Affinity Data by PubMed id=18482837

PubMed code 18482837

Found 5 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Peroxisome proliferator-activated receptor gamma (Rattus norvegicus)	BDBM50271605 (2-(4-(2-fluorobenzyloxy)benzyl)-3-hydroxynaphthale...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	200	n/a	n/a	n/a	n/a	n/a	n/a
National Institute of Pharmaceutical Education and Research Curated by ChEMBL					Assay Description Displacement of [3H]rosigliatzone from PPARgamma in rat adipocytes				Bioorg Med Chem Lett 18: 3192-5 (2008) Article DOI: 10.1016/j.bmcl.2008.04.072 BindingDB Entry DOI: 10.7270/Q2J9665P
					More data for this Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma (Rattus norvegicus)	BDBM50049240 ((+-)-5-((4-(2-(5-ethyl-2-pyridinyl)ethoxy)phenyl)m...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	700	n/a	n/a	n/a	n/a	n/a	n/a
National Institute of Pharmaceutical Education and Research Curated by ChEMBL					Assay Description Displacement of [3H]rosigliatzone from PPARgamma in rat adipocytes				Bioorg Med Chem Lett 18: 3192-5 (2008) Article DOI: 10.1016/j.bmcl.2008.04.072 BindingDB Entry DOI: 10.7270/Q2J9665P
					More data for this Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma (Rattus norvegicus)	BDBM50271732 (4-(2-(4-((3-hydroxy-1,4-dioxo-1,4-dihydronaphthale...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.90E+3	n/a	n/a	n/a	n/a	n/a	n/a
National Institute of Pharmaceutical Education and Research Curated by ChEMBL					Assay Description Displacement of [3H]rosigliatzone from PPARgamma in rat adipocytes				Bioorg Med Chem Lett 18: 3192-5 (2008) Article DOI: 10.1016/j.bmcl.2008.04.072 BindingDB Entry DOI: 10.7270/Q2J9665P
					More data for this Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma (Rattus norvegicus)	BDBM50271604 (2-(4-(benzyloxy)benzyl)-3-hydroxynaphthalene-1,4-d...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	3.60E+3	n/a	n/a	n/a	n/a	n/a	n/a
National Institute of Pharmaceutical Education and Research Curated by ChEMBL					Assay Description Displacement of [3H]rosigliatzone from PPARgamma in rat adipocytes				Bioorg Med Chem Lett 18: 3192-5 (2008) Article DOI: 10.1016/j.bmcl.2008.04.072 BindingDB Entry DOI: 10.7270/Q2J9665P
					More data for this Ligand-Target Pair
Peroxisome proliferator-activated receptor gamma (Rattus norvegicus)	BDBM50271662 (2-(4-(2-(4-methoxyphenoxy)ethoxy)benzyl)-3-hydroxy...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	5.62E+4	n/a	n/a	n/a	n/a	n/a	n/a
National Institute of Pharmaceutical Education and Research Curated by ChEMBL					Assay Description Displacement of [3H]rosigliatzone from PPARgamma in rat adipocytes				Bioorg Med Chem Lett 18: 3192-5 (2008) Article DOI: 10.1016/j.bmcl.2008.04.072 BindingDB Entry DOI: 10.7270/Q2J9665P
					More data for this Ligand-Target Pair

* indicates data uncertainty>20%