Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50207909 (CHEMBL239805 | N-(3-(4-ethylphenylsulfonamido)-2,3...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 150 | n/a | n/a | n/a | n/a | n/a | n/a |
Icagen Inc. Curated by ChEMBL | Assay Description Inhibition of Kv1.5 channel mediated delayed rectifier potassium current by patch-clamp technique | Bioorg Med Chem Lett 17: 2849-53 (2007) Article DOI: 10.1016/j.bmcl.2007.02.052 BindingDB Entry DOI: 10.7270/Q2VM4BZS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50099581 (CHEMBL288131 | N-((2R,3R)-3-(4-ethylphenylsulfonam...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 160 | n/a | n/a | n/a | n/a | n/a | n/a |
Icagen Inc. Curated by ChEMBL | Assay Description Inhibition of Kv1.5 channel mediated delayed rectifier potassium current by patch-clamp technique | Bioorg Med Chem Lett 17: 2849-53 (2007) Article DOI: 10.1016/j.bmcl.2007.02.052 BindingDB Entry DOI: 10.7270/Q2VM4BZS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50099581 (CHEMBL288131 | N-((2R,3R)-3-(4-ethylphenylsulfonam...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 160 | n/a | n/a | n/a | n/a | n/a | n/a |
Icagen Inc. Curated by ChEMBL | Assay Description Inhibition of Kv1.5 channel mediated delayed rectifier potassium current by patch-clamp technique | Bioorg Med Chem Lett 17: 2849-53 (2007) Article DOI: 10.1016/j.bmcl.2007.02.052 BindingDB Entry DOI: 10.7270/Q2VM4BZS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50207912 (CHEMBL239808 | N-((8R,9R)-9-(4-ethylphenylsulfonam...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
Icagen Inc. Curated by ChEMBL | Assay Description Inhibition of Kv1.5 channel mediated delayed rectifier potassium current by patch-clamp technique | Bioorg Med Chem Lett 17: 2849-53 (2007) Article DOI: 10.1016/j.bmcl.2007.02.052 BindingDB Entry DOI: 10.7270/Q2VM4BZS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50207906 (CHEMBL241513 | N-(3-((4-ethylphenylsulfonamido)met...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 240 | n/a | n/a | n/a | n/a | n/a | n/a |
Icagen Inc. Curated by ChEMBL | Assay Description Inhibition of Kv1.5 channel mediated delayed rectifier potassium current by patch-clamp technique | Bioorg Med Chem Lett 17: 2849-53 (2007) Article DOI: 10.1016/j.bmcl.2007.02.052 BindingDB Entry DOI: 10.7270/Q2VM4BZS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50207911 (CHEMBL398397 | N-((2S,3R)-3-(4-ethylphenylsulfonam...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 300 | n/a | n/a | n/a | n/a | n/a | n/a |
Icagen Inc. Curated by ChEMBL | Assay Description Inhibition of Kv1.5 channel mediated delayed rectifier potassium current by patch-clamp technique | Bioorg Med Chem Lett 17: 2849-53 (2007) Article DOI: 10.1016/j.bmcl.2007.02.052 BindingDB Entry DOI: 10.7270/Q2VM4BZS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50207907 (CHEMBL239807 | N-((7R,8R)-8-(4-ethylphenylsulfonam...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 440 | n/a | n/a | n/a | n/a | n/a | n/a |
Icagen Inc. Curated by ChEMBL | Assay Description Inhibition of Kv1.5 channel mediated delayed rectifier potassium current by patch-clamp technique | Bioorg Med Chem Lett 17: 2849-53 (2007) Article DOI: 10.1016/j.bmcl.2007.02.052 BindingDB Entry DOI: 10.7270/Q2VM4BZS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50207908 (CHEMBL391455 | N-((2S,3S)-3-(4-ethylphenylsulfonam...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 760 | n/a | n/a | n/a | n/a | n/a | n/a |
Icagen Inc. Curated by ChEMBL | Assay Description Inhibition of Kv1.5 channel mediated delayed rectifier potassium current by patch-clamp technique | Bioorg Med Chem Lett 17: 2849-53 (2007) Article DOI: 10.1016/j.bmcl.2007.02.052 BindingDB Entry DOI: 10.7270/Q2VM4BZS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50207910 (CHEMBL391488 | N-((2R,3R)-3-(4-ethylphenylsulfonam...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 880 | n/a | n/a | n/a | n/a | n/a | n/a |
Icagen Inc. Curated by ChEMBL | Assay Description Inhibition of Kv1.5 channel mediated delayed rectifier potassium current by patch-clamp technique | Bioorg Med Chem Lett 17: 2849-53 (2007) Article DOI: 10.1016/j.bmcl.2007.02.052 BindingDB Entry DOI: 10.7270/Q2VM4BZS | |||||||||||
More data for this Ligand-Target Pair |