Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50175766 (1-(1-butyl-4-(3-methoxyphenyl)-2-oxo-1,2-dihydro-1...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.40 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Pharmaceuticals Co., Ltd Curated by ChEMBL | Assay Description Inhibitory activity against ACAT in rat macrophages | Bioorg Med Chem Lett 16: 44-8 (2005) Article DOI: 10.1016/j.bmcl.2005.09.056 BindingDB Entry DOI: 10.7270/Q2PG1SH8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50175771 (1-(4-amino-2,6-diisopropylphenyl)-3-(1-butyl-4-(3-...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Pharmaceuticals Co., Ltd Curated by ChEMBL | Assay Description Inhibitory activity against ACAT in rat macrophages | Bioorg Med Chem Lett 16: 44-8 (2005) Article DOI: 10.1016/j.bmcl.2005.09.056 BindingDB Entry DOI: 10.7270/Q2PG1SH8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50175772 (1-(1-butyl-4-(3-methoxyphenyl)-2-oxo-1,2-dihydro-1...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Pharmaceuticals Co., Ltd Curated by ChEMBL | Assay Description Inhibitory activity against ACAT in rat macrophages | Bioorg Med Chem Lett 16: 44-8 (2005) Article DOI: 10.1016/j.bmcl.2005.09.056 BindingDB Entry DOI: 10.7270/Q2PG1SH8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50175767 (1-(3-amino-2,6-diisopropylphenyl)-3-(1-butyl-4-(3-...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 14 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Pharmaceuticals Co., Ltd Curated by ChEMBL | Assay Description Inhibitory activity against ACAT in rat macrophages | Bioorg Med Chem Lett 16: 44-8 (2005) Article DOI: 10.1016/j.bmcl.2005.09.056 BindingDB Entry DOI: 10.7270/Q2PG1SH8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50175765 (1-(4-amino-2,6-diisopropylphenyl)-3-(1-butyl-4-(3-...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 21 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Pharmaceuticals Co., Ltd Curated by ChEMBL | Assay Description Inhibitory activity against ACAT in rat macrophages | Bioorg Med Chem Lett 16: 44-8 (2005) Article DOI: 10.1016/j.bmcl.2005.09.056 BindingDB Entry DOI: 10.7270/Q2PG1SH8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50175775 (1-(3-amino-2,6-diisopropylphenyl)-3-(1-butyl-4-(3-...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 43 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Pharmaceuticals Co., Ltd Curated by ChEMBL | Assay Description Inhibitory activity against ACAT in rat macrophages | Bioorg Med Chem Lett 16: 44-8 (2005) Article DOI: 10.1016/j.bmcl.2005.09.056 BindingDB Entry DOI: 10.7270/Q2PG1SH8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50175773 (1-(4-amino-2,6-diisopropylphenyl)-3-(1-butyl-4-(3-...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 61 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Pharmaceuticals Co., Ltd Curated by ChEMBL | Assay Description Inhibitory activity against ACAT in rat macrophages | Bioorg Med Chem Lett 16: 44-8 (2005) Article DOI: 10.1016/j.bmcl.2005.09.056 BindingDB Entry DOI: 10.7270/Q2PG1SH8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50175769 (1-(4-(aminomethyl)-2,6-diisopropylphenyl)-3-(1-but...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 382 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Pharmaceuticals Co., Ltd Curated by ChEMBL | Assay Description Inhibitory activity against ACAT in rat macrophages | Bioorg Med Chem Lett 16: 44-8 (2005) Article DOI: 10.1016/j.bmcl.2005.09.056 BindingDB Entry DOI: 10.7270/Q2PG1SH8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50175768 (1-(4-amino-2,6-diisopropylphenyl)-3-(1-butyl-2-oxo...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 427 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Pharmaceuticals Co., Ltd Curated by ChEMBL | Assay Description Inhibitory activity against ACAT in rat macrophages | Bioorg Med Chem Lett 16: 44-8 (2005) Article DOI: 10.1016/j.bmcl.2005.09.056 BindingDB Entry DOI: 10.7270/Q2PG1SH8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50175764 (1-(4-amino-2,6-diisopropylphenyl)-3-(1-butyl-4-(3-...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 452 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Pharmaceuticals Co., Ltd Curated by ChEMBL | Assay Description Inhibitory activity against ACAT in rat macrophages | Bioorg Med Chem Lett 16: 44-8 (2005) Article DOI: 10.1016/j.bmcl.2005.09.056 BindingDB Entry DOI: 10.7270/Q2PG1SH8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50175763 (1-(4-amino-2,6-diisopropylphenyl)-3-(1-butyl-2-oxo...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 540 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Pharmaceuticals Co., Ltd Curated by ChEMBL | Assay Description Inhibitory activity against ACAT in rat macrophages | Bioorg Med Chem Lett 16: 44-8 (2005) Article DOI: 10.1016/j.bmcl.2005.09.056 BindingDB Entry DOI: 10.7270/Q2PG1SH8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50175774 (1-(1-butyl-4-(3-methoxyphenyl)-2-oxo-1,2-dihydro-1...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 680 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Pharmaceuticals Co., Ltd Curated by ChEMBL | Assay Description Inhibitory activity against ACAT in rat macrophages | Bioorg Med Chem Lett 16: 44-8 (2005) Article DOI: 10.1016/j.bmcl.2005.09.056 BindingDB Entry DOI: 10.7270/Q2PG1SH8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sterol O-acyltransferase 1 (Rattus norvegicus) | BDBM50175770 (1-(4-amino-2,6-diisopropylphenyl)-3-(1-butyl-4-(3-...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Pharmaceuticals Co., Ltd Curated by ChEMBL | Assay Description Inhibitory activity against ACAT in rat macrophages | Bioorg Med Chem Lett 16: 44-8 (2005) Article DOI: 10.1016/j.bmcl.2005.09.056 BindingDB Entry DOI: 10.7270/Q2PG1SH8 | |||||||||||
More data for this Ligand-Target Pair |