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PubMed code 15771417

Compile data set for download or QSAR
Found 48 hits of Enzyme Inhibition Constant Data   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Vascular endothelial growth factor receptor 2


(Homo sapiens (Human))		BDBM50162972
PNG
(4-(Benzothiazol-6-ylamino)-6-(benzyl-isopropyl-ami...)
Show SMILES CC(C)N(Cc1ccccc1)c1nc(Nc2ccc3ncsc3c2)[nH]c(=O)n1
Show InChI InChI=1S/C20H20N6OS/c1-13(2)26(11-14-6-4-3-5-7-14)19-23-18(24-20(27)25-19)22-15-8-9-16-17(10-15)28-12-21-16/h3-10,12-13H,11H2,1-2H3,(H2,22,23,24,25,27)
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n/an/a 18n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
In vitro inhibition of Vascular endothelial growth factor receptor 2 at 10 uM ATP

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Vascular endothelial growth factor receptor 2


(Homo sapiens (Human))		BDBM50162976
PNG
(4-(Benzothiazol-6-ylamino)-6-(1-methyl-1-phenyl-et...)
Show SMILES CC(C)(Nc1nc(Nc2ccc3ncsc3c2)[nH]c(=O)n1)c1ccccc1
Show InChI InChI=1S/C19H18N6OS/c1-19(2,12-6-4-3-5-7-12)25-17-22-16(23-18(26)24-17)21-13-8-9-14-15(10-13)27-11-20-14/h3-11H,1-2H3,(H3,21,22,23,24,25,26)
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n/an/a 35n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
In vitro inhibition of Vascular endothelial growth factor receptor 2 at 10 uM ATP

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Vascular endothelial growth factor receptor 2


(Homo sapiens (Human))		BDBM50162973
PNG
(CHEMBL177298 | N-[4-(Benzothiazol-6-ylamino)-6-(1-...)
Show SMILES CC(C)(Nc1nc(NO)nc(Nc2ccc3ncsc3c2)n1)c1ccccc1
Show InChI InChI=1S/C19H19N7OS/c1-19(2,12-6-4-3-5-7-12)25-17-22-16(23-18(24-17)26-27)21-13-8-9-14-15(10-13)28-11-20-14/h3-11,27H,1-2H3,(H3,21,22,23,24,25,26)
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n/an/a 40n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
In vitro inhibition of Vascular endothelial growth factor receptor 2 at 10 uM ATP

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Vascular endothelial growth factor receptor 2


(Homo sapiens (Human))		BDBM50162973
PNG
(CHEMBL177298 | N-[4-(Benzothiazol-6-ylamino)-6-(1-...)
Show SMILES CC(C)(Nc1nc(NO)nc(Nc2ccc3ncsc3c2)n1)c1ccccc1
Show InChI InChI=1S/C19H19N7OS/c1-19(2,12-6-4-3-5-7-12)25-17-22-16(23-18(24-17)26-27)21-13-8-9-14-15(10-13)28-11-20-14/h3-11,27H,1-2H3,(H3,21,22,23,24,25,26)
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n/an/a 40n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
In vitro inhibition of Vascular endothelial growth factor receptor 2 at 10 uM ATP

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Vascular endothelial growth factor receptor 2


(Homo sapiens (Human))		BDBM50162978
PNG
(4-(Benzothiazol-6-ylamino)-6-(benzyl-ethyl-amino)-...)
Show SMILES CCN(Cc1ccccc1)c1nc(Nc2ccc3ncsc3c2)[nH]c(=O)n1
Show InChI InChI=1S/C19H18N6OS/c1-2-25(11-13-6-4-3-5-7-13)18-22-17(23-19(26)24-18)21-14-8-9-15-16(10-14)27-12-20-15/h3-10,12H,2,11H2,1H3,(H2,21,22,23,24,26)
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n/an/a 49n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
In vitro inhibition of Vascular endothelial growth factor receptor 2 at 10 uM ATP

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Angiopoietin-1 receptor


(Homo sapiens (Human))		BDBM50162972
PNG
(4-(Benzothiazol-6-ylamino)-6-(benzyl-isopropyl-ami...)
Show SMILES CC(C)N(Cc1ccccc1)c1nc(Nc2ccc3ncsc3c2)[nH]c(=O)n1
Show InChI InChI=1S/C20H20N6OS/c1-13(2)26(11-14-6-4-3-5-7-14)19-23-18(24-20(27)25-19)22-15-8-9-16-17(10-15)28-12-21-16/h3-10,12-13H,11H2,1-2H3,(H2,22,23,24,25,27)
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n/an/a 180n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
Inhibition of tyrosine protein kinase receptor TIE-2

