Affinity Data by PubMed id=19957998

PubMed code 19957998

Found 8 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Solute carrier family 15 member 1 (Homo sapiens (Human))	BDBM50308747 ((S)-2-amino-3-methylbutanoic benzoic anhydride \| C...) Show SMILES CC(C)[C@H](N)C(=O)OC(=O)c1ccccc1 \|r\| Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL KEGG PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	3.90E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Michigan Curated by ChEMBL					Assay Description Inhibition of human PEPT1-mediated [3H]Gly-Sar uptake in human HeLa cells				J Med Chem 53: 624-32 (2010) Article DOI: 10.1021/jm9011559 BindingDB Entry DOI: 10.7270/Q2251J90
University of Michigan Curated by ChEMBL					More data for this Ligand-Target Pair
Solute carrier family 15 member 1 (Homo sapiens (Human))	BDBM50308748 ((2S,3S)-2-amino-3-methylpentanoic benzoic anhydrid...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL KEGG PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	6.30E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Michigan Curated by ChEMBL					Assay Description Inhibition of human PEPT1-mediated [3H]Gly-Sar uptake in human HeLa cells				J Med Chem 53: 624-32 (2010) Article DOI: 10.1021/jm9011559 BindingDB Entry DOI: 10.7270/Q2251J90
University of Michigan Curated by ChEMBL					More data for this Ligand-Target Pair
Solute carrier family 15 member 1 (Homo sapiens (Human))	BDBM50308745 (CHEMBL589585 \| L-Isoleucine[3-[(Aminoiminomethyl)a...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL KEGG PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	6.30E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Michigan Curated by ChEMBL					Assay Description Inhibition of human PEPT1-mediated [3H]Gly-Sar uptake in human HeLa cells				J Med Chem 53: 624-32 (2010) Article DOI: 10.1021/jm9011559 BindingDB Entry DOI: 10.7270/Q2251J90
University of Michigan Curated by ChEMBL					More data for this Ligand-Target Pair
Solute carrier family 15 member 1 (Homo sapiens (Human))	BDBM50308744 (CHEMBL590321 \| L-Valine[3-[(Aminoiminomethyl)amino...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL KEGG PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	6.50E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Michigan Curated by ChEMBL					Assay Description Inhibition of human PEPT1-mediated [3H]Gly-Sar uptake in human HeLa cells				J Med Chem 53: 624-32 (2010) Article DOI: 10.1021/jm9011559 BindingDB Entry DOI: 10.7270/Q2251J90
University of Michigan Curated by ChEMBL					More data for this Ligand-Target Pair
Solute carrier family 15 member 1 (Homo sapiens (Human))	BDBM50162073 ((S)-2-((2-amino-6-oxo-3H-purin-9(6H)-yl)methoxy)et...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars	Article PubMed	n/a	n/a	1.42E+6	n/a	n/a	n/a	n/a	n/a	n/a
University of Michigan Curated by ChEMBL					Assay Description Inhibition of human PEPT1-mediated [3H]Gly-Sar uptake in human HeLa cells				J Med Chem 53: 624-32 (2010) Article DOI: 10.1021/jm9011559 BindingDB Entry DOI: 10.7270/Q2251J90
University of Michigan Curated by ChEMBL					More data for this Ligand-Target Pair
Solute carrier family 15 member 1 (Homo sapiens (Human))	BDBM50308746 (CHEMBL603829 \| L-Phenylalanine[3-[(Aminoiminomethy...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL KEGG PC cid PC sid UniChem	Article PubMed	n/a	n/a	2.33E+6	n/a	n/a	n/a	n/a	n/a	n/a
University of Michigan Curated by ChEMBL					Assay Description Inhibition of human PEPT1-mediated [3H]Gly-Sar uptake in human HeLa cells				J Med Chem 53: 624-32 (2010) Article DOI: 10.1021/jm9011559 BindingDB Entry DOI: 10.7270/Q2251J90
University of Michigan Curated by ChEMBL					More data for this Ligand-Target Pair
Solute carrier family 15 member 1 (Homo sapiens (Human))	BDBM50308743 (CHEMBL590071 \| [3-(hydroxymethyl)phenyl]guanidine) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Patents	Article PubMed	n/a	n/a	>3.00E+6	n/a	n/a	n/a	n/a	n/a	n/a
University of Michigan Curated by ChEMBL					Assay Description Inhibition of human PEPT1-mediated [3H]Gly-Sar uptake in human HeLa cells				J Med Chem 53: 624-32 (2010) Article DOI: 10.1021/jm9011559 BindingDB Entry DOI: 10.7270/Q2251J90
University of Michigan Curated by ChEMBL					More data for this Ligand-Target Pair
Solute carrier family 15 member 1 (Homo sapiens (Human))	BDBM50308749 ((S)-2-amino-3-phenylpropanoic benzoic anhydride \| ...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL KEGG PC cid PC sid UniChem Patents	Article PubMed	n/a	n/a	>3.00E+6	n/a	n/a	n/a	n/a	n/a	n/a
University of Michigan Curated by ChEMBL					Assay Description Inhibition of human PEPT1-mediated [3H]Gly-Sar uptake in human HeLa cells				J Med Chem 53: 624-32 (2010) Article DOI: 10.1021/jm9011559 BindingDB Entry DOI: 10.7270/Q2251J90
University of Michigan Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%