Search and Browse
Download
Enter Data
| Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Peroxisome proliferator-activated receptor alpha (Homo sapiens (Human)) | BDBM28661 (2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet  | Purchase CHEMBL DrugBank MCE PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a |
Johnson & Johnson Pharmaceutical | Assay Description The HEK293 cells were co-transfected with DNA constructs containing the ligand-binding domain of PPAR and Gal4-luciferase reporter. The luciferase ac... | J Med Chem 50: 3954-63 (2007) Article DOI: 10.1021/jm070511x BindingDB Entry DOI: 10.7270/Q2H41PR5 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Peroxisome proliferator-activated receptor gamma (Homo sapiens (Human)) | BDBM28756 (2-methyl-2-[2-methyl-4-({3-[4-(trifluoromethyl)phe...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | >3.00E+3 | n/a | n/a | n/a | n/a |
Johnson & Johnson Pharmaceutical | Assay Description The HEK293 cells were co-transfected with DNA constructs containing the ligand-binding domain of PPAR and Gal4-luciferase reporter. The luciferase ac... | J Med Chem 50: 3954-63 (2007) Article DOI: 10.1021/jm070511x BindingDB Entry DOI: 10.7270/Q2H41PR5 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Peroxisome proliferator-activated receptor gamma (Homo sapiens (Human)) | BDBM28757 (2-methyl-2-[2-methyl-4-({3-[4-(trifluoromethoxy)ph...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | >3.00E+3 | n/a | n/a | n/a | n/a |
Johnson & Johnson Pharmaceutical | Assay Description The HEK293 cells were co-transfected with DNA constructs containing the ligand-binding domain of PPAR and Gal4-luciferase reporter. The luciferase ac... | J Med Chem 50: 3954-63 (2007) Article DOI: 10.1021/jm070511x BindingDB Entry DOI: 10.7270/Q2H41PR5 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Peroxisome proliferator-activated receptor gamma (Homo sapiens (Human)) | BDBM28661 (2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 850 | n/a | n/a | n/a | n/a |
Johnson & Johnson Pharmaceutical | Assay Description The HEK293 cells were co-transfected with DNA constructs containing the ligand-binding domain of PPAR and Gal4-luciferase reporter. The luciferase ac... | J Med Chem 50: 3954-63 (2007) Article DOI: 10.1021/jm070511x BindingDB Entry DOI: 10.7270/Q2H41PR5 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Peroxisome proliferator-activated receptor delta (Homo sapiens (Human)) | BDBM28749 (2-{2-methyl-4-[({3-[4-(trifluoromethyl)phenyl]-1,2...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 10 | n/a | n/a | n/a | n/a |
Johnson & Johnson Pharmaceutical | Assay Description The confluent HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The lucif... | J Med Chem 50: 3954-63 (2007) Article DOI: 10.1021/jm070511x BindingDB Entry DOI: 10.7270/Q2H41PR5 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Peroxisome proliferator-activated receptor delta (Homo sapiens (Human)) | BDBM28661 (2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid PDB UniChem Patents Similars | PDB Article PubMed | n/a | n/a | n/a | n/a | 1 | n/a | n/a | n/a | n/a |
Johnson & Johnson Pharmaceutical | Assay Description The confluent HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The lucif... | J Med Chem 50: 3954-63 (2007) Article DOI: 10.1021/jm070511x BindingDB Entry DOI: 10.7270/Q2H41PR5 | |||||||||||
| More data for this Ligand-Target Pair |  3D Structure (crystal) | ||||||||||||
| Peroxisome proliferator-activated receptor alpha (Homo sapiens (Human)) | BDBM28751 (2-methyl-2-{2-methyl-4-[({3-[4-(trifluoromethoxy)p...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 33 | n/a | n/a | n/a | n/a |
