Affinity Data by PubMed id=16640328

PubMed code 16640328

Found 13 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Protein kinase C eta type (Homo sapiens (Human))	BDBM50185931 (8-Octyl-benzolactam-V9 \| CHEMBL206866) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	144	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Kyoto University Curated by ChEMBL					Assay Description Displacement of [3H]phorbol 12,13-dibutyrate from PKC eta-C1B				J Med Chem 49: 2681-8 (2006) Article DOI: 10.1021/jm050857c BindingDB Entry DOI: 10.7270/Q2BR8RSR
Kyoto University Curated by ChEMBL					More data for this Ligand-Target Pair
Protein kinase C delta type (Homo sapiens (Human))	BDBM50185931 (8-Octyl-benzolactam-V9 \| CHEMBL206866) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	216	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Kyoto University Curated by ChEMBL					Assay Description Displacement of [3H]phorbol 12,13-dibutyrate from PKC delta-C1B				J Med Chem 49: 2681-8 (2006) Article DOI: 10.1021/jm050857c BindingDB Entry DOI: 10.7270/Q2BR8RSR
Kyoto University Curated by ChEMBL					More data for this Ligand-Target Pair
Protein kinase C theta type (Homo sapiens (Human))	BDBM50185931 (8-Octyl-benzolactam-V9 \| CHEMBL206866) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	290	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Kyoto University Curated by ChEMBL					Assay Description Displacement of [3H]phorbol 12,13-dibutyrate from PKC theta-C1B				J Med Chem 49: 2681-8 (2006) Article DOI: 10.1021/jm050857c BindingDB Entry DOI: 10.7270/Q2BR8RSR
Kyoto University Curated by ChEMBL					More data for this Ligand-Target Pair
Protein kinase C epsilon type (Homo sapiens (Human))	BDBM50185931 (8-Octyl-benzolactam-V9 \| CHEMBL206866) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	510	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Kyoto University Curated by ChEMBL					Assay Description Displacement of [3H]phorbol 12,13-dibutyrate from PKC epsilon-C1B				J Med Chem 49: 2681-8 (2006) Article DOI: 10.1021/jm050857c BindingDB Entry DOI: 10.7270/Q2BR8RSR
Kyoto University Curated by ChEMBL					More data for this Ligand-Target Pair
Protein kinase C gamma type (Homo sapiens (Human))	BDBM50185931 (8-Octyl-benzolactam-V9 \| CHEMBL206866) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	5.20E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Kyoto University Curated by ChEMBL					Assay Description Displacement of [3H]phorbol 12,13-dibutyrate from PKC gamma-C1B				J Med Chem 49: 2681-8 (2006) Article DOI: 10.1021/jm050857c BindingDB Entry DOI: 10.7270/Q2BR8RSR
Kyoto University Curated by ChEMBL					More data for this Ligand-Target Pair
Protein kinase C alpha type (Homo sapiens (Human))	BDBM50185931 (8-Octyl-benzolactam-V9 \| CHEMBL206866) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Kyoto University Curated by ChEMBL					Assay Description Displacement of [3H]phorbol 12,13-dibutyrate from PKC alpha-C1A				J Med Chem 49: 2681-8 (2006) Article DOI: 10.1021/jm050857c BindingDB Entry DOI: 10.7270/Q2BR8RSR
Kyoto University Curated by ChEMBL					More data for this Ligand-Target Pair
Protein kinase C alpha type (Homo sapiens (Human))	BDBM50185931 (8-Octyl-benzolactam-V9 \| CHEMBL206866) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Kyoto University Curated by ChEMBL					Assay Description Displacement of [3H]phorbol 12,13-dibutyrate from PKC alpha-C1B				J Med Chem 49: 2681-8 (2006) Article DOI: 10.1021/jm050857c BindingDB Entry DOI: 10.7270/Q2BR8RSR
Kyoto University Curated by ChEMBL					More data for this Ligand-Target Pair
Protein kinase C beta type (Homo sapiens (Human))	BDBM50185931 (8-Octyl-benzolactam-V9 \| CHEMBL206866) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Kyoto University Curated by ChEMBL					Assay Description Displacement of [3H]phorbol 12,13-dibutyrate from PKC beta-C1A				J Med Chem 49: 2681-8 (2006) Article DOI: 10.1021/jm050857c BindingDB Entry DOI: 10.7270/Q2BR8RSR
Kyoto University Curated by ChEMBL					More data for this Ligand-Target Pair
Protein kinase C eta type (Homo sapiens (Human))	BDBM50185931 (8-Octyl-benzolactam-V9 \| CHEMBL206866) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Kyoto University Curated by ChEMBL					Assay Description Displacement of [3H]phorbol 12,13-dibutyrate from PKC eta-C1A				J Med Chem 49: 2681-8 (2006) Article DOI: 10.1021/jm050857c BindingDB Entry DOI: 10.7270/Q2BR8RSR
Kyoto University Curated by ChEMBL					More data for this Ligand-Target Pair
Protein kinase C gamma type (Homo sapiens (Human))	BDBM50185931 (8-Octyl-benzolactam-V9 \| CHEMBL206866) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Kyoto University Curated by ChEMBL					Assay Description Displacement of [3H]phorbol 12,13-dibutyrate from PKC gamma-C1A				J Med Chem 49: 2681-8 (2006) Article DOI: 10.1021/jm050857c BindingDB Entry DOI: 10.7270/Q2BR8RSR
Kyoto University Curated by ChEMBL					More data for this Ligand-Target Pair
Protein kinase C epsilon type (Homo sapiens (Human))	BDBM50185931 (8-Octyl-benzolactam-V9 \| CHEMBL206866) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Kyoto University Curated by ChEMBL					Assay Description Displacement of [3H]phorbol 12,13-dibutyrate from PKC epsilon-C1A				J Med Chem 49: 2681-8 (2006) Article DOI: 10.1021/jm050857c BindingDB Entry DOI: 10.7270/Q2BR8RSR
Kyoto University Curated by ChEMBL					More data for this Ligand-Target Pair
Protein kinase C delta type (Homo sapiens (Human))	BDBM50185931 (8-Octyl-benzolactam-V9 \| CHEMBL206866) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Kyoto University Curated by ChEMBL					Assay Description Displacement of [3H]phorbol 12,13-dibutyrate from PKC delta-C1A				J Med Chem 49: 2681-8 (2006) Article DOI: 10.1021/jm050857c BindingDB Entry DOI: 10.7270/Q2BR8RSR
Kyoto University Curated by ChEMBL					More data for this Ligand-Target Pair
Protein kinase C beta type (Homo sapiens (Human))	BDBM50185931 (8-Octyl-benzolactam-V9 \| CHEMBL206866) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Kyoto University Curated by ChEMBL					Assay Description Displacement of [3H]phorbol 12,13-dibutyrate from PKC beta-C1B				J Med Chem 49: 2681-8 (2006) Article DOI: 10.1021/jm050857c BindingDB Entry DOI: 10.7270/Q2BR8RSR
Kyoto University Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%