Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
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Vascular endothelial growth factor receptor 2 (Homo sapiens (Human)) | BDBM9503 (2-[(pyridin-4-ylmethyl)amino]-N-[3-(trifluoromethy...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | 31 | n/a | n/a | n/a | n/a | n/a | n/a |
Gakushuin University Curated by ChEMBL | Assay Description Inhibition of recombinant KDR at 1 uM by ELISA | Bioorg Med Chem Lett 16: 5127-31 (2006) Article DOI: 10.1016/j.bmcl.2006.07.075 BindingDB Entry DOI: 10.7270/Q2DJ5F8Q | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) |