Johnson & Johnson Pharmaceutical | Assay Description The HEK293 cells were co-transfected with DNA constructs containing the ligand-binding domain of PPAR and Gal4-luciferase reporter. The luciferase ac... | J Med Chem 50: 3954-63 (2007) Article DOI: 10.1021/jm070511x BindingDB Entry DOI: 10.7270/Q2H41PR5 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Peroxisome proliferator-activated receptor gamma (Homo sapiens (Human)) | BDBM28750 (2-methyl-2-{2-methyl-4-[({3-[4-(trifluoromethyl)ph...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 407 | n/a | n/a | n/a | n/a |
Johnson & Johnson Pharmaceutical | Assay Description The HEK293 cells were co-transfected with DNA constructs containing the ligand-binding domain of PPAR and Gal4-luciferase reporter. The luciferase ac... | J Med Chem 50: 3954-63 (2007) Article DOI: 10.1021/jm070511x BindingDB Entry DOI: 10.7270/Q2H41PR5 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Peroxisome proliferator-activated receptor gamma (Homo sapiens (Human)) | BDBM28753 (2-[4-({[3-(4-tert-butylphenyl)-1,2,4-thiadiazol-5-...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | >3.00E+3 | n/a | n/a | n/a | n/a |
Johnson & Johnson Pharmaceutical | Assay Description The HEK293 cells were co-transfected with DNA constructs containing the ligand-binding domain of PPAR and Gal4-luciferase reporter. The luciferase ac... | J Med Chem 50: 3954-63 (2007) Article DOI: 10.1021/jm070511x BindingDB Entry DOI: 10.7270/Q2H41PR5 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Peroxisome proliferator-activated receptor delta (Homo sapiens (Human)) | BDBM28756 (2-methyl-2-[2-methyl-4-({3-[4-(trifluoromethyl)phe...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 3 | n/a | n/a | n/a | n/a |
Johnson & Johnson Pharmaceutical | Assay Description The confluent HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The lucif... | J Med Chem 50: 3954-63 (2007) Article DOI: 10.1021/jm070511x BindingDB Entry DOI: 10.7270/Q2H41PR5 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Peroxisome proliferator-activated receptor alpha (Homo sapiens (Human)) | BDBM28754 (2-methyl-2-{2-methyl-4-[({5-[4-(trifluoromethyl)ph...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 425 | n/a | n/a | n/a | n/a |
Johnson & Johnson Pharmaceutical | Assay Description The HEK293 cells were co-transfected with DNA constructs containing the ligand-binding domain of PPAR and Gal4-luciferase reporter. The luciferase ac... | J Med Chem 50: 3954-63 (2007) Article DOI: 10.1021/jm070511x BindingDB Entry DOI: 10.7270/Q2H41PR5 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Peroxisome proliferator-activated receptor gamma (Homo sapiens (Human)) | BDBM28749 (2-{2-methyl-4-[({3-[4-(trifluoromethyl)phenyl]-1,2...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | >3.00E+3 | n/a | n/a | n/a | n/a |
Johnson & Johnson Pharmaceutical | Assay Description The HEK293 cells were co-transfected with DNA constructs containing the ligand-binding domain of PPAR and Gal4-luciferase reporter. The luciferase ac... | J Med Chem 50: 3954-63 (2007) Article DOI: 10.1021/jm070511x BindingDB Entry DOI: 10.7270/Q2H41PR5 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Peroxisome proliferator-activated receptor gamma (Homo sapiens (Human)) | BDBM28755 (2-methyl-2-{2-methyl-4-[({5-[4-(trifluoromethoxy)p...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | >3.00E+3 | n/a | n/a | n/a | n/a |
Johnson & Johnson Pharmaceutical | Assay Description The HEK293 cells were co-transfected with DNA constructs containing the ligand-binding domain of PPAR and Gal4-luciferase reporter. The luciferase ac... | J Med Chem 50: 3954-63 (2007) Article DOI: 10.1021/jm070511x BindingDB Entry DOI: 10.7270/Q2H41PR5 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Peroxisome proliferator-activated receptor delta (Homo sapiens (Human)) | BDBM28755 (2-methyl-2-{2-methyl-4-[({5-[4-(trifluoromethoxy)p...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 58 | n/a | n/a | n/a | n/a |
