Affinity Data by PubMed id=19297156

PubMed code 19297156

Found 43 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (Homo sapiens (Human))	BDBM12915 (2-(4-Morpholinyl)-8-phenyl-4H-1-benzopyran-4-one \|...) Show SMILES O=c1cc(oc2c(cccc12)-c1ccccc1)N1CCOCC1 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars	Article PubMed	n/a	n/a	200	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kalpha by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform (Homo sapiens (Human))	BDBM12915 (2-(4-Morpholinyl)-8-phenyl-4H-1-benzopyran-4-one \|...) Show SMILES O=c1cc(oc2c(cccc12)-c1ccccc1)N1CCOCC1 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars	DrugBank PDB Article PubMed	n/a	n/a	1.20E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kgamma by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair				3D Structure (crystal)
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (Homo sapiens (Human))	BDBM50278545 (2-((4-fluoro-2-methylphenylamino)methyl)-6-morphol...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	5.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kalpha by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (Homo sapiens (Human))	BDBM50278506 (2-((4-fluoro-2-methylphenoxy)methyl)-6-morpholinoi...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	7.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kalpha by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (Homo sapiens (Human))	BDBM50278504 (2-((4-fluoro-2-methylphenoxy)methyl)-6-morpholinoi...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kalpha by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform (Homo sapiens (Human))	BDBM50278503 (2-((4-fluoro-2-methylphenoxy)methyl)-N-hydroxy-6-m...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kgamma by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (Homo sapiens (Human))	BDBM50278543 ((2-((4-fluoro-2-methylphenylamino)methyl)-6-morpho...) Show SMILES Cc1cc(F)ccc1NCc1cc(CO)cc(n1)N1CCOCC1 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	2.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kalpha by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform (Homo sapiens (Human))	BDBM50278506 (2-((4-fluoro-2-methylphenoxy)methyl)-6-morpholinoi...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	2.30E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kgamma by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (Homo sapiens (Human))	BDBM50278613 (6-((4-fluoro-2-methylphenylamino)methyl)-2,4'-bipy...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	2.90E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kalpha by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform (Homo sapiens (Human))	BDBM50278545 (2-((4-fluoro-2-methylphenylamino)methyl)-6-morphol...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	3.40E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kgamma by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (Homo sapiens (Human))	BDBM50278659 (2-morpholinoisonicotinic acid \| CHEMBL449172) Show SMILES OC(=O)c1ccnc(c1)N1CCOCC1 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	3.60E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kalpha by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform (Homo sapiens (Human))	BDBM50278613 (6-((4-fluoro-2-methylphenylamino)methyl)-2,4'-bipy...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	4.20E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kgamma by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform (Homo sapiens (Human))	BDBM50278616 (2-((4-fluoro-2-methylphenylamino)methyl)-6-(3-hydr...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	4.20E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kgamma by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (Homo sapiens (Human))	BDBM50278660 (CHEMBL450243 \| ethyl 2-morpholinoisonicotinate) Show SMILES CCOC(=O)c1ccnc(c1)N1CCOCC1 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	5.10E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kalpha by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (Homo sapiens (Human))	BDBM50278617 (2-((4-fluoro-2-methylphenylamino)methyl)-6-(2-hydr...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kalpha by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform (Homo sapiens (Human))	BDBM50278577 (2-((4-fluoro-2-methylphenylamino)methyl)-6-((2-hyd...) Show SMILES CN(CCO)c1cc(cc(CNc2ccc(F)cc2C)n1)C(O)=O Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kgamma by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform (Homo sapiens (Human))	BDBM50278656 (2-chloro-6-((4-fluoro-2-methylphenylamino)methyl)i...) Show SMILES Cc1cc(F)ccc1NCc1cc(cc(Cl)n1)C(O)=O Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kgamma by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (Homo sapiens (Human))	BDBM50278579 (2-(bis(2-hydroxyethyl)amino)-6-((4-fluoro-2-methyl...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kalpha by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform (Homo sapiens (Human))	BDBM50278544 (2-((4-fluoro-2-methylphenylamino)methyl)-6-morphol...) Show SMILES Cc1cc(F)ccc1NCc1cc(C=O)cc(n1)N1CCOCC1 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kgamma by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform (Homo sapiens (Human))	BDBM50278546 (2-((4-fluoro-2-methylphenylamino)methyl)-6-(pipera...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kgamma by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform (Homo sapiens (Human))	BDBM50278547 (2-((4-fluoro-2-methylphenylamino)methyl)-6-(piperi...