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Vascular endothelial growth factor receptor 2


(Homo sapiens (Human))		BDBM50162975
PNG
(4-(3H-Benzoimidazol-5-ylamino)-6-(1-methyl-1-pheny...)
Show SMILES CC(C)(Nc1nc(Nc2ccc3nc[nH]c3c2)[nH]c(=O)n1)c1ccccc1
Show InChI InChI=1S/C19H19N7O/c1-19(2,12-6-4-3-5-7-12)26-17-23-16(24-18(27)25-17)22-13-8-9-14-15(10-13)21-11-20-14/h3-11H,1-2H3,(H,20,21)(H3,22,23,24,25,26,27)
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n/an/a 240n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
In vitro inhibition of Vascular endothelial growth factor receptor 2 at 10 uM ATP

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Vascular endothelial growth factor receptor 2


(Homo sapiens (Human))		BDBM50162972
PNG
(4-(Benzothiazol-6-ylamino)-6-(benzyl-isopropyl-ami...)
Show SMILES CC(C)N(Cc1ccccc1)c1nc(Nc2ccc3ncsc3c2)[nH]c(=O)n1
Show InChI InChI=1S/C20H20N6OS/c1-13(2)26(11-14-6-4-3-5-7-14)19-23-18(24-20(27)25-19)22-15-8-9-16-17(10-15)28-12-21-16/h3-10,12-13H,11H2,1-2H3,(H2,22,23,24,25,27)
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n/an/a 280n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
Inhibition of KDR-induced MAP kinase autophosphorylation assay in HUVEC cells

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Vascular endothelial growth factor receptor 2


(Homo sapiens (Human))		BDBM50162974
PNG
(4-(Benzothiazol-5-ylamino)-6-(benzyl-methyl-amino)...)
Show SMILES CN(Cc1ccccc1)c1nc(Nc2ccc3scnc3c2)[nH]c(=O)n1
Show InChI InChI=1S/C18H16N6OS/c1-24(10-12-5-3-2-4-6-12)17-21-16(22-18(25)23-17)20-13-7-8-15-14(9-13)19-11-26-15/h2-9,11H,10H2,1H3,(H2,20,21,22,23,25)
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n/an/a 320n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
In vitro inhibition of Vascular endothelial growth factor receptor 2 at 10 uM ATP

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Vascular endothelial growth factor receptor 2


(Homo sapiens (Human))		BDBM50162974
PNG
(4-(Benzothiazol-5-ylamino)-6-(benzyl-methyl-amino)...)
Show SMILES CN(Cc1ccccc1)c1nc(Nc2ccc3scnc3c2)[nH]c(=O)n1
Show InChI InChI=1S/C18H16N6OS/c1-24(10-12-5-3-2-4-6-12)17-21-16(22-18(25)23-17)20-13-7-8-15-14(9-13)19-11-26-15/h2-9,11H,10H2,1H3,(H2,20,21,22,23,25)
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n/an/a 320n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
In vitro inhibition of Vascular endothelial growth factor receptor 2 at 10 uM ATP

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Angiopoietin-1 receptor


(Homo sapiens (Human))		BDBM50162978
PNG
(4-(Benzothiazol-6-ylamino)-6-(benzyl-ethyl-amino)-...)
Show SMILES CCN(Cc1ccccc1)c1nc(Nc2ccc3ncsc3c2)[nH]c(=O)n1
Show InChI InChI=1S/C19H18N6OS/c1-2-25(11-13-6-4-3-5-7-13)18-22-17(23-19(26)24-18)21-14-8-9-15-16(10-14)27-12-20-15/h3-10,12H,2,11H2,1H3,(H2,21,22,23,24,26)
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n/an/a 400n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
Inhibition of tyrosine protein kinase receptor TIE-2

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Vascular endothelial growth factor receptor 2


(Homo sapiens (Human))		BDBM50162976
PNG
(4-(Benzothiazol-6-ylamino)-6-(1-methyl-1-phenyl-et...)
Show SMILES CC(C)(Nc1nc(Nc2ccc3ncsc3c2)[nH]c(=O)n1)c1ccccc1
Show InChI InChI=1S/C19H18N6OS/c1-19(2,12-6-4-3-5-7-12)25-17-22-16(23-18(26)24-17)21-13-8-9-14-15(10-13)27-11-20-14/h3-11H,1-2H3,(H3,21,22,23,24,25,26)
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n/an/a 400n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
Inhibition of KDR-induced MAP kinase autophosphorylation assay in HUVEC cells

