Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50169445 ((1S,4R,6S)-2-Methyl-2-aza-bicyclo[2.2.2]octane-6-c...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Inhibition concentration (binding affinity) against human melanocortin receptor 4 by displacement of [125I]-NDP-alpha-MSH from the human receptors ex... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50169442 ((1R,4S,6R)-2-Methyl-2-aza-bicyclo[2.2.2]octane-6-c...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Inhibition concentration (binding affinity) against human melanocortin receptor 4 by displacement of [125I]-NDP-alpha-MSH from the human receptors ex... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50169444 ((1S,4S,6S)-2-Aza-bicyclo[2.2.2]octane-6-carboxylic...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 14 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Inhibition concentration (binding affinity) against human melanocortin receptor 4 by displacement of [125I]-NDP-alpha-MSH from the human receptors ex... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50024351 (CHEMBL2113031) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 16 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Inhibition concentration (binding affinity) against human melanocortin receptor 4 by displacement of [125I]-NDP-alpha-MSH from the human receptors ex... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50029747 ((4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 19 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Inhibition concentration (binding affinity) against human melanocortin receptor 4 by displacement of [125I]-NDP-alpha-MSH from the human receptors ex... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 3 (Homo sapiens (Human)) | BDBM50029747 ((4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 19 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Inhibition concentration (binding affinity) against human melanocortin receptor 3 by displacement of [125I]NDP-alpha-MSH from the human receptors exp... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50169443 ((1R,4S,6S)-2-Methyl-2-aza-bicyclo[2.2.2]octane-6-c...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 28 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Inhibition concentration (binding affinity) against human melanocortin receptor 4 by displacement of [125I]-NDP-alpha-MSH from the human receptors ex... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50169440 ((1S,4R,6S)-2-Aza-bicyclo[2.2.2]octane-6-carboxylic...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 41 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Inhibition concentration (binding affinity) against human melanocortin receptor 4 by displacement of [125I]-NDP-alpha-MSH from the human receptors ex... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50029747 ((4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 118 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Effective concentration (binding affinity) exhibited against human melanocortin receptor 5 by radio labeled ligand assay (Displacement of [125I]NDP-a... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 3 (Homo sapiens (Human)) | BDBM50169445 ((1S,4R,6S)-2-Methyl-2-aza-bicyclo[2.2.2]octane-6-c...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 410 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Inhibition concentration (binding affinity) against human melanocortin receptor 3 by displacement of [125I]NDP-alpha-MSH from the human receptors exp... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 3 (Homo sapiens (Human)) | BDBM50169444 ((1S,4S,6S)-2-Aza-bicyclo[2.2.2]octane-6-carboxylic...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 620 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Inhibition concentration (binding affinity) against human melanocortin receptor 3 by displacement of [125I]NDP-alpha-MSH from the human receptors exp... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 3 (Homo sapiens (Human)) | BDBM50024351 (CHEMBL2113031) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 620 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Inhibition concentration (binding affinity) against human melanocortin receptor 3 by displacement of [125I]NDP-alpha-MSH from the human receptors exp... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50024351 (CHEMBL2113031) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 940 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Inhibition concentration (binding affinity) against human melanocortin receptor 5 by displacement of [125I]NDP-alpha-MSH from the human receptors exp... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50169444 ((1S,4S,6S)-2-Aza-bicyclo[2.2.2]octane-6-carboxylic...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.02E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Effective concentration (binding affinity) exhibited against human melanocortin receptor 5 by radio labeled ligand assay (Displacement of [125I]NDP-a... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50169445 ((1S,4R,6S)-2-Methyl-2-aza-bicyclo[2.2.2]octane-6-c...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.08E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Effective concentration (binding affinity) exhibited against human melanocortin receptor 5 by radio labeled ligand assay (Displacement of [125I]NDP-a... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 3 (Homo sapiens (Human)) | BDBM50169443 ((1R,4S,6S)-2-Methyl-2-aza-bicyclo[2.2.2]octane-6-c...