Affinity Data by PubMed id=19640720

PubMed code 19640720

Found 4 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Mu-type opioid receptor (Rattus norvegicus (rat))	BDBM21015 ((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.01	n/a	n/a	n/a	n/a	n/a	n/a
Institute of Chemical Biology Curated by ChEMBL					Assay Description Displacement of [3H]DAMGO from mu opioid receptor in rat brain				Bioorg Med Chem 17: 5782-90 (2009) Article DOI: 10.1016/j.bmc.2009.07.024 BindingDB Entry DOI: 10.7270/Q2VQ32RF
Institute of Chemical Biology Curated by ChEMBL					More data for this Ligand-Target Pair
Kappa-type opioid receptor (Homo sapiens (Human))	BDBM50304074 (2-(2-methylquinolin-4-ylamino)-N-phenylacetamide \|...) Show SMILES Cc1cc(NCC(=O)Nc2ccccc2)c2ccccc2n1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.03	n/a	n/a	n/a	n/a	n/a	n/a
Institute of Chemical Biology Curated by ChEMBL					Assay Description Displacement of [3H]dynorphin from human kappa opioid receptor expressed in C6 giloma cells				Bioorg Med Chem 17: 5782-90 (2009) Article DOI: 10.1016/j.bmc.2009.07.024 BindingDB Entry DOI: 10.7270/Q2VQ32RF
Institute of Chemical Biology Curated by ChEMBL					More data for this Ligand-Target Pair
Mu-type opioid receptor (Rattus norvegicus (rat))	BDBM50304074 (2-(2-methylquinolin-4-ylamino)-N-phenylacetamide \|...) Show SMILES Cc1cc(NCC(=O)Nc2ccccc2)c2ccccc2n1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.15	n/a	n/a	n/a	n/a	n/a	n/a
Institute of Chemical Biology Curated by ChEMBL					Assay Description Displacement of [3H]DAMGO from mu opioid receptor in rat brain				Bioorg Med Chem 17: 5782-90 (2009) Article DOI: 10.1016/j.bmc.2009.07.024 BindingDB Entry DOI: 10.7270/Q2VQ32RF
Institute of Chemical Biology Curated by ChEMBL					More data for this Ligand-Target Pair
Kappa-type opioid receptor (Homo sapiens (Human))	BDBM50000296 (CHEMBL441765 \| CHEMBL482811 \| U-50488H \| US1149237...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL KEGG PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	1.99	n/a	n/a	n/a	n/a	n/a	n/a
Institute of Chemical Biology Curated by ChEMBL					Assay Description Displacement of [3H]dynorphin from human kappa opioid receptor expressed in C6 giloma cells				Bioorg Med Chem 17: 5782-90 (2009) Article DOI: 10.1016/j.bmc.2009.07.024 BindingDB Entry DOI: 10.7270/Q2VQ32RF
Institute of Chemical Biology Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%