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Insulin receptor


(Homo sapiens (Human))		BDBM50162973
PNG
(CHEMBL177298 | N-[4-(Benzothiazol-6-ylamino)-6-(1-...)
Show SMILES CC(C)(Nc1nc(NO)nc(Nc2ccc3ncsc3c2)n1)c1ccccc1
Show InChI InChI=1S/C19H19N7OS/c1-19(2,12-6-4-3-5-7-12)25-17-22-16(23-18(24-17)26-27)21-13-8-9-14-15(10-13)28-11-20-14/h3-11,27H,1-2H3,(H3,21,22,23,24,25,26)
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n/an/a 420n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
Inhibition of beta IRK tyrosine kinase

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Insulin receptor


(Homo sapiens (Human))		BDBM50162976
PNG
(4-(Benzothiazol-6-ylamino)-6-(1-methyl-1-phenyl-et...)
Show SMILES CC(C)(Nc1nc(Nc2ccc3ncsc3c2)[nH]c(=O)n1)c1ccccc1
Show InChI InChI=1S/C19H18N6OS/c1-19(2,12-6-4-3-5-7-12)25-17-22-16(23-18(26)24-17)21-13-8-9-14-15(10-13)27-11-20-14/h3-11H,1-2H3,(H3,21,22,23,24,25,26)
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n/an/a 550n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
Inhibition of beta IRK tyrosine kinase

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Vascular endothelial growth factor receptor 2


(Homo sapiens (Human))		BDBM50162978
PNG
(4-(Benzothiazol-6-ylamino)-6-(benzyl-ethyl-amino)-...)
Show SMILES CCN(Cc1ccccc1)c1nc(Nc2ccc3ncsc3c2)[nH]c(=O)n1
Show InChI InChI=1S/C19H18N6OS/c1-2-25(11-13-6-4-3-5-7-13)18-22-17(23-19(26)24-18)21-14-8-9-15-16(10-14)27-12-20-15/h3-10,12H,2,11H2,1H3,(H2,21,22,23,24,26)
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n/an/a 600n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
Inhibition of KDR-induced MAP kinase autophosphorylation assay in HUVEC cells

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Angiopoietin-1 receptor


(Homo sapiens (Human))		BDBM50162973
PNG
(CHEMBL177298 | N-[4-(Benzothiazol-6-ylamino)-6-(1-...)
Show SMILES CC(C)(Nc1nc(NO)nc(Nc2ccc3ncsc3c2)n1)c1ccccc1
Show InChI InChI=1S/C19H19N7OS/c1-19(2,12-6-4-3-5-7-12)25-17-22-16(23-18(24-17)26-27)21-13-8-9-14-15(10-13)28-11-20-14/h3-11,27H,1-2H3,(H3,21,22,23,24,25,26)
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n/an/a 700n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
Inhibition of tyrosine protein kinase receptor TIE-2

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Angiopoietin-1 receptor


(Homo sapiens (Human))		BDBM50162976
PNG
(4-(Benzothiazol-6-ylamino)-6-(1-methyl-1-phenyl-et...)
Show SMILES CC(C)(Nc1nc(Nc2ccc3ncsc3c2)[nH]c(=O)n1)c1ccccc1
Show InChI InChI=1S/C19H18N6OS/c1-19(2,12-6-4-3-5-7-12)25-17-22-16(23-18(26)24-17)21-13-8-9-14-15(10-13)27-11-20-14/h3-11H,1-2H3,(H3,21,22,23,24,25,26)
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n/an/a 1.00E+3n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
Inhibition of tyrosine protein kinase receptor TIE-2

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Vascular endothelial growth factor receptor 2


(Homo sapiens (Human))		BDBM50162977
PNG
(4-(Benzothiazol-6-yl-methyl-amino)-6-(1-methyl-1-p...)
Show SMILES CN(c1ccc2ncsc2c1)c1nc(NC(C)(C)c2ccccc2)nc(=O)[nH]1
Show InChI InChI=1S/C20H20N6OS/c1-20(2,13-7-5-4-6-8-13)25-17-22-18(24-19(27)23-17)26(3)14-9-10-15-16(11-14)28-12-21-15/h4-12H,1-3H3,(H2,22,23,24,25,27)
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n/an/a 1.60E+3n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
In vitro inhibition of Vascular endothelial growth factor receptor 2 at 10 uM ATP

