Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50150842 (4-[((R)-N-Cyclohexyl-3-methyl-piperazine-1-carboxi...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cells | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50150835 (4-[N''-(2-Amino-2-methyl-propyl)-N''''-cyclohexyl-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 5.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cells | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50150837 (4-[((S)-N-(R)-Cyclohexyl-2,5-dimethyl-piperazine-1...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 5.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cells | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50150829 (4-[(N-Cyclohexyl-3,5-dimethyl-piperazine-1-carboxi...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 11 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cells | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50150830 (4-[(N-Cyclohexyl-piperazine-1-carboximidoyl)-amino...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 18 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cells | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50150833 (4-[((S)-N-Cyclohexyl-3-methyl-piperazine-1-carboxi...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 21 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cells | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50150836 (4-(N''-Cyclohexyl-N''''-pyrrolidin-3-yl-guanidino)...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 26 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cells | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50150831 (4-[(N-Cyclohexyl-3-methylamino-pyrrolidine-1-carbo...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 36 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cells | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50150840 (4-[(4-Benzyl-N-cyclohexyl-piperazine-1-carboximido...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 44 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cells | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50150834 (4-[(N-Cyclohexyl-4-methyl-piperazine-1-carboximido...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 50 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cells | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50150849 (4-[N''-Cyclohexyl-N''''-(3,5-difluoro-benzyl)-guan...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cells | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50150845 (4-[(N-Cyclohexyl-4-pyrrolidin-1-yl-piperidine-1-ca...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 77 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cells | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50150847 (CHEMBL184612 | N-[2-(2,4-Dichloro-phenyl)-ethyl]-4...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 91 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cells | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50150839 (4-[(N-Cyclohexyl-3,5-dimethyl-piperidine-1-carboxi...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 144 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cells | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50150832 (4-[(4-Amino-N-cyclohexyl-piperidine-1-carboximidoy...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 230 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cells | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50150838 (4-[(N-Cyclohexyl-4-phenyl-piperazine-1-carboximido...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 290 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cells | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50150844 (4-[(N-Cyclohexyl-4-pyrimidin-2-yl-piperazine-1-car...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 305 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cells | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50150850 (4-[(N-Cyclohexyl-2,6-dimethyl-morpholine-4-carboxi...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 350 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cells | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50150843 (4-(N''''-Cyclohexyl-N'',N''-dipropyl-guanidino)-N-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 360 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cells | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM50150837 (4-[((S)-N-(R)-Cyclohexyl-2,5-dimethyl-piperazine-1...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 360 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Binding affinity for human melanocortin 1 receptor | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM50150830 (4-[(N-Cyclohexyl-piperazine-1-carboximidoyl)-amino...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 400 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Binding affinity for human melanocortin 1 receptor | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50150848 (4-[(N-Cyclohexyl-3-oxo-piperazine-1-carboximidoyl)...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 560 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cells | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50150833 (4-[((S)-N-Cyclohexyl-3-methyl-piperazine-1-carboxi...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 580 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Binding affinity for human melanocortin 4 receptor | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50150829 (4-[(N-Cyclohexyl-3,5-dimethyl-piperazine-1-carboxi...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 590 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Binding affinity for human melanocortin 4 receptor | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50150830 (4-[(N-Cyclohexyl-piperazine-1-carboximidoyl)-amino...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 650 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Binding affinity for human melanocortin 4 receptor | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50150842 (4-[((R)-N-Cyclohexyl-3-methyl-piperazine-1-carboxi...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 840 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Binding affinity for human melanocortin 4 receptor | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50150837 (4-[((S)-N-(R)-Cyclohexyl-2,5-dimethyl-piperazine-1...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 840 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Binding affinity for human melanocortin 4 receptor | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50150841 (4-[(N-Cyclohexyl-2-methyl-3-oxo-piperazine-1-carbo...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.05E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cells | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50150835 (4-[N''-(2-Amino-2-methyl-propyl)-N''''-cyclohexyl-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Binding affinity for human melanocortin 4 receptor | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50150831 (4-[(N-Cyclohexyl-3-methylamino-pyrrolidine-1-carbo...