Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
ATP-dependent translocase ABCB1 (Homo sapiens (Human)) | BDBM50420188 (COELENTERAZINE) | PDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 147 | n/a | n/a | n/a | n/a |
Washington University School of Medicine Curated by ChEMBL | Assay Description TP_TRANSPORTER: efflux in KB 8-5-11 Rluc cells | Proc Natl Acad Sci USA 101: 1702-7 (2004) Article DOI: 10.1073/pnas.0304326101 BindingDB Entry DOI: 10.7270/Q22R3SXK | |||||||||||
More data for this Ligand-Target Pair |