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.35E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Inhibition concentration (binding affinity) against human melanocortin receptor 3 by displacement of [125I]NDP-alpha-MSH from the human receptors exp... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 3 (Homo sapiens (Human)) | BDBM50169440 ((1S,4R,6S)-2-Aza-bicyclo[2.2.2]octane-6-carboxylic...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.06E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Inhibition concentration (binding affinity) against human melanocortin receptor 3 by displacement of [125I]NDP-alpha-MSH from the human receptors exp... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50169442 ((1R,4S,6R)-2-Methyl-2-aza-bicyclo[2.2.2]octane-6-c...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Inhibition concentration (binding affinity) against mouse melanocortin receptor 4 by displacement of [125I]-NDP-alpha-MSH from the human receptors ex... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Rattus norvegicus) | BDBM50169442 ((1R,4S,6R)-2-Methyl-2-aza-bicyclo[2.2.2]octane-6-c...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Inhibition concentration (binding affinity) against rat melanocortin receptor 4 by displacement of [125I]-NDP-alpha-MSH from the human receptors expr... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50169443 ((1R,4S,6S)-2-Methyl-2-aza-bicyclo[2.2.2]octane-6-c...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 6.46E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Inhibition concentration (binding affinity) against human melanocortin receptor 5 by displacement of [125I]NDP-alpha-MSH from the human receptors exp... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50169442 ((1R,4S,6R)-2-Methyl-2-aza-bicyclo[2.2.2]octane-6-c...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Inhibition concentration (binding affinity) against dog melanocortin receptor 4 by displacement of [125I]-NDP-alpha-MSH from the human receptors expr... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50169440 ((1S,4R,6S)-2-Aza-bicyclo[2.2.2]octane-6-carboxylic...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.87E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Effective concentration (binding affinity) exhibited against human melanocortin receptor 5 by radio labeled ligand assay (Displacement of [125I]NDP-a... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adrenocorticotropic hormone receptor (Homo sapiens (Human)) | BDBM50169442 ((1R,4S,6R)-2-Methyl-2-aza-bicyclo[2.2.2]octane-6-c...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Inhibition concentration (binding affinity) against human melanocortin receptor 2 by displacement of [125I]NDP-alpha-MSH from the human receptors exp... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM50169442 ((1R,4S,6R)-2-Methyl-2-aza-bicyclo[2.2.2]octane-6-c...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.50E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Inhibition concentration (binding affinity) against human melanocortin receptor 1 by displacement of [125I]NDP-alpha-MSH from the human receptors exp... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 3 (Homo sapiens (Human)) | BDBM50169442 ((1R,4S,6R)-2-Methyl-2-aza-bicyclo[2.2.2]octane-6-c...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.42E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Inhibition concentration (binding affinity) against human melanocortin receptor 3 by displacement of [125I]NDP-alpha-MSH from the human receptors exp... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50169442 ((1R,4S,6R)-2-Methyl-2-aza-bicyclo[2.2.2]octane-6-c...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.45E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Inhibition concentration (binding affinity) against human melanocortin receptor 5 by displacement of [125I]NDP-alpha-MSH from the human receptors exp... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50169445 ((1S,4R,6S)-2-Methyl-2-aza-bicyclo[2.2.2]octane-6-c...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 34 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Inhibition concentration (binding affinity) exhibited against human melanocortin receptor 4 by radio labeled ligand assay (Displacement of [125I]-NDP... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50169442 ((1R,4S,6R)-2-Methyl-2-aza-bicyclo[2.2.2]octane-6-c...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 8.50E+5 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Effective concentration (binding affinity) exhibited against human melanocortin receptor 5 by radio labeled ligand assay (Displacement of [125I]-NDP-... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50029747 ((4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 17 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Inhibition concentration (binding affinity) exhibited against human melanocortin receptor 5 by radio labeled ligand assay (Displacement of [125I]-NDP... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50169442 ((1R,4S,6R)-2-Methyl-2-aza-bicyclo[2.2.2]octane-6-c...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.10E+4 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Concentration of compound at 50% maximum cAMP accumulation in human melanocortin receptor (hMC4R) | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50169444 ((1S,4S,6S)-2-Aza-bicyclo[2.2.2]octane-6-carboxylic...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 52 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Inhibition concentration (binding affinity) exhibited against human melanocortin receptor 4 by radio labeled ligand assay (Displacement of [125I]-NDP... