Affinity Data by PubMed id=16480267

PubMed code 16480267

Found 3 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Vitamin D3 receptor (Homo sapiens (Human))	BDBM50182484 ((1R,3R)-5-{2-[1-((1R,5S)-5-adamantan-1-yl-5-hydrox...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	50	n/a	n/a	n/a	n/a	n/a	n/a
Tokyo Medical and Dental University Curated by ChEMBL					Assay Description Antagonistic activity against human VDR in presence of 1,25(OH)2D3				J Med Chem 49: 1313-24 (2006) Article DOI: 10.1021/jm050795q BindingDB Entry DOI: 10.7270/Q23X867H
Tokyo Medical and Dental University Curated by ChEMBL					More data for this Ligand-Target Pair
Vitamin D3 receptor (Homo sapiens (Human))	BDBM50182485 ((S)-5-((R)-2-(4-(2-((3R,5R)-3,5-dihydroxy-4-methyl...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	300	n/a	n/a	n/a	n/a	n/a	n/a
Tokyo Medical and Dental University Curated by ChEMBL					Assay Description Inhibition of transactivation of human VDR in COS7 cells				J Med Chem 49: 1313-24 (2006) Article DOI: 10.1021/jm050795q BindingDB Entry DOI: 10.7270/Q23X867H
Tokyo Medical and Dental University Curated by ChEMBL					More data for this Ligand-Target Pair
Vitamin D3 receptor (Homo sapiens (Human))	BDBM50182484 ((1R,3R)-5-{2-[1-((1R,5S)-5-adamantan-1-yl-5-hydrox...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	400	n/a	n/a	n/a	n/a	n/a	n/a
Tokyo Medical and Dental University Curated by ChEMBL					Assay Description Inhibition of transactivation of human VDR in COS7 cells				J Med Chem 49: 1313-24 (2006) Article DOI: 10.1021/jm050795q BindingDB Entry DOI: 10.7270/Q23X867H
Tokyo Medical and Dental University Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%