Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Muscarinic acetylcholine receptor M3 (Homo sapiens (Human)) | BDBM50259847 (CHEMBL480464 | cremastrine) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 126 | n/a | n/a | n/a | n/a | n/a | n/a |
Mitsubishi Pharma Corporation Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human cloned muscarinic M3 receptor expressed in insect Sf9 cells | J Nat Prod 68: 572-3 (2005) Article DOI: 10.1021/np049650x BindingDB Entry DOI: 10.7270/Q2HH6JVJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M4 (Homo sapiens (Human)) | BDBM50259847 (CHEMBL480464 | cremastrine) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 498 | n/a | n/a | n/a | n/a | n/a | n/a |
Mitsubishi Pharma Corporation Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human cloned muscarinic M4 receptor expressed in insect Sf9 cells | J Nat Prod 68: 572-3 (2005) Article DOI: 10.1021/np049650x BindingDB Entry DOI: 10.7270/Q2HH6JVJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M1 (Homo sapiens (Human)) | BDBM50259847 (CHEMBL480464 | cremastrine) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 505 | n/a | n/a | n/a | n/a | n/a | n/a |
Mitsubishi Pharma Corporation Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human cloned muscarinic M1 receptor expressed in insect Sf9 cells | J Nat Prod 68: 572-3 (2005) Article DOI: 10.1021/np049650x BindingDB Entry DOI: 10.7270/Q2HH6JVJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M5 (Homo sapiens (Human)) | BDBM50259847 (CHEMBL480464 | cremastrine) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.22E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Mitsubishi Pharma Corporation Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human cloned muscarinic M5 receptor expressed in insect Sf9 cells | J Nat Prod 68: 572-3 (2005) Article DOI: 10.1021/np049650x BindingDB Entry DOI: 10.7270/Q2HH6JVJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscarinic acetylcholine receptor M2 (Homo sapiens (Human)) | BDBM50259847 (CHEMBL480464 | cremastrine) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | >5.52E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Mitsubishi Pharma Corporation Curated by ChEMBL | Assay Description Displacement of [3H]NMS from human cloned muscarinic M2 receptor expressed in insect Sf9 cells | J Nat Prod 68: 572-3 (2005) Article DOI: 10.1021/np049650x BindingDB Entry DOI: 10.7270/Q2HH6JVJ | |||||||||||
More data for this Ligand-Target Pair |