Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM22885 (3-[(2S)-1-(1H-imidazol-5-yl)propan-2-yl]-2-(2-{[(5...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vrije Universiteit Curated by ChEMBL | Assay Description Evaluated for antagonistic activity at histamine H3 receptor in rat cerebral cortex and is represented as Ki | J Med Chem 33: 4-11 (1990) BindingDB Entry DOI: 10.7270/Q2GB230D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM85411 (GT 2174) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | PubMed | 50 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vrije Universiteit Curated by ChEMBL | Assay Description Evaluated for antagonist activity against histamine H3 receptor and is represented as -log Ki. | J Med Chem 33: 4-11 (1990) BindingDB Entry DOI: 10.7270/Q2GB230D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM22886 (3-[(2R)-1-(1H-imidazol-5-yl)propan-2-yl]-2-(2-{[(5...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vrije Universiteit Curated by ChEMBL | Assay Description Evaluated for antagonistic activity at histamine H3 receptor in rat cerebral cortex and is represented as Ki. | J Med Chem 33: 4-11 (1990) BindingDB Entry DOI: 10.7270/Q2GB230D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM50406098 (CHEMBL12494) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | 79 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vrije Universiteit Curated by ChEMBL | Assay Description Evaluated for antagonist activity against Histamine H3 receptor and represented as KB. | J Med Chem 33: 4-11 (1990) BindingDB Entry DOI: 10.7270/Q2GB230D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM50406100 (CHEMBL12459) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 200 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vrije Universiteit Curated by ChEMBL | Assay Description Evaluated for antagonist activity against Histamine H3 receptor and represented as KB. | J Med Chem 33: 4-11 (1990) BindingDB Entry DOI: 10.7270/Q2GB230D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM50406095 (CHEMBL275090) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 631 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vrije Universiteit Curated by ChEMBL | Assay Description Evaluated for antagonist activity against histamine H3 receptor and is represented as -log Ki. | J Med Chem 33: 4-11 (1990) BindingDB Entry DOI: 10.7270/Q2GB230D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM50406101 (CHEMBL12550) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | 631 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vrije Universiteit Curated by ChEMBL | Assay Description Evaluated for antagonist activity against Histamine H3 receptor and represented as KB. | J Med Chem 33: 4-11 (1990) BindingDB Entry DOI: 10.7270/Q2GB230D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM50406099 (CHEMBL416338) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vrije Universiteit Curated by ChEMBL | Assay Description Evaluated for antagonist activity against histamine H3 receptor and is represented as -log Ki. | J Med Chem 33: 4-11 (1990) BindingDB Entry DOI: 10.7270/Q2GB230D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM50406097 (CHEMBL12551) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vrije Universiteit Curated by ChEMBL | Assay Description Evaluated for antagonist activity against histamine H3 receptor and is represented as -log Ki. | J Med Chem 33: 4-11 (1990) BindingDB Entry DOI: 10.7270/Q2GB230D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM50406093 (CHEMBL276903) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vrije Universiteit Curated by ChEMBL | Assay Description Evaluated for antagonist activity against Histamine H3 receptor and represented as KB. | J Med Chem 33: 4-11 (1990) BindingDB Entry DOI: 10.7270/Q2GB230D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM50406096 (CHEMBL12025) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vrije Universiteit Curated by ChEMBL | Assay Description Evaluated for antagonist activity against Histamine H3 receptor and represented as KB. | J Med Chem 33: 4-11 (1990) BindingDB Entry DOI: 10.7270/Q2GB230D | |||||||||||
More data for this Ligand-Target Pair |