Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Peptidylglycine alpha-amidating monooxygenase (Rattus norvegicus) | BDBM50273316 (CHEMBL509495 | N-dansyl-Tyr-Val-D-Ala) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.70E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of South Florida Curated by ChEMBL | Assay Description Inhibition of rat recombinant peptidylglycine alpha-amidating monooxygenase assessed as inhibition of N-dansyl-Tyr-Val-Gly amidation | Bioorg Med Chem 16: 10061-74 (2008) Article DOI: 10.1016/j.bmc.2008.10.013 BindingDB Entry DOI: 10.7270/Q22R3RHS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidylglycine alpha-amidating monooxygenase (Rattus norvegicus) | BDBM50273962 (CHEMBL445286 | Phenylthioacetylglycine) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 3.80E+6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of South Florida Curated by ChEMBL | Assay Description Inhibition of rat recombinant peptidylglycine alpha-amidating monooxygenase assessed as inhibition of N-dansyl-Tyr-Val-Gly amidation | Bioorg Med Chem 16: 10061-74 (2008) Article DOI: 10.1016/j.bmc.2008.10.013 BindingDB Entry DOI: 10.7270/Q22R3RHS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidylglycine alpha-amidating monooxygenase (Rattus norvegicus) | BDBM50273494 (6-O-Palmitoyl-L-ascorbate | CHEMBL457018) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of South Florida Curated by ChEMBL | Assay Description Inhibition of rat recombinant peptidylglycine alpha-amidating monooxygenase in presence of DMSO | Bioorg Med Chem 16: 10061-74 (2008) Article DOI: 10.1016/j.bmc.2008.10.013 BindingDB Entry DOI: 10.7270/Q22R3RHS | |||||||||||
More data for this Ligand-Target Pair |