Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146108 (Arg-Arg-Pro-Hyp-Gly-Thi-Cys-Tic-Oic-Arg | CHEMBL27...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.0900 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 0.06 nM to bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146111 (CHEMBL542173 | N-(4-{(E)-2-[({[2,4-Dichloro-3-(4-d...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.470 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 1 nM to human bradykinin receptor B2 expressed in CHO cells by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146108 (Arg-Arg-Pro-Hyp-Gly-Thi-Cys-Tic-Oic-Arg | CHEMBL27...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.490 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 1 nM to human bradykinin receptor B2 expressed in CHO cells by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067281 (4-{(E)-2-[({[2,4-Dichloro-3-(2-methyl-quinolin-8-y...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.510 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 0.06 nM to bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146120 (4-{(E)-2-[({[2,4-Dichloro-3-(2-methyl-4-piperidin-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.520 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 1 nM to human bradykinin receptor B2 expressed in CHO cells by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146102 (4-{(E)-2-[({[2,4-Dichloro-3-(2-methyl-4-morpholin-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.640 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 1 nM to human bradykinin receptor B2 expressed in CHO cells by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146101 (4-{(E)-2-[({[2,4-Dichloro-3-(4-dimethylamino-2-met...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.700 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 1 nM to human bradykinin receptor B2 expressed in CHO cells by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146109 (4-{(E)-2-[({[2,4-Dichloro-3-(2-methyl-4-piperidin-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.760 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 1 nM to human bradykinin receptor B2 expressed in CHO cells by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146119 (4-{(E)-2-[({[2,4-Dichloro-3-(2-methyl-4-morpholin-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.880 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 1 nM to human bradykinin receptor B2 expressed in CHO cells by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146104 (CHEMBL545021 | N-(4-{(E)-2-[({[2,4-Dichloro-3-(2-m...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 1 nM to human bradykinin receptor B2 expressed in CHO cells by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067281 (4-{(E)-2-[({[2,4-Dichloro-3-(2-methyl-quinolin-8-y...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.10 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 1 nM to human bradykinin receptor B2 expressed in CHO cells by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146097 (4-{(E)-2-[({[2,4-Dichloro-3-(2-methyl-4-piperidin-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.10 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 1 nM to human bradykinin receptor B2 expressed in CHO cells by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146115 (5-{(E)-2-[({[2,4-Dichloro-3-(2-methyl-4-morpholin-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.10 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 1 nM to human bradykinin receptor B2 expressed in CHO cells by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146106 (5-{(E)-2-[({[2,4-Dichloro-3-(4-dimethylamino-2-met...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 0.06 nM to bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146121 ((E)-N-({[2,4-Dichloro-3-(2-methyl-4-piperidin-1-yl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 1 nM to human bradykinin receptor B2 expressed in CHO cells by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146106 (5-{(E)-2-[({[2,4-Dichloro-3-(4-dimethylamino-2-met...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.60 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 1 nM to human bradykinin receptor B2 expressed in CHO cells by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146114 (CHEMBL539792 | N-(4-{(E)-2-[({[2,4-Dichloro-3-(2-m...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.60 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 1 nM to human bradykinin receptor B2 expressed in CHO cells by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146098 ((E)-N-({[2,4-Dichloro-3-(2-methyl-4-morpholin-4-yl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.80 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 1 nM to human bradykinin receptor B2 expressed in CHO cells by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146110 ((E)-3-(6-Acetylamino-pyridin-3-yl)-N-({[2,4-dichlo...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.80 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 1 nM to human bradykinin receptor B2 expressed in CHO cells by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50142950 (4-{(E)-2-[({[2,4-Dichloro-3-(4-dimethylamino-2-met...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.80 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 0.06 nM to bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146124 (4-{(E)-2-[({[2,4-Dichloro-3-(4-dimethylamino-2-met...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 1 nM to human bradykinin receptor B2 expressed in CHO cells by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50142945 (4-{(E)-2-[({[2,4-Dichloro-3-(4-dimethylamino-2-met...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.10 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 1 nM to human bradykinin receptor B2 expressed in CHO cells by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146113 (3-[3-({[2,4-Dichloro-3-(4-dimethylamino-2-methyl-q...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 1 nM to human bradykinin receptor B2 expressed in CHO cells by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146117 (4-{(E)-2-[({[2,4-Dichloro-3-(2-methyl-4-piperidin-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 1 nM to human bradykinin receptor B2 expressed in CHO cells by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146122 (4-{(E)-2-[({[2,4-Dichloro-3-(2-methyl-4-morpholin-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.70 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 1 nM to human bradykinin receptor B2 expressed in CHO cells by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50142945 (4-{(E)-2-[({[2,4-Dichloro-3-(4-dimethylamino-2-met...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.90 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 0.06 nM to bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50142950 (4-{(E)-2-[({[2,4-Dichloro-3-(4-dimethylamino-2-met...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 1 nM to human bradykinin receptor B2 expressed in CHO cells by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146112 (5-{(E)-2-[({[2,4-Dichloro-3-(4-dimethylamino-2-met...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 1 nM to human bradykinin receptor B2 expressed in CHO cells by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146116 ((E)-3-(6-Acetylamino-pyridin-3-yl)-N-({[2,4-dichlo...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 1 nM to human bradykinin receptor B2 expressed in CHO cells by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146099 ((E)-3-(4-Acetylamino-3-methyl-phenyl)-N-({[2,4-dic...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.80 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 1 nM to human bradykinin receptor B2 expressed in CHO cells by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146101 (4-{(E)-2-[({[2,4-Dichloro-3-(4-dimethylamino-2-met...