Affinity Data by PubMed id=16970390

PubMed code 16970390

Found 6 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM17446 ((3R,4S,5S,6R)-5-methoxy-4-[(2R,3R)-2-methyl-3-(3-m...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL DrugBank MCE PC cid PC sid PDB UniChem Patents Similars	Article PubMed	n/a	n/a	1	n/a	n/a	n/a	n/a	n/a	n/a
The Johns Hopkins University School of Medicine Curated by ChEMBL					Assay Description Inhibition of human MetAP2				J Med Chem 49: 5645-8 (2006) Article DOI: 10.1021/jm060559v BindingDB Entry DOI: 10.7270/Q2PN959W
					More data for this Ligand-Target Pair				3D Structure (docked)
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM50194619 (6S-(1'R,2'R-1',5'-dimethyl-1',2'-oxiranyl-4'-hexen...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	3.23E+3	n/a	n/a	n/a	n/a	n/a	n/a
The Johns Hopkins University School of Medicine Curated by ChEMBL					Assay Description Inhibition of human MetAP2				J Med Chem 49: 5645-8 (2006) Article DOI: 10.1021/jm060559v BindingDB Entry DOI: 10.7270/Q2PN959W
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM50194620 ((1R,2S,3S)-1-hydroxy-3-methoxy-2-[(2R,3R)-2-methyl...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	8.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
The Johns Hopkins University School of Medicine Curated by ChEMBL					Assay Description Inhibition of human MetAP2				J Med Chem 49: 5645-8 (2006) Article DOI: 10.1021/jm060559v BindingDB Entry DOI: 10.7270/Q2PN959W
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM50194621 (6S-(1'R,2'R-1',5'-dimethyl-1',2'-oxiranyl-4'-hexen...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.32E+4	n/a	n/a	n/a	n/a	n/a	n/a
The Johns Hopkins University School of Medicine Curated by ChEMBL					Assay Description Inhibition of human MetAP2				J Med Chem 49: 5645-8 (2006) Article DOI: 10.1021/jm060559v BindingDB Entry DOI: 10.7270/Q2PN959W
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM50194623 ((1S,5S,6R,E)-5-(hydroxymethyl)-1-methoxy-6-(6-meth...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	3.38E+4	n/a	n/a	n/a	n/a	n/a	n/a
The Johns Hopkins University School of Medicine Curated by ChEMBL					Assay Description Inhibition of human MetAP2				J Med Chem 49: 5645-8 (2006) Article DOI: 10.1021/jm060559v BindingDB Entry DOI: 10.7270/Q2PN959W
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM50194622 ((1S,5S,6R)-5-(hydroxymethyl)-1-methoxy-6'-(6'-meth...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	5.75E+4	n/a	n/a	n/a	n/a	n/a	n/a
The Johns Hopkins University School of Medicine Curated by ChEMBL					Assay Description Inhibition of human MetAP2				J Med Chem 49: 5645-8 (2006) Article DOI: 10.1021/jm060559v BindingDB Entry DOI: 10.7270/Q2PN959W
					More data for this Ligand-Target Pair

* indicates data uncertainty>20%