Affinity Data by PubMed id=17055271

PubMed code 17055271

Found 18 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Dipeptidyl peptidase 4 (Homo sapiens (Human))	BDBM50050513 ((R)-1-((S)-2-amino-3-methylbutanoyl)pyrrolidin-2-y...) Show SMILES CC(C)[C@H](N)C(=O)N1CCC[C@H]1B(O)O \|r\| Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	0.100	n/a	n/a	n/a	n/a	n/a	n/a
Tufts University School of Medicine Curated by ChEMBL					Assay Description Inhibition of human DPP4				Bioorg Med Chem Lett 17: 507-10 (2007) Article DOI: 10.1016/j.bmcl.2006.10.012 BindingDB Entry DOI: 10.7270/Q2T43SQH
Tufts University School of Medicine Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50196928 ((R)-1-((S)-2,4-diaminobutanamido)pentylboronic aci...) Show SMILES CCCC[C@H](NC(=O)[C@@H](N)CCN)B(O)O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	0.480	n/a	n/a	n/a	n/a	n/a	n/a
Tufts University School of Medicine Curated by ChEMBL					Assay Description Inhibition of human DPP2				Bioorg Med Chem Lett 17: 507-10 (2007) Article DOI: 10.1016/j.bmcl.2006.10.012 BindingDB Entry DOI: 10.7270/Q2T43SQH
Tufts University School of Medicine Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50196929 ((S)-2,4-diamino-1-((3aR,6aR)-hexahydrocyclopenta[b...) Show SMILES NCC[C@H](N)C(=O)N1CC[C@H]2CCC[C@@H]12 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	0.880	n/a	n/a	n/a	n/a	n/a	n/a
Tufts University School of Medicine Curated by ChEMBL					Assay Description Inhibition of human DPP2				Bioorg Med Chem Lett 17: 507-10 (2007) Article DOI: 10.1016/j.bmcl.2006.10.012 BindingDB Entry DOI: 10.7270/Q2T43SQH
Tufts University School of Medicine Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 9 (Homo sapiens (Human))	BDBM50050513 ((R)-1-((S)-2-amino-3-methylbutanoyl)pyrrolidin-2-y...) Show SMILES CC(C)[C@H](N)C(=O)N1CCC[C@H]1B(O)O \|r\| Show InChI	PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	2	n/a	n/a	n/a	n/a	n/a	n/a
Tufts University School of Medicine Curated by ChEMBL					Assay Description Inhibition of human DPP9				Bioorg Med Chem Lett 17: 507-10 (2007) Article DOI: 10.1016/j.bmcl.2006.10.012 BindingDB Entry DOI: 10.7270/Q2T43SQH
Tufts University School of Medicine Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 8 (Homo sapiens (Human))	BDBM50050513 ((R)-1-((S)-2-amino-3-methylbutanoyl)pyrrolidin-2-y...) Show SMILES CC(C)[C@H](N)C(=O)N1CCC[C@H]1B(O)O \|r\| Show InChI	PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	17	n/a	n/a	n/a	n/a	n/a	n/a
Tufts University School of Medicine Curated by ChEMBL					Assay Description Inhibition of human DPP8				Bioorg Med Chem Lett 17: 507-10 (2007) Article DOI: 10.1016/j.bmcl.2006.10.012 BindingDB Entry DOI: 10.7270/Q2T43SQH
Tufts University School of Medicine Curated by ChEMBL					More data for this Ligand-Target Pair
Prolyl endopeptidase FAP (Homo sapiens (Human))	BDBM50050513 ((R)-1-((S)-2-amino-3-methylbutanoyl)pyrrolidin-2-y...) Show SMILES CC(C)[C@H](N)C(=O)N1CCC[C@H]1B(O)O \|r\| Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	24	n/a	n/a	n/a	n/a	n/a	n/a
Tufts University School of Medicine Curated by ChEMBL					Assay Description Inhibition of human FAP				Bioorg Med Chem Lett 17: 507-10 (2007) Article DOI: 10.1016/j.bmcl.2006.10.012 BindingDB Entry DOI: 10.7270/Q2T43SQH