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Vascular endothelial growth factor receptor 2


(Homo sapiens (Human))		BDBM50162981
PNG
(4-(Benzothiazol-6-ylamino)-6-benzylamino-[1,3,5]tr...)
Show SMILES O=c1nc(NCc2ccccc2)nc(Nc2ccc3ncsc3c2)[nH]1
Show InChI InChI=1S/C17H14N6OS/c24-17-22-15(18-9-11-4-2-1-3-5-11)21-16(23-17)20-12-6-7-13-14(8-12)25-10-19-13/h1-8,10H,9H2,(H3,18,20,21,22,23,24)
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n/an/a 2.00E+3n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
In vitro inhibition of Vascular endothelial growth factor receptor 2 at 10 uM ATP

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Platelet-derived growth factor receptor alpha/beta


(Homo sapiens (Human))		BDBM50162978
PNG
(4-(Benzothiazol-6-ylamino)-6-(benzyl-ethyl-amino)-...)
Show SMILES CCN(Cc1ccccc1)c1nc(Nc2ccc3ncsc3c2)[nH]c(=O)n1
Show InChI InChI=1S/C19H18N6OS/c1-2-25(11-13-6-4-3-5-7-13)18-22-17(23-19(26)24-18)21-14-8-9-15-16(10-14)27-12-20-15/h3-10,12H,2,11H2,1H3,(H2,21,22,23,24,26)
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n/an/a 2.50E+3n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
Inhibition of PDGF-R2 tyrosine kinase

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Platelet-derived growth factor receptor alpha/beta


(Homo sapiens (Human))		BDBM50162973
PNG
(CHEMBL177298 | N-[4-(Benzothiazol-6-ylamino)-6-(1-...)
Show SMILES CC(C)(Nc1nc(NO)nc(Nc2ccc3ncsc3c2)n1)c1ccccc1
Show InChI InChI=1S/C19H19N7OS/c1-19(2,12-6-4-3-5-7-12)25-17-22-16(23-18(24-17)26-27)21-13-8-9-14-15(10-13)28-11-20-14/h3-11,27H,1-2H3,(H3,21,22,23,24,25,26)
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n/an/a 3.90E+3n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
Inhibition of PDGF-R2 tyrosine kinase

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Insulin receptor


(Homo sapiens (Human))		BDBM50162978
PNG
(4-(Benzothiazol-6-ylamino)-6-(benzyl-ethyl-amino)-...)
Show SMILES CCN(Cc1ccccc1)c1nc(Nc2ccc3ncsc3c2)[nH]c(=O)n1
Show InChI InChI=1S/C19H18N6OS/c1-2-25(11-13-6-4-3-5-7-13)18-22-17(23-19(26)24-18)21-14-8-9-15-16(10-14)27-12-20-15/h3-10,12H,2,11H2,1H3,(H2,21,22,23,24,26)
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n/an/a 4.00E+3n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
Inhibition of beta IRK tyrosine kinase

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Macrophage colony-stimulating factor 1 receptor


(Homo sapiens (Human))		BDBM50162978
PNG
(4-(Benzothiazol-6-ylamino)-6-(benzyl-ethyl-amino)-...)
Show SMILES CCN(Cc1ccccc1)c1nc(Nc2ccc3ncsc3c2)[nH]c(=O)n1
Show InChI InChI=1S/C19H18N6OS/c1-2-25(11-13-6-4-3-5-7-13)18-22-17(23-19(26)24-18)21-14-8-9-15-16(10-14)27-12-20-15/h3-10,12H,2,11H2,1H3,(H2,21,22,23,24,26)
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n/an/a 4.30E+3n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
Inhibition of c-fms tyrosine kinase

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Vascular endothelial growth factor receptor 2


(Homo sapiens (Human))		BDBM50162980
PNG
(CHEMBL175760 | N-Benzothiazol-6-yl-6-chloro-N''-(1...)
Show SMILES CC(C)(Nc1nc(Cl)nc(Nc2ccc3ncsc3c2)n1)c1ccccc1
Show InChI InChI=1S/C19H17ClN6S/c1-19(2,12-6-4-3-5-7-12)26-18-24-16(20)23-17(25-18)22-13-8-9-14-15(10-13)27-11-21-14/h3-11H,1-2H3,(H2,22,23,24,25,26)
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n/an/a 5.50E+3n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
In vitro inhibition of Vascular endothelial growth factor receptor 2 at 10 uM ATP

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Vascular endothelial growth factor receptor 2


