Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50251393 (CHEMBL519266 | Rhynchophylline) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.73E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
China Medical University Curated by ChEMBL | Assay Description Inhibition of human ERG channel | J Nat Prod 72: 830-4 (2010) Article DOI: 10.1021/np800729q BindingDB Entry DOI: 10.7270/Q2R78F7D | |||||||||||
More data for this Ligand-Target Pair |