Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
CAAX prenyl protease 1 homolog (Mus musculus) | BDBM558 (N-{3-[(1R)-1-[(6R)-4-hydroxy-2-oxo-6-(2-phenylethy...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | MMDB PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description Inhibition of mouse ZMPSTE24 expressed n delta ste24 delta rce1 yeast | Proc Natl Acad Sci USA 104: 13432-7 (2007) Article DOI: 10.1073/pnas.0704212104 BindingDB Entry DOI: 10.7270/Q2X067X8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
CAAX prenyl protease 1 homolog (Mus musculus) | BDBM578 ((2S)-N-[(2S,4S,5S)-5-[2-(2,6-dimethylphenoxy)aceta...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL MCE MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 1.84E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description Inhibition of mouse ZMPSTE24 expressed n delta ste24 delta rce1 yeast | Proc Natl Acad Sci USA 104: 13432-7 (2007) Article DOI: 10.1073/pnas.0704212104 BindingDB Entry DOI: 10.7270/Q2X067X8 | |||||||||||
More data for this Ligand-Target Pair |