(Homo sapiens (Human))		BDBM50162980
PNG
(CHEMBL175760 | N-Benzothiazol-6-yl-6-chloro-N''-(1...)
Show SMILES CC(C)(Nc1nc(Cl)nc(Nc2ccc3ncsc3c2)n1)c1ccccc1
Show InChI InChI=1S/C19H17ClN6S/c1-19(2,12-6-4-3-5-7-12)26-18-24-16(20)23-17(25-18)22-13-8-9-14-15(10-13)27-11-21-14/h3-11H,1-2H3,(H2,22,23,24,25,26)
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n/an/a 5.50E+3n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
In vitro inhibition of Vascular endothelial growth factor receptor 2 at 10 uM ATP

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Vascular endothelial growth factor receptor 2


(Homo sapiens (Human))		BDBM50162979
PNG
(CHEMBL175506 | N-Benzothiazol-6-yl-6-methoxy-N''-(...)
Show SMILES COc1nc(Nc2ccc3ncsc3c2)nc(NC(C)(C)c2ccccc2)n1
Show InChI InChI=1S/C20H20N6OS/c1-20(2,13-7-5-4-6-8-13)26-18-23-17(24-19(25-18)27-3)22-14-9-10-15-16(11-14)28-12-21-15/h4-12H,1-3H3,(H2,22,23,24,25,26)
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n/an/a 6.10E+3n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
In vitro inhibition of Vascular endothelial growth factor receptor 2 at 10 uM ATP

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Platelet-derived growth factor receptor alpha/beta


(Homo sapiens (Human))		BDBM50162976
PNG
(4-(Benzothiazol-6-ylamino)-6-(1-methyl-1-phenyl-et...)
Show SMILES CC(C)(Nc1nc(Nc2ccc3ncsc3c2)[nH]c(=O)n1)c1ccccc1
Show InChI InChI=1S/C19H18N6OS/c1-19(2,12-6-4-3-5-7-12)25-17-22-16(23-18(26)24-17)21-13-8-9-14-15(10-13)27-11-20-14/h3-11H,1-2H3,(H3,21,22,23,24,25,26)
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n/an/a 8.00E+3n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
Inhibition of PDGF-R2 tyrosine kinase

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Vascular endothelial growth factor receptor 2


(Homo sapiens (Human))		BDBM50162977
PNG
(4-(Benzothiazol-6-yl-methyl-amino)-6-(1-methyl-1-p...)
Show SMILES CN(c1ccc2ncsc2c1)c1nc(NC(C)(C)c2ccccc2)nc(=O)[nH]1
Show InChI InChI=1S/C20H20N6OS/c1-20(2,13-7-5-4-6-8-13)25-17-22-18(24-19(27)23-17)26(3)14-9-10-15-16(11-14)28-12-21-15/h4-12H,1-3H3,(H2,22,23,24,25,27)
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n/an/a 9.90E+3n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
Inhibition of KDR-induced MAP kinase autophosphorylation assay in HUVEC cells

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Fibroblast growth factor receptor 1


(Mus musculus)		BDBM50162978
PNG
(4-(Benzothiazol-6-ylamino)-6-(benzyl-ethyl-amino)-...)
Show SMILES CCN(Cc1ccccc1)c1nc(Nc2ccc3ncsc3c2)[nH]c(=O)n1
Show InChI InChI=1S/C19H18N6OS/c1-2-25(11-13-6-4-3-5-7-13)18-22-17(23-19(26)24-18)21-14-8-9-15-16(10-14)27-12-20-15/h3-10,12H,2,11H2,1H3,(H2,21,22,23,24,26)
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n/an/a>1.00E+4n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
Inhibition of mouse Fibroblast growth factor receptor 1 expressed in NIH 3T3 fibroblasts

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Epidermal growth factor receptor


(Homo sapiens (Human))		BDBM50162973
PNG
(CHEMBL177298 | N-[4-(Benzothiazol-6-ylamino)-6-(1-...)
Show SMILES CC(C)(Nc1nc(NO)nc(Nc2ccc3ncsc3c2)n1)c1ccccc1
Show InChI InChI=1S/C19H19N7OS/c1-19(2,12-6-4-3-5-7-12)25-17-22-16(23-18(24-17)26-27)21-13-8-9-14-15(10-13)28-11-20-14/h3-11,27H,1-2H3,(H3,21,22,23,24,25,26)
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n/an/a>1.00E+4n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
Inhibition of human epidermal growth factor receptor

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Fibroblast growth factor receptor 1


