Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Glucagon receptor (Homo sapiens (Human)) | BDBM50183179 (CHEMBL380387 | naphthalen-1-yl-[4-(3-pyrrolidin-1-...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Central Drug Research Institute Curated by ChEMBL | Assay Description Inhibition of [125I]glucagon binding to glucagon receptor | Bioorg Med Chem Lett 16: 2719-23 (2006) Article DOI: 10.1016/j.bmcl.2006.02.013 BindingDB Entry DOI: 10.7270/Q2NP2418 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50183180 (4-[2-(4-methoxybenzylamino-propoxy)-phenyl]-naphth...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Central Drug Research Institute Curated by ChEMBL | Assay Description Inhibition of [125I]glucagon binding to glucagon receptor | Bioorg Med Chem Lett 16: 2719-23 (2006) Article DOI: 10.1016/j.bmcl.2006.02.013 BindingDB Entry DOI: 10.7270/Q2NP2418 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50183181 (CHEMBL208053 | naphthalen-1-yl-[4-(2-pyrrolidin-1-...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Central Drug Research Institute Curated by ChEMBL | Assay Description Inhibition of [125I]glucagon binding to glucagon receptor | Bioorg Med Chem Lett 16: 2719-23 (2006) Article DOI: 10.1016/j.bmcl.2006.02.013 BindingDB Entry DOI: 10.7270/Q2NP2418 | |||||||||||
More data for this Ligand-Target Pair |