Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Proto-oncogene tyrosine-protein kinase ROS (Homo sapiens (Human)) | BDBM50300460 (2-(4-(2,3'-bipyridin-4-yl)-3-(3-hydroxy-5-methylph...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 209 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Science and Technology Curated by ChEMBL | Assay Description Inhibition of ROS1 by HotSpot assay | Bioorg Med Chem Lett 19: 5622-6 (2009) Article DOI: 10.1016/j.bmcl.2009.08.029 BindingDB Entry DOI: 10.7270/Q28P60JF | |||||||||||
More data for this Ligand-Target Pair |