(Mus musculus)		BDBM50162972
PNG
(4-(Benzothiazol-6-ylamino)-6-(benzyl-isopropyl-ami...)
Show SMILES CC(C)N(Cc1ccccc1)c1nc(Nc2ccc3ncsc3c2)[nH]c(=O)n1
Show InChI InChI=1S/C20H20N6OS/c1-13(2)26(11-14-6-4-3-5-7-14)19-23-18(24-20(27)25-19)22-15-8-9-16-17(10-15)28-12-21-16/h3-10,12-13H,11H2,1-2H3,(H2,22,23,24,25,27)
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n/an/a>1.00E+4n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
Inhibition of mouse Fibroblast growth factor receptor 1 expressed in NIH 3T3 fibroblasts

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Fibroblast growth factor receptor 1


(Mus musculus)		BDBM50162976
PNG
(4-(Benzothiazol-6-ylamino)-6-(1-methyl-1-phenyl-et...)
Show SMILES CC(C)(Nc1nc(Nc2ccc3ncsc3c2)[nH]c(=O)n1)c1ccccc1
Show InChI InChI=1S/C19H18N6OS/c1-19(2,12-6-4-3-5-7-12)25-17-22-16(23-18(26)24-17)21-13-8-9-14-15(10-13)27-11-20-14/h3-11H,1-2H3,(H3,21,22,23,24,25,26)
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n/an/a>1.00E+4n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
Inhibition of mouse Fibroblast growth factor receptor 1 expressed in NIH 3T3 fibroblasts

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Fibroblast growth factor receptor 1


(Mus musculus)		BDBM50162973
PNG
(CHEMBL177298 | N-[4-(Benzothiazol-6-ylamino)-6-(1-...)
Show SMILES CC(C)(Nc1nc(NO)nc(Nc2ccc3ncsc3c2)n1)c1ccccc1
Show InChI InChI=1S/C19H19N7OS/c1-19(2,12-6-4-3-5-7-12)25-17-22-16(23-18(24-17)26-27)21-13-8-9-14-15(10-13)28-11-20-14/h3-11,27H,1-2H3,(H3,21,22,23,24,25,26)
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n/an/a>1.00E+4n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
Inhibition of mouse Fibroblast growth factor receptor 1 expressed in NIH 3T3 fibroblasts

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Insulin receptor


(Homo sapiens (Human))		BDBM50162978
PNG
(4-(Benzothiazol-6-ylamino)-6-(benzyl-ethyl-amino)-...)
Show SMILES CCN(Cc1ccccc1)c1nc(Nc2ccc3ncsc3c2)[nH]c(=O)n1
Show InChI InChI=1S/C19H18N6OS/c1-2-25(11-13-6-4-3-5-7-13)18-22-17(23-19(26)24-18)21-14-8-9-15-16(10-14)27-12-20-15/h3-10,12H,2,11H2,1H3,(H2,21,22,23,24,26)
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n/an/a>1.00E+4n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
Inhibition of human Insulin receptor expressed in CHO cells

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Epidermal growth factor receptor


(Homo sapiens (Human))		BDBM50162978
PNG
(4-(Benzothiazol-6-ylamino)-6-(benzyl-ethyl-amino)-...)
Show SMILES CCN(Cc1ccccc1)c1nc(Nc2ccc3ncsc3c2)[nH]c(=O)n1
Show InChI InChI=1S/C19H18N6OS/c1-2-25(11-13-6-4-3-5-7-13)18-22-17(23-19(26)24-18)21-14-8-9-15-16(10-14)27-12-20-15/h3-10,12H,2,11H2,1H3,(H2,21,22,23,24,26)
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n/an/a>1.00E+4n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
Inhibition of human epidermal growth factor receptor

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Insulin receptor


(Homo sapiens (Human))		BDBM50162973
PNG
(CHEMBL177298 | N-[4-(Benzothiazol-6-ylamino)-6-(1-...)
Show SMILES CC(C)(Nc1nc(NO)nc(Nc2ccc3ncsc3c2)n1)c1ccccc1
Show InChI InChI=1S/C19H19N7OS/c1-19(2,12-6-4-3-5-7-12)25-17-22-16(23-18(24-17)26-27)21-13-8-9-14-15(10-13)28-11-20-14/h3-11,27H,1-2H3,(H3,21,22,23,24,25,26)
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n/an/a>1.00E+4n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
Inhibition of human Insulin receptor expressed in CHO cells

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Epidermal growth factor receptor


