Affinity Data by PubMed id=16610788

PubMed code 16610788

Found 5 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Cholecystokinin receptor type A (Homo sapiens (Human))	BDBM50185261 (4-(3,4-dichlorobenzamido)-5-((3-methoxypropyl)(pen...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	195	n/a	n/a	n/a	n/a	n/a	n/a
University of Naples Federico II Curated by ChEMBL					Assay Description Displacement of [111In]-DTPAGlu-Gly-[Tyr27(SO3)]-CCK8 from human CCK1 receptor in A431 cells				J Med Chem 49: 2456-62 (2006) Article DOI: 10.1021/jm051050n BindingDB Entry DOI: 10.7270/Q2Q81CPS
University of Naples Federico II Curated by ChEMBL					More data for this Ligand-Target Pair
Cholecystokinin receptor type A (Homo sapiens (Human))	BDBM50185262 ((+/-)-2-(2-(1H-indole-2-carboxamido)benzamido)-3-p...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	197	n/a	n/a	n/a	n/a	n/a	n/a
University of Naples Federico II Curated by ChEMBL					Assay Description Displacement of [111In]-DTPAGlu-Gly-[Tyr27(SO3)]-CCK8 from human CCK1 receptor in A431 cells				J Med Chem 49: 2456-62 (2006) Article DOI: 10.1021/jm051050n BindingDB Entry DOI: 10.7270/Q2Q81CPS
University of Naples Federico II Curated by ChEMBL					More data for this Ligand-Target Pair
Cholecystokinin receptor type A (Homo sapiens (Human))	BDBM50185259 (2(R,S)-{2-[(1H-indole-2-carbonyl)amino]-benzoylami...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	2.80E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Naples Federico II Curated by ChEMBL					Assay Description Displacement of [111In]-DTPAGlu-Gly-[Tyr27(SO3)]-CCK8 from human CCK1 receptor in A431 cells				J Med Chem 49: 2456-62 (2006) Article DOI: 10.1021/jm051050n BindingDB Entry DOI: 10.7270/Q2Q81CPS
University of Naples Federico II Curated by ChEMBL					More data for this Ligand-Target Pair
Cholecystokinin receptor type A (Homo sapiens (Human))	BDBM50185260 ((+/-)-2-(2-cinnamamidobenzamido)-3-phenylpropanoic...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	4.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Naples Federico II Curated by ChEMBL					Assay Description Displacement of [111In]-DTPAGlu-Gly-[Tyr27(SO3)]-CCK8 from human CCK1 receptor in A431 cells				J Med Chem 49: 2456-62 (2006) Article DOI: 10.1021/jm051050n BindingDB Entry DOI: 10.7270/Q2Q81CPS
University of Naples Federico II Curated by ChEMBL					More data for this Ligand-Target Pair
Cholecystokinin receptor type A (Homo sapiens (Human))	BDBM50185263 (2(R,S)-{2-[(2-acetylaminocinnamoyl)amino]benzoylam...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.27E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Naples Federico II Curated by ChEMBL					Assay Description Displacement of [111In]-DTPAGlu-Gly-[Tyr27(SO3)]-CCK8 from human CCK1 receptor in A431 cells				J Med Chem 49: 2456-62 (2006) Article DOI: 10.1021/jm051050n BindingDB Entry DOI: 10.7270/Q2Q81CPS
University of Naples Federico II Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%