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kgamma by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform (Homo sapiens (Human))	BDBM50278615 (2-((4-fluoro-2-methylphenylamino)methyl)-6-(4-hydr...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kgamma by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform (Homo sapiens (Human))	BDBM50278617 (2-((4-fluoro-2-methylphenylamino)methyl)-6-(2-hydr...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kgamma by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (Homo sapiens (Human))	BDBM50278616 (2-((4-fluoro-2-methylphenylamino)methyl)-6-(3-hydr...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kalpha by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform (Homo sapiens (Human))	BDBM50278576 (2-((4-fluoro-2-methylphenylamino)methyl)-6-(3-hydr...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kgamma by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform (Homo sapiens (Human))	BDBM50278579 (2-(bis(2-hydroxyethyl)amino)-6-((4-fluoro-2-methyl...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kgamma by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform (Homo sapiens (Human))	BDBM50278658 ((2-((4-fluoro-2-methylphenylamino)methyl)-6-(3-hyd...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kgamma by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (Homo sapiens (Human))	BDBM50278577 (2-((4-fluoro-2-methylphenylamino)methyl)-6-((2-hyd...) Show SMILES CN(CCO)c1cc(cc(CNc2ccc(F)cc2C)n1)C(O)=O Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kalpha by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (Homo sapiens (Human))	BDBM50278578 (2-((4-fluoro-2-methylphenylamino)methyl)-6-(2-hydr...) Show SMILES Cc1cc(F)ccc1NCc1cc(cc(NCCO)n1)C(O)=O Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kalpha by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform (Homo sapiens (Human))	BDBM50278614 (6-((4-fluoro-2-methylphenylamino)methyl)-2,3'-bipy...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kgamma by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform (Homo sapiens (Human))	BDBM50278578 (2-((4-fluoro-2-methylphenylamino)methyl)-6-(2-hydr...) Show SMILES Cc1cc(F)ccc1NCc1cc(cc(NCCO)n1)C(O)=O Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kgamma by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform (Homo sapiens (Human))	BDBM50278660 (CHEMBL450243 \| ethyl 2-morpholinoisonicotinate) Show SMILES CCOC(=O)c1ccnc(c1)N1CCOCC1 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kgamma by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform (Homo sapiens (Human))	BDBM50278659 (2-morpholinoisonicotinic acid \| CHEMBL449172) Show SMILES OC(=O)c1ccnc(c1)N1CCOCC1 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kgamma by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (Homo sapiens (Human))	BDBM50278658 ((2-((4-fluoro-2-methylphenylamino)methyl)-6-(3-hyd...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kalpha by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (Homo sapiens (Human))	BDBM50278656 (2-chloro-6-((4-fluoro-2-methylphenylamino)methyl)i...) Show SMILES Cc1cc(F)ccc1NCc1cc(cc(Cl)n1)C(O)=O Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kalpha by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (Homo sapiens (Human))	BDBM50278544 (2-((4-fluoro-2-methylphenylamino)methyl)-6-morphol...) Show SMILES Cc1cc(F)ccc1NCc1cc(C=O)cc(n1)N1CCOCC1 Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kalpha by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform (Homo sapiens (Human))	BDBM50278657 (2-((4-fluoro-2-methylphenylamino)methyl)-N-(2-hydr...) Show SMILES Cc1cc(F)ccc1NCc1cc(cc(NCCO)n1)C(=O)NCCO Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL KEGG PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kgamma by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform (Homo sapiens (Human))	BDBM50278575 (2-((4-fluoro-2-methylphenylamino)methyl)-6-(pyrrol...) Show SMILES Cc1cc(F)ccc1NCc1cc(cc(n1)N1CCCC1)C(O)=O Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kgamma by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (Homo sapiens (Human))	BDBM50278657 (2-((4-fluoro-2-methylphenylamino)methyl)-N-(2-hydr...) Show SMILES Cc1cc(F)ccc1NCc1cc(cc(NCCO)n1)C(=O)NCCO Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL KEGG PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kalpha by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (Homo sapiens (Human))	BDBM50278614 (6-((4-fluoro-2-methylphenylamino)methyl)-2,3'-bipy...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kalpha by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (Homo sapiens (Human))	BDBM50278615 (2-((4-fluoro-2-methylphenylamino)methyl)-6-(4-hydr...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kalpha by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (Homo sapiens (Human))	BDBM50278546 (2-((4-fluoro-2-methylphenylamino)methyl)-6-(pipera...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kalpha by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (Homo sapiens (Human))	BDBM50278576 (2-((4-fluoro-2-methylphenylamino)methyl)-6-(3-hydr...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Cincinnati Curated by ChEMBL					Assay Description Inhibition of PI3Kalpha by luminescent kinase glo assay				Bioorg Med Chem Lett 19: 2215-9 (2009) Article DOI: 10.1016/j.bmcl.2009.02.115 BindingDB Entry DOI: 10.7270/Q2KP833D
University of Cincinnati Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%