Johnson & Johnson Pharmaceutical | Assay Description The confluent HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The lucif... | J Med Chem 50: 3954-63 (2007) Article DOI: 10.1021/jm070511x BindingDB Entry DOI: 10.7270/Q2H41PR5 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Peroxisome proliferator-activated receptor delta (Homo sapiens (Human)) | BDBM28757 (2-methyl-2-[2-methyl-4-({3-[4-(trifluoromethoxy)ph...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 12 | n/a | n/a | n/a | n/a |
Johnson & Johnson Pharmaceutical | Assay Description The confluent HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The lucif... | J Med Chem 50: 3954-63 (2007) Article DOI: 10.1021/jm070511x BindingDB Entry DOI: 10.7270/Q2H41PR5 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Peroxisome proliferator-activated receptor gamma (Homo sapiens (Human)) | BDBM28754 (2-methyl-2-{2-methyl-4-[({5-[4-(trifluoromethyl)ph...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | >3.00E+3 | n/a | n/a | n/a | n/a |
Johnson & Johnson Pharmaceutical | Assay Description The HEK293 cells were co-transfected with DNA constructs containing the ligand-binding domain of PPAR and Gal4-luciferase reporter. The luciferase ac... | J Med Chem 50: 3954-63 (2007) Article DOI: 10.1021/jm070511x BindingDB Entry DOI: 10.7270/Q2H41PR5 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Peroxisome proliferator-activated receptor delta (Homo sapiens (Human)) | BDBM28751 (2-methyl-2-{2-methyl-4-[({3-[4-(trifluoromethoxy)p...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 3 | n/a | n/a | n/a | n/a |
Johnson & Johnson Pharmaceutical | Assay Description The confluent HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The lucif... | J Med Chem 50: 3954-63 (2007) Article DOI: 10.1021/jm070511x BindingDB Entry DOI: 10.7270/Q2H41PR5 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Peroxisome proliferator-activated receptor alpha (Homo sapiens (Human)) | BDBM28755 (2-methyl-2-{2-methyl-4-[({5-[4-(trifluoromethoxy)p...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 656 | n/a | n/a | n/a | n/a |
Johnson & Johnson Pharmaceutical | Assay Description The HEK293 cells were co-transfected with DNA constructs containing the ligand-binding domain of PPAR and Gal4-luciferase reporter. The luciferase ac... | J Med Chem 50: 3954-63 (2007) Article DOI: 10.1021/jm070511x BindingDB Entry DOI: 10.7270/Q2H41PR5 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Peroxisome proliferator-activated receptor alpha (Homo sapiens (Human)) | BDBM28757 (2-methyl-2-[2-methyl-4-({3-[4-(trifluoromethoxy)ph...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 94 | n/a | n/a | n/a | n/a |
Johnson & Johnson Pharmaceutical | Assay Description The HEK293 cells were co-transfected with DNA constructs containing the ligand-binding domain of PPAR and Gal4-luciferase reporter. The luciferase ac... | J Med Chem 50: 3954-63 (2007) Article DOI: 10.1021/jm070511x BindingDB Entry DOI: 10.7270/Q2H41PR5 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Peroxisome proliferator-activated receptor alpha (Homo sapiens (Human)) | BDBM28758 (1-{2-methyl-4-[({3-[4-(trifluoromethoxy)phenyl]-1,...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 736 | n/a | n/a | n/a | n/a |