(Homo sapiens (Human))		BDBM50162972
PNG
(4-(Benzothiazol-6-ylamino)-6-(benzyl-isopropyl-ami...)
Show SMILES CC(C)N(Cc1ccccc1)c1nc(Nc2ccc3ncsc3c2)[nH]c(=O)n1
Show InChI InChI=1S/C20H20N6OS/c1-13(2)26(11-14-6-4-3-5-7-14)19-23-18(24-20(27)25-19)22-15-8-9-16-17(10-15)28-12-21-16/h3-10,12-13H,11H2,1-2H3,(H2,22,23,24,25,27)
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n/an/a>1.00E+4n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
Inhibition of human epidermal growth factor receptor

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Epidermal growth factor receptor


(Homo sapiens (Human))		BDBM50162976
PNG
(4-(Benzothiazol-6-ylamino)-6-(1-methyl-1-phenyl-et...)
Show SMILES CC(C)(Nc1nc(Nc2ccc3ncsc3c2)[nH]c(=O)n1)c1ccccc1
Show InChI InChI=1S/C19H18N6OS/c1-19(2,12-6-4-3-5-7-12)25-17-22-16(23-18(26)24-17)21-13-8-9-14-15(10-13)27-11-20-14/h3-11H,1-2H3,(H3,21,22,23,24,25,26)
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n/an/a>1.00E+4n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
Inhibition of human epidermal growth factor receptor

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Insulin receptor


(Homo sapiens (Human))		BDBM50162972
PNG
(4-(Benzothiazol-6-ylamino)-6-(benzyl-isopropyl-ami...)
Show SMILES CC(C)N(Cc1ccccc1)c1nc(Nc2ccc3ncsc3c2)[nH]c(=O)n1
Show InChI InChI=1S/C20H20N6OS/c1-13(2)26(11-14-6-4-3-5-7-14)19-23-18(24-20(27)25-19)22-15-8-9-16-17(10-15)28-12-21-16/h3-10,12-13H,11H2,1-2H3,(H2,22,23,24,25,27)
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n/an/a>1.00E+4n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
Inhibition of human Insulin receptor expressed in CHO cells

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Insulin receptor


(Homo sapiens (Human))		BDBM50162976
PNG
(4-(Benzothiazol-6-ylamino)-6-(1-methyl-1-phenyl-et...)
Show SMILES CC(C)(Nc1nc(Nc2ccc3ncsc3c2)[nH]c(=O)n1)c1ccccc1
Show InChI InChI=1S/C19H18N6OS/c1-19(2,12-6-4-3-5-7-12)25-17-22-16(23-18(26)24-17)21-13-8-9-14-15(10-13)27-11-20-14/h3-11H,1-2H3,(H3,21,22,23,24,25,26)
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n/an/a>1.00E+4n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
Inhibition of human Insulin receptor expressed in CHO cells

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Insulin receptor


(Homo sapiens (Human))		BDBM50162972
PNG
(4-(Benzothiazol-6-ylamino)-6-(benzyl-isopropyl-ami...)
Show SMILES CC(C)N(Cc1ccccc1)c1nc(Nc2ccc3ncsc3c2)[nH]c(=O)n1
Show InChI InChI=1S/C20H20N6OS/c1-13(2)26(11-14-6-4-3-5-7-14)19-23-18(24-20(27)25-19)22-15-8-9-16-17(10-15)28-12-21-16/h3-10,12-13H,11H2,1-2H3,(H2,22,23,24,25,27)
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n/an/a 1.10E+4n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
Inhibition of beta IRK tyrosine kinase

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Macrophage colony-stimulating factor 1 receptor


(Homo sapiens (Human))		BDBM50162972
PNG
(4-(Benzothiazol-6-ylamino)-6-(benzyl-isopropyl-ami...)
Show SMILES CC(C)N(Cc1ccccc1)c1nc(Nc2ccc3ncsc3c2)[nH]c(=O)n1
Show InChI InChI=1S/C20H20N6OS/c1-13(2)26(11-14-6-4-3-5-7-14)19-23-18(24-20(27)25-19)22-15-8-9-16-17(10-15)28-12-21-16/h3-10,12-13H,11H2,1-2H3,(H2,22,23,24,25,27)
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n/an/a>1.25E+4n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
Inhibition of c-fms tyrosine kinase

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Macrophage colony-stimulating factor 1 receptor