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50169442 ((1R,4S,6R)-2-Methyl-2-aza-bicyclo[2.2.2]octane-6-c...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 8.50E+5 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Concentration of compound at 50% maximum cAMP accumulation in human melanocortin receptor (hMC5R) | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Rattus norvegicus) | BDBM50169442 ((1R,4S,6R)-2-Methyl-2-aza-bicyclo[2.2.2]octane-6-c...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 5.00E+3 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Concentration of compound at 50% maximum cAMP accumulation in rat melanocortin receptor (rMC4R) | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50169440 ((1S,4R,6S)-2-Aza-bicyclo[2.2.2]octane-6-carboxylic...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 238 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Inhibition concentration (binding affinity) exhibited against human melanocortin receptor 4 by radio labeled ligand assay (Displacement of [125I]-NDP... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50169442 ((1R,4S,6R)-2-Methyl-2-aza-bicyclo[2.2.2]octane-6-c...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 8.50E+5 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Effective concentration (binding affinity) exhibited against human melanocortin receptor 5 by radio labeled ligand assay (Displacement of [125I]-NDP-... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50169442 ((1R,4S,6R)-2-Methyl-2-aza-bicyclo[2.2.2]octane-6-c...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.10E+4 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Effective concentration (binding affinity) exhibited against human melanocortin receptor 4 by radio labeled ligand assay (Displacement of [125I]-NDP-... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50024351 (CHEMBL2113031) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 20 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Inhibition concentration (binding affinity) exhibited against human melanocortin receptor 4 by radio labeled ligand assay (Displacement of [125I]-NDP... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 3 (Homo sapiens (Human)) | BDBM50029747 ((4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.10 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Inhibition concentration (binding affinity) exhibited against human melanocortin receptor 3 by radio labeled ligand assay (Displacement of [125I]-NDP... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM50169442 ((1R,4S,6R)-2-Methyl-2-aza-bicyclo[2.2.2]octane-6-c...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.60E+5 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Concentration of compound at 50% maximum cAMP accumulation in human melanocortin receptor (hMC1R) | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50169442 ((1R,4S,6R)-2-Methyl-2-aza-bicyclo[2.2.2]octane-6-c...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 6.00E+3 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Concentration of compound at 50% maximum cAMP accumulation in mouse melanocortin receptor (mMC4R) | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50169443 ((1R,4S,6S)-2-Methyl-2-aza-bicyclo[2.2.2]octane-6-c...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 165 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Effective concentration (binding affinity) exhibited against human melanocortin receptor 4 by radio labeled ligand assay (Displacement of [125I]-NDP-... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocyte-stimulating hormone receptor (Homo sapiens (Human)) | BDBM50169442 ((1R,4S,6R)-2-Methyl-2-aza-bicyclo[2.2.2]octane-6-c...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.60E+5 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Effective concentration (binding affinity) exhibited against human melanocortin receptor 1 by radio labeled ligand assay (Displacement of [125I]-NDP-... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50169443 ((1R,4S,6S)-2-Methyl-2-aza-bicyclo[2.2.2]octane-6-c...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 850 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Inhibition concentration (binding affinity) exhibited against human melanocortin receptor 5 by radio labeled ligand assay (Displacement of [125I]-NDP... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50169442 ((1R,4S,6R)-2-Methyl-2-aza-bicyclo[2.2.2]octane-6-c...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.10E+4 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Concentration of compound at 50% maximum cAMP accumulation in dog melanocortin receptor (dMC4R) | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Homo sapiens (Human)) | BDBM50029747 ((4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.90 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Inhibition concentration (binding affinity) exhibited against human melanocortin receptor 4 by radio labeled ligand assay (Displacement of [125I]-NDP... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Homo sapiens (Human)) | BDBM50169440 ((1S,4R,6S)-2-Aza-bicyclo[2.2.2]octane-6-carboxylic...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.98E+3 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Inhibition concentration (binding affinity) exhibited against human melanocortin receptor 5 by radio labeled ligand assay (Displacement of [125I]-NDP... | Bioorg Med Chem Lett 15: 3501-5 (2005) Article DOI: 10.1016/j.bmcl.2005.05.109 BindingDB Entry DOI: 10.7270/Q2Q81CKF | |||||||||||
More data for this Ligand-Target Pair |