Johnson & Johnson Pharmaceutical | Assay Description The HEK293 cells were co-transfected with DNA constructs containing the ligand-binding domain of PPAR and Gal4-luciferase reporter. The luciferase ac... | J Med Chem 50: 3954-63 (2007) Article DOI: 10.1021/jm070511x BindingDB Entry DOI: 10.7270/Q2H41PR5 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Peroxisome proliferator-activated receptor gamma (Homo sapiens (Human)) | BDBM28758 (1-{2-methyl-4-[({3-[4-(trifluoromethoxy)phenyl]-1,...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | >3.00E+3 | n/a | n/a | n/a | n/a |
Johnson & Johnson Pharmaceutical | Assay Description The HEK293 cells were co-transfected with DNA constructs containing the ligand-binding domain of PPAR and Gal4-luciferase reporter. The luciferase ac... | J Med Chem 50: 3954-63 (2007) Article DOI: 10.1021/jm070511x BindingDB Entry DOI: 10.7270/Q2H41PR5 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Peroxisome proliferator-activated receptor delta (Homo sapiens (Human)) | BDBM28752 (2-[4-({[3-(4-chlorophenyl)-1,2,4-thiadiazol-5-yl]m...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 18 | n/a | n/a | n/a | n/a |
Johnson & Johnson Pharmaceutical | Assay Description The confluent HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The lucif... | J Med Chem 50: 3954-63 (2007) Article DOI: 10.1021/jm070511x BindingDB Entry DOI: 10.7270/Q2H41PR5 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Peroxisome proliferator-activated receptor delta (Homo sapiens (Human)) | BDBM28753 (2-[4-({[3-(4-tert-butylphenyl)-1,2,4-thiadiazol-5-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 93 | n/a | n/a | n/a | n/a |
Johnson & Johnson Pharmaceutical | Assay Description The confluent HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The lucif... | J Med Chem 50: 3954-63 (2007) Article DOI: 10.1021/jm070511x BindingDB Entry DOI: 10.7270/Q2H41PR5 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Peroxisome proliferator-activated receptor alpha (Homo sapiens (Human)) | BDBM28750 (2-methyl-2-{2-methyl-4-[({3-[4-(trifluoromethyl)ph...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 79 | n/a | n/a | n/a | n/a |
Johnson & Johnson Pharmaceutical | Assay Description The HEK293 cells were co-transfected with DNA constructs containing the ligand-binding domain of PPAR and Gal4-luciferase reporter. The luciferase ac... | J Med Chem 50: 3954-63 (2007) Article DOI: 10.1021/jm070511x BindingDB Entry DOI: 10.7270/Q2H41PR5 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Peroxisome proliferator-activated receptor alpha (Homo sapiens (Human)) | BDBM28756 (2-methyl-2-[2-methyl-4-({3-[4-(trifluoromethyl)phe...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 94 | n/a | n/a | n/a | n/a |
Johnson & Johnson Pharmaceutical | Assay Description The HEK293 cells were co-transfected with DNA constructs containing the ligand-binding domain of PPAR and Gal4-luciferase reporter. The luciferase ac... | J Med Chem 50: 3954-63 (2007) Article DOI: 10.1021/jm070511x BindingDB Entry DOI: 10.7270/Q2H41PR5 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Peroxisome proliferator-activated receptor gamma (Homo sapiens (Human)) | BDBM28751 (2-methyl-2-{2-methyl-4-[({3-[4-(trifluoromethoxy)p...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | >3.00E+3 | n/a | n/a | n/a | n/a |
Johnson & Johnson Pharmaceutical | Assay Description The HEK293 cells were co-transfected with DNA constructs containing the ligand-binding domain of PPAR and Gal4-luciferase reporter. The luciferase ac... | J Med Chem 50: 3954-63 (2007) Article DOI: 10.1021/jm070511x BindingDB Entry DOI: 10.7270/Q2H41PR5 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Peroxisome proliferator-activated receptor delta (Homo sapiens (Human)) | BDBM28754 (2-methyl-2-{2-methyl-4-[({5-[4-(trifluoromethyl)ph...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 26 | n/a | n/a | n/a | n/a |