Tufts University School of Medicine Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50050513 ((R)-1-((S)-2-amino-3-methylbutanoyl)pyrrolidin-2-y...) Show SMILES CC(C)[C@H](N)C(=O)N1CCC[C@H]1B(O)O \|r\| Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	30	n/a	n/a	n/a	n/a	n/a	n/a
Tufts University School of Medicine Curated by ChEMBL					Assay Description Inhibition of human DPP2				Bioorg Med Chem Lett 17: 507-10 (2007) Article DOI: 10.1016/j.bmcl.2006.10.012 BindingDB Entry DOI: 10.7270/Q2T43SQH
Tufts University School of Medicine Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 9 (Homo sapiens (Human))	BDBM50196928 ((R)-1-((S)-2,4-diaminobutanamido)pentylboronic aci...) Show SMILES CCCC[C@H](NC(=O)[C@@H](N)CCN)B(O)O Show InChI	PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	800	n/a	n/a	n/a	n/a	n/a	n/a
Tufts University School of Medicine Curated by ChEMBL					Assay Description Inhibition of human DPP9				Bioorg Med Chem Lett 17: 507-10 (2007) Article DOI: 10.1016/j.bmcl.2006.10.012 BindingDB Entry DOI: 10.7270/Q2T43SQH
Tufts University School of Medicine Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 8 (Homo sapiens (Human))	BDBM50196928 ((R)-1-((S)-2,4-diaminobutanamido)pentylboronic aci...) Show SMILES CCCC[C@H](NC(=O)[C@@H](N)CCN)B(O)O Show InChI	PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	4.30E+3	n/a	n/a	n/a	n/a	n/a	n/a
Tufts University School of Medicine Curated by ChEMBL					Assay Description Inhibition of human DPP8				Bioorg Med Chem Lett 17: 507-10 (2007) Article DOI: 10.1016/j.bmcl.2006.10.012 BindingDB Entry DOI: 10.7270/Q2T43SQH
Tufts University School of Medicine Curated by ChEMBL					More data for this Ligand-Target Pair
Prolyl endopeptidase (Homo sapiens (Human))	BDBM50050513 ((R)-1-((S)-2-amino-3-methylbutanoyl)pyrrolidin-2-y...) Show SMILES CC(C)[C@H](N)C(=O)N1CCC[C@H]1B(O)O \|r\| Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	7.96E+3	n/a	n/a	n/a	n/a	n/a	n/a
Tufts University School of Medicine Curated by ChEMBL					Assay Description Inhibition of prolyl oligopeptidase				Bioorg Med Chem Lett 17: 507-10 (2007) Article DOI: 10.1016/j.bmcl.2006.10.012 BindingDB Entry DOI: 10.7270/Q2T43SQH
Tufts University School of Medicine Curated by ChEMBL					More data for this Ligand-Target Pair
Prolyl endopeptidase (Homo sapiens (Human))	BDBM50196929 ((S)-2,4-diamino-1-((3aR,6aR)-hexahydrocyclopenta[b...) Show SMILES NCC[C@H](N)C(=O)N1CC[C@H]2CCC[C@@H]12 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>2.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
Tufts University School of Medicine Curated by ChEMBL					Assay Description Inhibition of prolyl oligopeptidase				Bioorg Med Chem Lett 17: 507-10 (2007) Article DOI: 10.1016/j.bmcl.2006.10.012 BindingDB Entry DOI: 10.7270/Q2T43SQH
Tufts University School of Medicine Curated by ChEMBL					More data for this Ligand-Target Pair
Prolyl endopeptidase (Homo sapiens (Human))	BDBM50196928 ((R)-1-((S)-2,4-diaminobutanamido)pentylboronic aci...) Show SMILES CCCC[C@H](NC(=O)[C@@H](N)CCN)B(O)O Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>2.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
Tufts University School of Medicine Curated by ChEMBL					Assay Description Inhibition of prolyl oligopeptidase				Bioorg Med Chem Lett 17: 507-10 (2007) Article DOI: 10.1016/j.bmcl.2006.10.012 BindingDB Entry DOI: 10.7270/Q2T43SQH
