Affinity Data by PubMed id=20143782

PubMed code 20143782

Found 3 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
5-hydroxytryptamine receptor 2A (Homo sapiens (Human))	BDBM50307812 (1-[3-(4-Bromo-2-methyl-2Hpyrazol-3-yl)-4-methoxyph...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	n/a	n/a	0.700	n/a	n/a	n/a	n/a
Arena Pharmaceuticals, Inc Curated by ChEMBL					Assay Description Activity at human 5HT2A receptor expressed in HEK293 cells assessed as [3H]inositol phosphate production by scintillation counting				J Med Chem 53: 1923-36 (2010) Article DOI: 10.1021/jm9007328 BindingDB Entry DOI: 10.7270/Q24B31FP
Arena Pharmaceuticals, Inc Curated by ChEMBL					More data for this Ligand-Target Pair
5-hydroxytryptamine receptor 2A (Homo sapiens (Human))	BDBM50307811 (1-(3-(4-bromo-1-methyl-1H-pyrazol-5-yl)phenyl)-3-(...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	19	n/a	n/a	n/a	n/a
Arena Pharmaceuticals, Inc Curated by ChEMBL					Assay Description Activity at human 5HT2A receptor expressed in HEK293 cells assessed as [3H]inositol phosphate production by scintillation counting				J Med Chem 53: 1923-36 (2010) Article DOI: 10.1021/jm9007328 BindingDB Entry DOI: 10.7270/Q24B31FP
Arena Pharmaceuticals, Inc Curated by ChEMBL					More data for this Ligand-Target Pair
5-hydroxytryptamine receptor 2A (Homo sapiens (Human))	BDBM50307813 (1-(3-(4-bromo-1-methyl-1H-pyrazol-5-yl)phenyl)-3-(...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	120	n/a	n/a	n/a	n/a
Arena Pharmaceuticals, Inc Curated by ChEMBL					Assay Description Activity at human 5HT2A receptor expressed in HEK293 cells assessed as [3H]inositol phosphate production by scintillation counting				J Med Chem 53: 1923-36 (2010) Article DOI: 10.1021/jm9007328 BindingDB Entry DOI: 10.7270/Q24B31FP
Arena Pharmaceuticals, Inc Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%