Found 21 hits of Enzyme Inhibition Constant Data Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kJ/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
cAMP-specific 3',5'-cyclic phosphodiesterase 4B
(Homo sapiens (Human)) | BDBM50317611
(4-(3,5-dichloropyridin-4-ylamino)-8-(3-(dimethylam...)Show SMILES COc1ccc2c(Nc3c(Cl)cncc3Cl)cc(=O)oc2c1OCCCN(C)C Show InChI InChI=1S/C20H21Cl2N3O4/c1-25(2)7-4-8-28-20-16(27-3)6-5-12-15(9-17(26)29-19(12)20)24-18-13(21)10-23-11-14(18)22/h5-6,9-11H,4,7-8H2,1-3H3,(H,23,24) | PDB
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| n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
Kalypsys, Inc.
Curated by ChEMBL
| Assay Description
Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hr |
Bioorg Med Chem Lett 20: 2928-32 (2010)
Article DOI: 10.1016/j.bmcl.2010.03.023
BindingDB Entry DOI: 10.7270/Q2VD6ZMF |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4B
(Homo sapiens (Human)) | BDBM50317609
(8-(4-(3,5-dichloropyridin-4-ylamino)-7-methoxy-2-o...)Show SMILES COc1ccc2c(Nc3c(Cl)cncc3Cl)cc(=O)oc2c1OCCCCCCCC(O)=O Show InChI InChI=1S/C23H24Cl2N2O6/c1-31-18-9-8-14-17(27-21-15(24)12-26-13-16(21)25)11-20(30)33-22(14)23(18)32-10-6-4-2-3-5-7-19(28)29/h8-9,11-13H,2-7,10H2,1H3,(H,26,27)(H,28,29) | PDB
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| n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
Kalypsys, Inc.
Curated by ChEMBL
| Assay Description
Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hr |
Bioorg Med Chem Lett 20: 2928-32 (2010)
Article DOI: 10.1016/j.bmcl.2010.03.023
BindingDB Entry DOI: 10.7270/Q2VD6ZMF |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4B
(Homo sapiens (Human)) | BDBM50317610
(9-(4-(3,5-dichloropyridin-4-ylamino)-7-methoxy-2-o...)Show SMILES COc1ccc2c(Nc3c(Cl)cncc3Cl)cc(=O)oc2c1OCCCCCCCCC(O)=O Show InChI InChI=1S/C24H26Cl2N2O6/c1-32-19-10-9-15-18(28-22-16(25)13-27-14-17(22)26)12-21(31)34-23(15)24(19)33-11-7-5-3-2-4-6-8-20(29)30/h9-10,12-14H,2-8,11H2,1H3,(H,27,28)(H,29,30) | PDB
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| n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
Kalypsys, Inc.
Curated by ChEMBL
| Assay Description
Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hr |
Bioorg Med Chem Lett 20: 2928-32 (2010)
Article DOI: 10.1016/j.bmcl.2010.03.023
BindingDB Entry DOI: 10.7270/Q2VD6ZMF |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4B
(Homo sapiens (Human)) | BDBM50317616
(4-(3,5-dichloropyridin-4-ylamino)-8-(8-(dimethylam...)Show SMILES COc1ccc2c(Nc3c(Cl)cncc3Cl)cc(=O)oc2c1OCCCCCCCCN(C)C Show InChI InChI=1S/C25H31Cl2N3O4/c1-30(2)12-8-6-4-5-7-9-13-33-25-21(32-3)11-10-17-20(14-22(31)34-24(17)25)29-23-18(26)15-28-16-19(23)27/h10-11,14-16H,4-9,12-13H2,1-3H3,(H,28,29) | PDB
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| n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
Kalypsys, Inc.
Curated by ChEMBL
| Assay Description
Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hr |
Bioorg Med Chem Lett 20: 2928-32 (2010)
Article DOI: 10.1016/j.bmcl.2010.03.023
BindingDB Entry DOI: 10.7270/Q2VD6ZMF |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4B
(Homo sapiens (Human)) | BDBM14775
(3-(cyclopentyloxy)-N-(3,5-dichloropyridin-4-yl)-4-...)Show InChI InChI=1S/C18H18Cl2N2O3/c1-24-15-7-6-11(8-16(15)25-12-4-2-3-5-12)18(23)22-17-13(19)9-21-10-14(17)20/h6-10,12H,2-5H2,1H3,(H,21,22,23) | PDB
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| PDB
Article
PubMed
| n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
Kalypsys, Inc.