Johnson & Johnson Pharmaceutical | Assay Description The confluent HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The lucif... | J Med Chem 50: 3954-63 (2007) Article DOI: 10.1021/jm070511x BindingDB Entry DOI: 10.7270/Q2H41PR5 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Peroxisome proliferator-activated receptor alpha (Homo sapiens (Human)) | BDBM28752 (2-[4-({[3-(4-chlorophenyl)-1,2,4-thiadiazol-5-yl]m...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 186 | n/a | n/a | n/a | n/a |
Johnson & Johnson Pharmaceutical | Assay Description The HEK293 cells were co-transfected with DNA constructs containing the ligand-binding domain of PPAR and Gal4-luciferase reporter. The luciferase ac... | J Med Chem 50: 3954-63 (2007) Article DOI: 10.1021/jm070511x BindingDB Entry DOI: 10.7270/Q2H41PR5 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Peroxisome proliferator-activated receptor delta (Homo sapiens (Human)) | BDBM28750 (2-methyl-2-{2-methyl-4-[({3-[4-(trifluoromethyl)ph...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 6 | n/a | n/a | n/a | n/a |
Johnson & Johnson Pharmaceutical | Assay Description The confluent HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The lucif... | J Med Chem 50: 3954-63 (2007) Article DOI: 10.1021/jm070511x BindingDB Entry DOI: 10.7270/Q2H41PR5 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Peroxisome proliferator-activated receptor delta (Homo sapiens (Human)) | BDBM28758 (1-{2-methyl-4-[({3-[4-(trifluoromethoxy)phenyl]-1,...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a |
Johnson & Johnson Pharmaceutical | Assay Description The confluent HEK293 cells were co-transfected with DNA construct containing PPARdelta-Gal4 chimeric receptor and Gal4-luciferase reporter. The lucif... | J Med Chem 50: 3954-63 (2007) Article DOI: 10.1021/jm070511x BindingDB Entry DOI: 10.7270/Q2H41PR5 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Peroxisome proliferator-activated receptor alpha (Homo sapiens (Human)) | BDBM28749 (2-{2-methyl-4-[({3-[4-(trifluoromethyl)phenyl]-1,2...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 468 | n/a | n/a | n/a | n/a |
Johnson & Johnson Pharmaceutical | Assay Description The HEK293 cells were co-transfected with DNA constructs containing the ligand-binding domain of PPAR and Gal4-luciferase reporter. The luciferase ac... | J Med Chem 50: 3954-63 (2007) Article DOI: 10.1021/jm070511x BindingDB Entry DOI: 10.7270/Q2H41PR5 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Peroxisome proliferator-activated receptor alpha (Homo sapiens (Human)) | BDBM28753 (2-[4-({[3-(4-tert-butylphenyl)-1,2,4-thiadiazol-5-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 64 | n/a | n/a | n/a | n/a |
Johnson & Johnson Pharmaceutical | Assay Description The HEK293 cells were co-transfected with DNA constructs containing the ligand-binding domain of PPAR and Gal4-luciferase reporter. The luciferase ac... | J Med Chem 50: 3954-63 (2007) Article DOI: 10.1021/jm070511x BindingDB Entry DOI: 10.7270/Q2H41PR5 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Peroxisome proliferator-activated receptor gamma (Homo sapiens (Human)) | BDBM28752 (2-[4-({[3-(4-chlorophenyl)-1,2,4-thiadiazol-5-yl]m...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | >3.00E+3 | n/a | n/a | n/a | n/a |
Johnson & Johnson Pharmaceutical | Assay Description The HEK293 cells were co-transfected with DNA constructs containing the ligand-binding domain of PPAR and Gal4-luciferase reporter. The luciferase ac... | J Med Chem 50: 3954-63 (2007) Article DOI: 10.1021/jm070511x BindingDB Entry DOI: 10.7270/Q2H41PR5 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