(Homo sapiens (Human))		BDBM50162976
PNG
(4-(Benzothiazol-6-ylamino)-6-(1-methyl-1-phenyl-et...)
Show SMILES CC(C)(Nc1nc(Nc2ccc3ncsc3c2)[nH]c(=O)n1)c1ccccc1
Show InChI InChI=1S/C19H18N6OS/c1-19(2,12-6-4-3-5-7-12)25-17-22-16(23-18(26)24-17)21-13-8-9-14-15(10-13)27-11-20-14/h3-11H,1-2H3,(H3,21,22,23,24,25,26)
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n/an/a>1.25E+4n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
Inhibition of c-fms tyrosine kinase

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Platelet-derived growth factor receptor alpha/beta


(Homo sapiens (Human))		BDBM50162972
PNG
(4-(Benzothiazol-6-ylamino)-6-(benzyl-isopropyl-ami...)
Show SMILES CC(C)N(Cc1ccccc1)c1nc(Nc2ccc3ncsc3c2)[nH]c(=O)n1
Show InChI InChI=1S/C20H20N6OS/c1-13(2)26(11-14-6-4-3-5-7-14)19-23-18(24-20(27)25-19)22-15-8-9-16-17(10-15)28-12-21-16/h3-10,12-13H,11H2,1-2H3,(H2,22,23,24,25,27)
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n/an/a>1.25E+4n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
Inhibition of PDGF-R2 tyrosine kinase

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Macrophage colony-stimulating factor 1 receptor


(Homo sapiens (Human))		BDBM50162973
PNG
(CHEMBL177298 | N-[4-(Benzothiazol-6-ylamino)-6-(1-...)
Show SMILES CC(C)(Nc1nc(NO)nc(Nc2ccc3ncsc3c2)n1)c1ccccc1
Show InChI InChI=1S/C19H19N7OS/c1-19(2,12-6-4-3-5-7-12)25-17-22-16(23-18(24-17)26-27)21-13-8-9-14-15(10-13)28-11-20-14/h3-11,27H,1-2H3,(H3,21,22,23,24,25,26)
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n/an/a 1.40E+4n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
Inhibition of c-fms tyrosine kinase

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Vascular endothelial growth factor receptor 2


(Homo sapiens (Human))		BDBM50162975
PNG
(4-(3H-Benzoimidazol-5-ylamino)-6-(1-methyl-1-pheny...)
Show SMILES CC(C)(Nc1nc(Nc2ccc3nc[nH]c3c2)[nH]c(=O)n1)c1ccccc1
Show InChI InChI=1S/C19H19N7O/c1-19(2,12-6-4-3-5-7-12)26-17-23-16(24-18(27)25-17)22-13-8-9-14-15(10-13)21-11-20-14/h3-11H,1-2H3,(H,20,21)(H3,22,23,24,25,26,27)
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n/an/a>2.00E+4n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
In vitro inhibition of Vascular endothelial growth factor receptor 2 at 10 uM ATP

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Vascular endothelial growth factor receptor 2


(Homo sapiens (Human))		BDBM50162981
PNG
(4-(Benzothiazol-6-ylamino)-6-benzylamino-[1,3,5]tr...)
Show SMILES O=c1nc(NCc2ccccc2)nc(Nc2ccc3ncsc3c2)[nH]1
Show InChI InChI=1S/C17H14N6OS/c24-17-22-15(18-9-11-4-2-1-3-5-11)21-16(23-17)20-12-6-7-13-14(8-12)25-10-19-13/h1-8,10H,9H2,(H3,18,20,21,22,23,24)
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n/an/a>3.00E+4n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
Inhibition of KDR-induced MAP kinase autophosphorylation assay in HUVEC cells

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
Vascular endothelial growth factor receptor 2


(Homo sapiens (Human))		BDBM50162979
PNG
(CHEMBL175506 | N-Benzothiazol-6-yl-6-methoxy-N''-(...)
Show SMILES COc1nc(Nc2ccc3ncsc3c2)nc(NC(C)(C)c2ccccc2)n1
Show InChI InChI=1S/C20H20N6OS/c1-20(2,13-7-5-4-6-8-13)26-18-23-17(24-19(25-18)27-3)22-14-9-10-15-16(11-14)28-12-21-15/h4-12H,1-3H3,(H2,22,23,24,25,26)
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n/an/a>3.00E+4n/an/an/an/an/an/a



Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL


Assay Description
Inhibition of KDR-induced MAP kinase autophosphorylation assay in HUVEC cells

J Med Chem 48: 1717-20 (2005)


Article DOI: 10.1021/jm049372z
BindingDB Entry DOI: 10.7270/Q2GM86TF
More data for this
Ligand-Target Pair
* indicates data uncertainty>20%