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Binding affinity for human melanocortin 4 receptor | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50150836 (4-(N''-Cyclohexyl-N''''-pyrrolidin-3-yl-guanidino)...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Binding affinity for human melanocortin 4 receptor | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50150846 (4-{[N-Cyclohexyl-4-(2,5-dimethyl-phenyl)-piperazin...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.76E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Inhibition of [125I]-NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK-293 cells | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM50150836 (4-(N''-Cyclohexyl-N''''-pyrrolidin-3-yl-guanidino)...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Binding affinity for human melanocortin 1 receptor | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 3 (Homo sapiens (Human)) | BDBM50150830 (4-[(N-Cyclohexyl-piperazine-1-carboximidoyl)-amino...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Binding affinity for human melanocortin 3 receptor | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 3 (Homo sapiens (Human)) | BDBM50150831 (4-[(N-Cyclohexyl-3-methylamino-pyrrolidine-1-carbo...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Binding affinity for human melanocortin 3 receptor | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 3 (Homo sapiens (Human)) | BDBM50150835 (4-[N''-(2-Amino-2-methyl-propyl)-N''''-cyclohexyl-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Binding affinity for human melanocortin 3 receptor | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 3 (Homo sapiens (Human)) | BDBM50150836 (4-(N''-Cyclohexyl-N''''-pyrrolidin-3-yl-guanidino)...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Binding affinity for human melanocortin 3 receptor | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 3 (Homo sapiens (Human)) | BDBM50150837 (4-[((S)-N-(R)-Cyclohexyl-2,5-dimethyl-piperazine-1...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Binding affinity for human melanocortin 3 receptor | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 3 (Homo sapiens (Human)) | BDBM50150833 (4-[((S)-N-Cyclohexyl-3-methyl-piperazine-1-carboxi...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Binding affinity for human melanocortin 3 receptor | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 3 (Homo sapiens (Human)) | BDBM50150842 (4-[((R)-N-Cyclohexyl-3-methyl-piperazine-1-carboxi...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Binding affinity for human melanocortin 3 receptor | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 3 (Homo sapiens (Human)) | BDBM50150829 (4-[(N-Cyclohexyl-3,5-dimethyl-piperazine-1-carboxi...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 3.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Binding affinity for human melanocortin 3 receptor | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50150842 (4-[((R)-N-Cyclohexyl-3-methyl-piperazine-1-carboxi...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 70 | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Inhibition of human Melanocortin 5 receptor | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50150829 (4-[(N-Cyclohexyl-3,5-dimethyl-piperazine-1-carboxi...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 80 | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Inhibition of [125I]NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK293 cells | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50150837 (4-[((S)-N-(R)-Cyclohexyl-2,5-dimethyl-piperazine-1...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 380 | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Inhibition of human Melanocortin 5 receptor | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50150833 (4-[((S)-N-Cyclohexyl-3-methyl-piperazine-1-carboxi...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 380 | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Inhibition of [125I]NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK293 cells | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50150830 (4-[(N-Cyclohexyl-piperazine-1-carboximidoyl)-amino...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 460 | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Inhibition of [125I]NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK293 cells | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50150835 (4-[N''-(2-Amino-2-methyl-propyl)-N''''-cyclohexyl-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 530 | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Inhibition of [125I]NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK293 cells | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50150836 (4-(N''-Cyclohexyl-N''''-pyrrolidin-3-yl-guanidino)...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 530 | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Inhibition of [125I]NDP-MSH binding to human Melanocortin 5 receptor expressed in HEK293 cells | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50150831 (4-[(N-Cyclohexyl-3-methylamino-pyrrolidine-1-carbo...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 630 | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Inhibition of human Melanocortin 5 receptor | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50150835 (4-[N''-(2-Amino-2-methyl-propyl)-N''''-cyclohexyl-...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.90E+3 | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Binding affinity for human melanocortin 4 receptor | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50150831 (4-[(N-Cyclohexyl-3-methylamino-pyrrolidine-1-carbo...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 4.60E+3 | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Agonistic activity for human Melanocortin 4 receptor as stimulated cAMP release | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50150842 (4-[((R)-N-Cyclohexyl-3-methyl-piperazine-1-carboxi...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.70E+3 | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Binding affinity for human melanocortin 4 receptor | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50150829 (4-[(N-Cyclohexyl-3,5-dimethyl-piperazine-1-carboxi...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 4.00E+3 | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Binding affinity for human melanocortin 4 receptor | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50150830 (4-[(N-Cyclohexyl-piperazine-1-carboximidoyl)-amino...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.90E+3 | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Agonistic activity for human Melanocortin 4 receptor as stimulated cAMP release | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50150833 (4-[((S)-N-Cyclohexyl-3-methyl-piperazine-1-carboxi...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.80E+3 | n/a | n/a | n/a | n/a |
Neurocrine Biosciences, Inc. Curated by ChEMBL | Assay Description Binding affinity for human melanocortin 4 receptor | J Med Chem 47: 4083-8 (2004) Article DOI: 10.1021/jm0400496 BindingDB Entry DOI: 10.7270/Q2JH3KM0 | |||||||||||
More data for this Ligand-Target Pair |