (2003) BindingDB Entry DOI: 10.7270/Q2BK1BQH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| D(4) dopamine receptor (Homo sapiens (Human)) | BDBM50185473 (4-(3-(4-chlorophenyl)-3-hydroxy-8-aza-bicyclo[3.2....) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 12 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A & M University Curated by ChEMBL | Assay Description Cataleptogenic effect against cloned human dopamine receptor D4 in male Sprague-Dawley rats in a bar test | Bioorg Med Chem Lett 13: 3779-82 (2003) BindingDB Entry DOI: 10.7270/Q2BK1BQH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| D(4) dopamine receptor (Homo sapiens (Human)) | BDBM50001884 (2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid UniChem Patents Similars | DrugBank PubMed | 54 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A & M University Curated by ChEMBL | Assay Description In vitro ability to inhibit the binding of [3H]-spiperone to cloned human dopamine receptor D4 using apomorphine induced climbing test in male Swiss ... | Bioorg Med Chem Lett 13: 3779-82 (2003) BindingDB Entry DOI: 10.7270/Q2BK1BQH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| D(4) dopamine receptor (Homo sapiens (Human)) | BDBM50001884 (2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid UniChem Patents Similars | DrugBank PubMed | 54 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A & M University Curated by ChEMBL | Assay Description In vitro ability to inhibit the binding of [3H]spiperone to cloned human dopamine receptor D4 using apomorphine induced climbing test in male Swiss m... | Bioorg Med Chem Lett 13: 3779-82 (2003) BindingDB Entry DOI: 10.7270/Q2BK1BQH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| D(2) dopamine receptor (Homo sapiens (Human)) | BDBM50001884 (2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid UniChem Patents Similars | DrugBank PubMed | 130 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A & M University Curated by ChEMBL | Assay Description In vitro ability to inhibit the binding of [3H]-spiperone to cloned human Dopamine receptor D2 using apomorphine induced climbing test in male Swiss ... | Bioorg Med Chem Lett 13: 3779-82 (2003) BindingDB Entry DOI: 10.7270/Q2BK1BQH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| D(2) dopamine receptor (Homo sapiens (Human)) | BDBM50001884 (2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid UniChem Patents Similars | DrugBank PubMed | 135 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A & M University Curated by ChEMBL | Assay Description Cataleptogenic effect against cloned human Dopamine receptor D2 in male Sprague-Dawley rats in a bar test | Bioorg Med Chem Lett 13: 3779-82 (2003) BindingDB Entry DOI: 10.7270/Q2BK1BQH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| D(3) dopamine receptor (Homo sapiens (Human)) | BDBM50001884 (2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid UniChem Patents Similars | PubMed | 240 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A & M University Curated by ChEMBL | Assay Description Cataleptogenic effect against cloned human Dopamine receptor D3 in male Sprague-Dawley rats in a bar test | Bioorg Med Chem Lett 13: 3779-82 (2003) BindingDB Entry DOI: 10.7270/Q2BK1BQH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| D(3) dopamine receptor (Homo sapiens (Human)) | BDBM50001884 (2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid UniChem Patents Similars | PubMed | 240 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Florida A & M University Curated by ChEMBL | Assay Description In vitro ability to inhibit the binding of [3H]-7-OH-DPAT to cloned human Dopamine receptor D3 using apomorphine induced climbing test in male Swiss ... | Bioorg Med Chem Lett 13: 3779-82 (2003) BindingDB Entry DOI: 10.7270/Q2BK1BQH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