Curated by ChEMBL
| Assay Description
Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hr |
Bioorg Med Chem Lett 20: 2928-32 (2010)
Article DOI: 10.1016/j.bmcl.2010.03.023
BindingDB Entry DOI: 10.7270/Q2VD6ZMF |
More data for this
Ligand-Target Pair | 
3D Structure (crystal) |
cAMP-specific 3',5'-cyclic phosphodiesterase 4B
(Homo sapiens (Human)) | BDBM50317615
(4-(3,5-dichloropyridin-4-ylamino)-8-(7-(dimethylam...)Show SMILES COc1ccc2c(Nc3c(Cl)cncc3Cl)cc(=O)oc2c1OCCCCCCCN(C)C Show InChI InChI=1S/C24H29Cl2N3O4/c1-29(2)11-7-5-4-6-8-12-32-24-20(31-3)10-9-16-19(13-21(30)33-23(16)24)28-22-17(25)14-27-15-18(22)26/h9-10,13-15H,4-8,11-12H2,1-3H3,(H,27,28) | PDB
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| n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
Kalypsys, Inc.
Curated by ChEMBL
| Assay Description
Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hr |
Bioorg Med Chem Lett 20: 2928-32 (2010)
Article DOI: 10.1016/j.bmcl.2010.03.023
BindingDB Entry DOI: 10.7270/Q2VD6ZMF |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4B
(Homo sapiens (Human)) | BDBM50317614
(4-(3,5-dichloropyridin-4-ylamino)-8-(6-(dimethylam...)Show SMILES COc1ccc2c(Nc3c(Cl)cncc3Cl)cc(=O)oc2c1OCCCCCCN(C)C Show InChI InChI=1S/C23H27Cl2N3O4/c1-28(2)10-6-4-5-7-11-31-23-19(30-3)9-8-15-18(12-20(29)32-22(15)23)27-21-16(24)13-26-14-17(21)25/h8-9,12-14H,4-7,10-11H2,1-3H3,(H,26,27) | PDB
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| n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kalypsys, Inc.
Curated by ChEMBL
| Assay Description
Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hr |
Bioorg Med Chem Lett 20: 2928-32 (2010)
Article DOI: 10.1016/j.bmcl.2010.03.023
BindingDB Entry DOI: 10.7270/Q2VD6ZMF |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4B
(Homo sapiens (Human)) | BDBM50317604
(2-(4-(3,5-dichloropyridin-4-ylamino)-7-methoxy-2-o...)Show SMILES COc1ccc2c(Nc3c(Cl)cncc3Cl)cc(=O)oc2c1OCC(O)=O Show InChI InChI=1S/C17H12Cl2N2O6/c1-25-12-3-2-8-11(21-15-9(18)5-20-6-10(15)19)4-14(24)27-16(8)17(12)26-7-13(22)23/h2-6H,7H2,1H3,(H,20,21)(H,22,23) | PDB
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| n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kalypsys, Inc.
Curated by ChEMBL
| Assay Description
Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hr |
Bioorg Med Chem Lett 20: 2928-32 (2010)
Article DOI: 10.1016/j.bmcl.2010.03.023
BindingDB Entry DOI: 10.7270/Q2VD6ZMF |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4B
(Homo sapiens (Human)) | BDBM50317603
(8-(cyclopentyloxy)-4-(3,5-dichloropyridin-4-ylamin...)Show SMILES COc1ccc2c(Nc3c(Cl)cncc3Cl)cc(=O)oc2c1OC1CCCC1 Show InChI InChI=1S/C20H18Cl2N2O4/c1-26-16-7-6-12-15(24-18-13(21)9-23-10-14(18)22)8-17(25)28-19(12)20(16)27-11-4-2-3-5-11/h6-11H,2-5H2,1H3,(H,23,24) | PDB
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Article
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| n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kalypsys, Inc.
Curated by ChEMBL
| Assay Description
Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hr |
Bioorg Med Chem Lett 20: 2928-32 (2010)
Article DOI: 10.1016/j.bmcl.2010.03.023
BindingDB Entry DOI: 10.7270/Q2VD6ZMF |
More data for this
Ligand-Target Pair |
3D Structure (crystal) |
cAMP-specific 3',5'-cyclic phosphodiesterase 4B
(Homo sapiens (Human)) | BDBM50317608
(7-(4-(3,5-dichloropyridin-4-ylamino)-7-methoxy-2-o...)Show SMILES COc1ccc2c(Nc3c(Cl)cncc3Cl)cc(=O)oc2c1OCCCCCCC(O)=O Show InChI InChI=1S/C22H22Cl2N2O6/c1-30-17-8-7-13-16(26-20-14(23)11-25-12-15(20)24)10-19(29)32-21(13)22(17)31-9-5-3-2-4-6-18(27)28/h7-8,10-12H,2-6,9H2,1H3,(H,25,26)(H,27,28) | PDB
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| n/a | n/a | 17 | n/a | n/a | n/a | n/a | n/a | n/a |
Kalypsys, Inc.