Tufts University School of Medicine Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 8 (Homo sapiens (Human))	BDBM50196929 ((S)-2,4-diamino-1-((3aR,6aR)-hexahydrocyclopenta[b...) Show SMILES NCC[C@H](N)C(=O)N1CC[C@H]2CCC[C@@H]12 Show InChI	PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>2.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
Tufts University School of Medicine Curated by ChEMBL					Assay Description Inhibition of human DPP8				Bioorg Med Chem Lett 17: 507-10 (2007) Article DOI: 10.1016/j.bmcl.2006.10.012 BindingDB Entry DOI: 10.7270/Q2T43SQH
Tufts University School of Medicine Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 9 (Homo sapiens (Human))	BDBM50196929 ((S)-2,4-diamino-1-((3aR,6aR)-hexahydrocyclopenta[b...) Show SMILES NCC[C@H](N)C(=O)N1CC[C@H]2CCC[C@@H]12 Show InChI	PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>2.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
Tufts University School of Medicine Curated by ChEMBL					Assay Description Inhibition of human DPP9				Bioorg Med Chem Lett 17: 507-10 (2007) Article DOI: 10.1016/j.bmcl.2006.10.012 BindingDB Entry DOI: 10.7270/Q2T43SQH
Tufts University School of Medicine Curated by ChEMBL					More data for this Ligand-Target Pair
Prolyl endopeptidase FAP (Homo sapiens (Human))	BDBM50196929 ((S)-2,4-diamino-1-((3aR,6aR)-hexahydrocyclopenta[b...) Show SMILES NCC[C@H](N)C(=O)N1CC[C@H]2CCC[C@@H]12 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>3.30E+4	n/a	n/a	n/a	n/a	n/a	n/a
Tufts University School of Medicine Curated by ChEMBL					Assay Description Inhibition of human FAP				Bioorg Med Chem Lett 17: 507-10 (2007) Article DOI: 10.1016/j.bmcl.2006.10.012 BindingDB Entry DOI: 10.7270/Q2T43SQH
Tufts University School of Medicine Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 4 (Homo sapiens (Human))	BDBM50196928 ((R)-1-((S)-2,4-diaminobutanamido)pentylboronic aci...) Show SMILES CCCC[C@H](NC(=O)[C@@H](N)CCN)B(O)O Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>3.30E+4	n/a	n/a	n/a	n/a	n/a	n/a
Tufts University School of Medicine Curated by ChEMBL					Assay Description Inhibition of human DPP4				Bioorg Med Chem Lett 17: 507-10 (2007) Article DOI: 10.1016/j.bmcl.2006.10.012 BindingDB Entry DOI: 10.7270/Q2T43SQH
Tufts University School of Medicine Curated by ChEMBL					More data for this Ligand-Target Pair
Prolyl endopeptidase FAP (Homo sapiens (Human))	BDBM50196928 ((R)-1-((S)-2,4-diaminobutanamido)pentylboronic aci...) Show SMILES CCCC[C@H](NC(=O)[C@@H](N)CCN)B(O)O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>3.30E+4	n/a	n/a	n/a	n/a	n/a	n/a
Tufts University School of Medicine Curated by ChEMBL					Assay Description Inhibition of human FAP				Bioorg Med Chem Lett 17: 507-10 (2007) Article DOI: 10.1016/j.bmcl.2006.10.012 BindingDB Entry DOI: 10.7270/Q2T43SQH
Tufts University School of Medicine Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 4 (Homo sapiens (Human))	BDBM50196929 ((S)-2,4-diamino-1-((3aR,6aR)-hexahydrocyclopenta[b...) Show SMILES NCC[C@H](N)C(=O)N1CC[C@H]2CCC[C@@H]12 Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>3.30E+4	n/a	n/a	n/a	n/a	n/a	n/a
Tufts University School of Medicine Curated by ChEMBL					Assay Description Inhibition of human DPP4				Bioorg Med Chem Lett 17: 507-10 (2007) Article DOI: 10.1016/j.bmcl.2006.10.012 BindingDB Entry DOI: 10.7270/Q2T43SQH
Tufts University School of Medicine Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%