Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Transient receptor potential cation channel subfamily V member 1 (Rattus norvegicus (rat)) | BDBM50248768 (1,3-dibenzyl urea | CHEMBL504463) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
Central Drug Research Institute Curated by ChEMBL | Assay Description Antagonist activity at TRPV1 in rat DRG neuron assessed as inhibition of calcium uptake | Eur J Med Chem 44: 432-6 (2008) Article DOI: 10.1016/j.ejmech.2007.12.018 BindingDB Entry DOI: 10.7270/Q2FX797G | |||||||||||
More data for this Ligand-Target Pair |