Curated by ChEMBL
| Assay Description
Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hr |
Bioorg Med Chem Lett 20: 2928-32 (2010)
Article DOI: 10.1016/j.bmcl.2010.03.023
BindingDB Entry DOI: 10.7270/Q2VD6ZMF |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4B
(Homo sapiens (Human)) | BDBM50317613
(4-(3,5-dichloropyridin-4-ylamino)-8-(5-(dimethylam...)Show SMILES COc1ccc2c(Nc3c(Cl)cncc3Cl)cc(=O)oc2c1OCCCCCN(C)C Show InChI InChI=1S/C22H25Cl2N3O4/c1-27(2)9-5-4-6-10-30-22-18(29-3)8-7-14-17(11-19(28)31-21(14)22)26-20-15(23)12-25-13-16(20)24/h7-8,11-13H,4-6,9-10H2,1-3H3,(H,25,26) | PDB
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| n/a | n/a | 21 | n/a | n/a | n/a | n/a | n/a | n/a |
Kalypsys, Inc.
Curated by ChEMBL
| Assay Description
Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hr |
Bioorg Med Chem Lett 20: 2928-32 (2010)
Article DOI: 10.1016/j.bmcl.2010.03.023
BindingDB Entry DOI: 10.7270/Q2VD6ZMF |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4B
(Homo sapiens (Human)) | BDBM50317607
(6-(4-(3,5-dichloropyridin-4-ylamino)-7-methoxy-2-o...)Show SMILES COc1ccc2c(Nc3c(Cl)cncc3Cl)cc(=O)oc2c1OCCCCCC(O)=O Show InChI InChI=1S/C21H20Cl2N2O6/c1-29-16-7-6-12-15(25-19-13(22)10-24-11-14(19)23)9-18(28)31-20(12)21(16)30-8-4-2-3-5-17(26)27/h6-7,9-11H,2-5,8H2,1H3,(H,24,25)(H,26,27) | PDB
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| Article
PubMed
| n/a | n/a | 43 | n/a | n/a | n/a | n/a | n/a | n/a |
Kalypsys, Inc.
Curated by ChEMBL
| Assay Description
Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hr |
Bioorg Med Chem Lett 20: 2928-32 (2010)
Article DOI: 10.1016/j.bmcl.2010.03.023
BindingDB Entry DOI: 10.7270/Q2VD6ZMF |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4B
(Homo sapiens (Human)) | BDBM50317612
(4-(3,5-dichloropyridin-4-ylamino)-8-(4-(dimethylam...)Show SMILES COc1ccc2c(Nc3c(Cl)cncc3Cl)cc(=O)oc2c1OCCCCN(C)C Show InChI InChI=1S/C21H23Cl2N3O4/c1-26(2)8-4-5-9-29-21-17(28-3)7-6-13-16(10-18(27)30-20(13)21)25-19-14(22)11-24-12-15(19)23/h6-7,10-12H,4-5,8-9H2,1-3H3,(H,24,25) | PDB
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| Article
PubMed
| n/a | n/a | 45 | n/a | n/a | n/a | n/a | n/a | n/a |
Kalypsys, Inc.
Curated by ChEMBL
| Assay Description
Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hr |
Bioorg Med Chem Lett 20: 2928-32 (2010)
Article DOI: 10.1016/j.bmcl.2010.03.023
BindingDB Entry DOI: 10.7270/Q2VD6ZMF |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4B
(Homo sapiens (Human)) | BDBM50317606
(5-(4-(3,5-dichloropyridin-4-ylamino)-7-methoxy-2-o...)Show SMILES COc1ccc2c(Nc3c(Cl)cncc3Cl)cc(=O)oc2c1OCCCCC(O)=O Show InChI InChI=1S/C20H18Cl2N2O6/c1-28-15-6-5-11-14(24-18-12(21)9-23-10-13(18)22)8-17(27)30-19(11)20(15)29-7-3-2-4-16(25)26/h5-6,8-10H,2-4,7H2,1H3,(H,23,24)(H,25,26) | PDB
UniProtKB/SwissProt
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PubMed
| n/a | n/a | 80 | n/a | n/a | n/a | n/a | n/a | n/a |
Kalypsys, Inc.
