Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Galanin receptor type 1 (RAT) | BDBM50149871 ((R)-2-((3-(biphenyl-4-yloxy)-3-(4-fluorophenyl)pro...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
Taisho Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cells | Bioorg Med Chem Lett 18: 6321-3 (2008) Article DOI: 10.1016/j.bmcl.2008.10.104 BindingDB Entry DOI: 10.7270/Q2BZ65WC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Galanin receptor type 1 (RAT) | BDBM50256665 ((3S,6S,9S,12S)-3-benzyl-9,12-di-sec-butyl-6-((2S,3...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
Taisho Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cells | Bioorg Med Chem Lett 18: 6321-3 (2008) Article DOI: 10.1016/j.bmcl.2008.10.104 BindingDB Entry DOI: 10.7270/Q2BZ65WC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Galanin receptor type 1 (RAT) | BDBM50256666 ((3S,6S,9S,12S)-3-benzyl-12-sec-butyl-6-((2S,3R)-3-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 10.2 | n/a | n/a | n/a | n/a | n/a | n/a |
Taisho Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cells | Bioorg Med Chem Lett 18: 6321-3 (2008) Article DOI: 10.1016/j.bmcl.2008.10.104 BindingDB Entry DOI: 10.7270/Q2BZ65WC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Galanin receptor type 1 (RAT) | BDBM50256705 ((3S,6S,9S,12S)-3-benzyl-6-((2S,3R)-3-hydroxybutan-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 11.1 | n/a | n/a | n/a | n/a | n/a | n/a |
Taisho Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cells | Bioorg Med Chem Lett 18: 6321-3 (2008) Article DOI: 10.1016/j.bmcl.2008.10.104 BindingDB Entry DOI: 10.7270/Q2BZ65WC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Galanin receptor type 1 (RAT) | BDBM50256704 ((3S,6S,9S,12S)-3-benzyl-9-sec-butyl-6-((2S,3R)-3-h...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 11.4 | n/a | n/a | n/a | n/a | n/a | n/a |
Taisho Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cells | Bioorg Med Chem Lett 18: 6321-3 (2008) Article DOI: 10.1016/j.bmcl.2008.10.104 BindingDB Entry DOI: 10.7270/Q2BZ65WC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Galanin receptor type 1 (RAT) | BDBM50256664 ((S)-2-((2S,5S,8S,11S)-5-benzyl-8,11-di-sec-butyl-3...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 20.4 | n/a | n/a | n/a | n/a | n/a | n/a |
Taisho Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cells | Bioorg Med Chem Lett 18: 6321-3 (2008) Article DOI: 10.1016/j.bmcl.2008.10.104 BindingDB Entry DOI: 10.7270/Q2BZ65WC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Galanin receptor type 2 (RAT) | BDBM50256745 ((2S)-2-amino-3-((2-(benzyloxy)phenyl)(3-fluorophen...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | 21.1 | n/a | n/a | n/a | n/a | n/a | n/a |
Taisho Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cells | Bioorg Med Chem Lett 18: 6321-3 (2008) Article DOI: 10.1016/j.bmcl.2008.10.104 BindingDB Entry DOI: 10.7270/Q2BZ65WC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Galanin receptor type 1 (RAT) | BDBM50256706 ((3S,6S,9S,12S)-3-benzyl-6,9,12-tri-sec-butyl-1,4,7...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 29.6 | n/a | n/a | n/a | n/a | n/a | n/a |
Taisho Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cells | Bioorg Med Chem Lett 18: 6321-3 (2008) Article DOI: 10.1016/j.bmcl.2008.10.104 BindingDB Entry DOI: 10.7270/Q2BZ65WC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Galanin receptor type 2 (RAT) | BDBM50256746 ((3S,6S,9S,15aR)-9-sec-butyl-6-((1-methoxy-1H-indol...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 87.7 | n/a | n/a | n/a | n/a | n/a | n/a |
Taisho Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cells | Bioorg Med Chem Lett 18: 6321-3 (2008) Article DOI: 10.1016/j.bmcl.2008.10.104 BindingDB Entry DOI: 10.7270/Q2BZ65WC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Galanin receptor type 1 (RAT) | BDBM50256746 ((3S,6S,9S,15aR)-9-sec-butyl-6-((1-methoxy-1H-indol...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 94.6 | n/a | n/a | n/a | n/a | n/a | n/a |
Taisho Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of [3H]glycine uptake at rat glycine transporter 1 expressed in african green monkey COS7 cells | Bioorg Med Chem Lett 18: 6321-3 (2008) Article DOI: 10.1016/j.bmcl.2008.10.104 BindingDB Entry DOI: 10.7270/Q2BZ65WC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Galanin receptor type 2 (RAT) | BDBM50256706 ((3S,6S,9S,12S)-3-benzyl-6,9,12-tri-sec-butyl-1,4,7...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 226 | n/a | n/a | n/a | n/a | n/a | n/a |
Taisho Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cells | Bioorg Med Chem Lett 18: 6321-3 (2008) Article DOI: 10.1016/j.bmcl.2008.10.104 BindingDB Entry DOI: 10.7270/Q2BZ65WC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Galanin receptor type 2 (RAT) | BDBM50256665 ((3S,6S,9S,12S)-3-benzyl-9,12-di-sec-butyl-6-((2S,3...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 278 | n/a | n/a | n/a | n/a | n/a | n/a |
Taisho Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cells | Bioorg Med Chem Lett 18: 6321-3 (2008) Article DOI: 10.1016/j.bmcl.2008.10.104 BindingDB Entry DOI: 10.7270/Q2BZ65WC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Galanin receptor type 2 (RAT) | BDBM50256704 ((3S,6S,9S,12S)-3-benzyl-9-sec-butyl-6-((2S,3R)-3-h...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 450 | n/a | n/a | n/a | n/a | n/a | n/a |
Taisho Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cells | Bioorg Med Chem Lett 18: 6321-3 (2008) Article DOI: 10.1016/j.bmcl.2008.10.104 BindingDB Entry DOI: 10.7270/Q2BZ65WC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Galanin receptor type 2 (RAT) | BDBM50256705 ((3S,6S,9S,12S)-3-benzyl-6-((2S,3R)-3-hydroxybutan-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 542 | n/a | n/a | n/a | n/a | n/a | n/a |
Taisho Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cells | Bioorg Med Chem Lett 18: 6321-3 (2008) Article DOI: 10.1016/j.bmcl.2008.10.104 BindingDB Entry DOI: 10.7270/Q2BZ65WC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Galanin receptor type 2 (RAT) | BDBM50256666 ((3S,6S,9S,12S)-3-benzyl-12-sec-butyl-6-((2S,3R)-3-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 574 | n/a | n/a | n/a | n/a | n/a | n/a |
Taisho Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cells | Bioorg Med Chem Lett 18: 6321-3 (2008) Article DOI: 10.1016/j.bmcl.2008.10.104 BindingDB Entry DOI: 10.7270/Q2BZ65WC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Galanin receptor type 2 (RAT) | BDBM50256664 ((S)-2-((2S,5S,8S,11S)-5-benzyl-8,11-di-sec-butyl-3...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.26E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Taisho Pharmaceutical Co., Ltd Curated by ChEMBL | Assay Description Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cells | Bioorg Med Chem Lett 18: 6321-3 (2008) Article DOI: 10.1016/j.bmcl.2008.10.104 BindingDB Entry DOI: 10.7270/Q2BZ65WC | |||||||||||
More data for this Ligand-Target Pair |