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.10 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 0.06 nM to bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146124 (4-{(E)-2-[({[2,4-Dichloro-3-(4-dimethylamino-2-met...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.60 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 0.06 nM to bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146100 (4-{(E)-2-[({[2,4-Dichloro-3-(4-dimethylamino-2-met...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.90 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 1 nM to human bradykinin receptor B2 expressed in CHO cells by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146116 ((E)-3-(6-Acetylamino-pyridin-3-yl)-N-({[2,4-dichlo...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 0.06 nM to bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146111 (CHEMBL542173 | N-(4-{(E)-2-[({[2,4-Dichloro-3-(4-d...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.90 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 0.06 nM to bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146112 (5-{(E)-2-[({[2,4-Dichloro-3-(4-dimethylamino-2-met...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8.10 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 0.06 nM to bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146122 (4-{(E)-2-[({[2,4-Dichloro-3-(2-methyl-4-morpholin-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 0.06 nM to bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146113 (3-[3-({[2,4-Dichloro-3-(4-dimethylamino-2-methyl-q...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 0.06 nM to bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146098 ((E)-N-({[2,4-Dichloro-3-(2-methyl-4-morpholin-4-yl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 13 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 0.06 nM to bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146123 (4-[(E)-2-({[(3-{4-[Bis-(2-methoxy-ethyl)-amino]-2-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 19 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 1 nM to human bradykinin receptor B2 expressed in CHO cells by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146099 ((E)-3-(4-Acetylamino-3-methyl-phenyl)-N-({[2,4-dic...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 21 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 0.06 nM to bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146100 (4-{(E)-2-[({[2,4-Dichloro-3-(4-dimethylamino-2-met...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 28 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 0.06 nM to bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146121 ((E)-N-({[2,4-Dichloro-3-(2-methyl-4-piperidin-1-yl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 28 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 0.06 nM to bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146104 (CHEMBL545021 | N-(4-{(E)-2-[({[2,4-Dichloro-3-(2-m...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 29 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 0.06 nM to bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146109 (4-{(E)-2-[({[2,4-Dichloro-3-(2-methyl-4-piperidin-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 0.06 nM to bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146096 (4-{(E)-2-[({[3-(4-Azepan-1-yl-2-methyl-quinolin-8-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 37 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 1 nM to human bradykinin receptor B2 expressed in CHO cells by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146102 (4-{(E)-2-[({[2,4-Dichloro-3-(2-methyl-4-morpholin-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 37 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 0.06 nM to bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146117 (4-{(E)-2-[({[2,4-Dichloro-3-(2-methyl-4-piperidin-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 0.06 nM to bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146105 (4-((E)-2-{[({2,4-Dichloro-3-[4-(2-methoxy-ethylami...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 41 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 1 nM to human bradykinin receptor B2 expressed in CHO cells by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146119 (4-{(E)-2-[({[2,4-Dichloro-3-(2-methyl-4-morpholin-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 43 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 0.06 nM to bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146105 (4-((E)-2-{[({2,4-Dichloro-3-[4-(2-methoxy-ethylami...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 49 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 0.06 nM to bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146110 ((E)-3-(6-Acetylamino-pyridin-3-yl)-N-({[2,4-dichlo...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 65 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 0.06 nM to bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146097 (4-{(E)-2-[({[2,4-Dichloro-3-(2-methyl-4-piperidin-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 68 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 0.06 nM to bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146114 (CHEMBL539792 | N-(4-{(E)-2-[({[2,4-Dichloro-3-(2-m...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 75 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 0.06 nM to bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146115 (5-{(E)-2-[({[2,4-Dichloro-3-(2-methyl-4-morpholin-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 85 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 0.06 nM to bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146103 (4-{(E)-2-[({[2,4-Dichloro-3-(2-methyl-4-pyrrolidin...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 87 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 1 nM to human bradykinin receptor B2 expressed in CHO cells by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146107 (4-((E)-2-{[({2,4-Dichloro-3-[2-methyl-4-(4-methyl-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 98 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 1 nM to human bradykinin receptor B2 expressed in CHO cells by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146120 (4-{(E)-2-[({[2,4-Dichloro-3-(2-methyl-4-piperidin-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 240 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 0.06 nM to bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146123 (4-[(E)-2-({[(3-{4-[Bis-(2-methoxy-ethyl)-amino]-2-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 560 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 0.06 nM to bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146096 (4-{(E)-2-[({[3-(4-Azepan-1-yl-2-methyl-quinolin-8-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 840 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 0.06 nM to bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146107 (4-((E)-2-{[({2,4-Dichloro-3-[2-methyl-4-(4-methyl-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 0.06 nM to bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146118 (4-((E)-2-{[({2,4-Dichloro-3-[4-(2-dimethylamino-et...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 0.06 nM to bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146103 (4-{(E)-2-[({[2,4-Dichloro-3-(2-methyl-4-pyrrolidin...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 0.06 nM to bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50146118 (4-((E)-2-{[({2,4-Dichloro-3-[4-(2-dimethylamino-et...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Co Ltd Curated by ChEMBL | Assay Description Inhibition of specific binding of [3H]BK at 1 nM to human bradykinin receptor B2 expressed in CHO cells by 50%. | J Med Chem 47: 2667-77 (2004) Article DOI: 10.1021/jm030326t BindingDB Entry DOI: 10.7270/Q2B27W2Q | |||||||||||
More data for this Ligand-Target Pair |