Curated by ChEMBL
| Assay Description
Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hr |
Bioorg Med Chem Lett 20: 2928-32 (2010)
Article DOI: 10.1016/j.bmcl.2010.03.023
BindingDB Entry DOI: 10.7270/Q2VD6ZMF |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4B
(Homo sapiens (Human)) | BDBM50092350
((5-Cyclopentyloxy-6-methoxy-phthalazin-1-yl)-(3,5-...)Show InChI InChI=1S/C19H18Cl2N4O2/c1-26-16-7-6-12-13(18(16)27-11-4-2-3-5-11)8-23-25-19(12)24-17-14(20)9-22-10-15(17)21/h6-11H,2-5H2,1H3,(H,22,24,25) | PDB
UniProtKB/SwissProt
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PC cid
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UniChem
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| Article
PubMed
| n/a | n/a | 400 | n/a | n/a | n/a | n/a | n/a | n/a |
Kalypsys, Inc.
Curated by ChEMBL
| Assay Description
Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hr |
Bioorg Med Chem Lett 20: 2928-32 (2010)
Article DOI: 10.1016/j.bmcl.2010.03.023
BindingDB Entry DOI: 10.7270/Q2VD6ZMF |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4B
(Homo sapiens (Human)) | BDBM50317599
(5-(cyclopentyloxy)-N-(3,5-dichloropyridin-4-yl)-6-...)Show InChI InChI=1S/C20H19Cl2N3O2/c1-26-17-7-6-14-13(19(17)27-12-4-2-3-5-12)8-9-24-20(14)25-18-15(21)10-23-11-16(18)22/h6-12H,2-5H2,1H3,(H,23,24,25) | PDB
UniProtKB/SwissProt
antibodypedia
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AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Patents
| Article
PubMed
| n/a | n/a | 500 | n/a | n/a | n/a | n/a | n/a | n/a |
Kalypsys, Inc.
Curated by ChEMBL
| Assay Description
Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hr |
Bioorg Med Chem Lett 20: 2928-32 (2010)
Article DOI: 10.1016/j.bmcl.2010.03.023
BindingDB Entry DOI: 10.7270/Q2VD6ZMF |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4B
(Homo sapiens (Human)) | BDBM50317605
(4-(4-(3,5-dichloropyridin-4-ylamino)-7-methoxy-2-o...)Show SMILES COc1ccc2c(Nc3c(Cl)cncc3Cl)cc(=O)oc2c1OCCCC(O)=O Show InChI InChI=1S/C19H16Cl2N2O6/c1-27-14-5-4-10-13(23-17-11(20)8-22-9-12(17)21)7-16(26)29-18(10)19(14)28-6-2-3-15(24)25/h4-5,7-9H,2-3,6H2,1H3,(H,22,23)(H,24,25) | PDB
UniProtKB/SwissProt
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PC cid
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UniChem
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| Article
PubMed
| n/a | n/a | 1.18E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Kalypsys, Inc.
Curated by ChEMBL
| Assay Description
Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hr |
Bioorg Med Chem Lett 20: 2928-32 (2010)
Article DOI: 10.1016/j.bmcl.2010.03.023
BindingDB Entry DOI: 10.7270/Q2VD6ZMF |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4B
(Homo sapiens (Human)) | BDBM50317600
(8-(cyclopentyloxy)-N-(3,5-dichloropyridin-4-yl)-7-...)Show InChI InChI=1S/C19H18Cl2N4O2/c1-26-15-7-6-12-16(18(15)27-11-4-2-3-5-11)23-10-24-19(12)25-17-13(20)8-22-9-14(17)21/h6-11H,2-5H2,1H3,(H,22,23,24,25) | PDB
UniProtKB/SwissProt
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AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Patents
| Article
PubMed
| n/a | n/a | 2.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Kalypsys, Inc.
Curated by ChEMBL
| Assay Description
Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hr |
Bioorg Med Chem Lett 20: 2928-32 (2010)
Article DOI: 10.1016/j.bmcl.2010.03.023
BindingDB Entry DOI: 10.7270/Q2VD6ZMF |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4B
(Homo sapiens (Human)) | BDBM50317598
(8-(cyclopentyloxy)-N-(3,5-dichloropyridin-4-yl)-7-...)Show InChI InChI=1S/C20H19Cl2N3O2/c1-26-17-7-6-13-16(25-19-14(21)10-23-11-15(19)22)8-9-24-18(13)20(17)27-12-4-2-3-5-12/h6-12H,2-5H2,1H3,(H,23,24,25) | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Patents
| Article
PubMed
| n/a | n/a | 3.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Kalypsys, Inc.
Curated by ChEMBL
| Assay Description
Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hr |
Bioorg Med Chem Lett 20: 2928-32 (2010)
Article DOI: 10.1016/j.bmcl.2010.03.023
BindingDB Entry DOI: 10.7270/Q2VD6ZMF |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4B
(Homo sapiens (Human)) | BDBM50317601
(3,5-dichloro-N-(7-(cyclopentyloxy)-6-methoxybenzof...)Show InChI InChI=1S/C19H18Cl2N2O3/c1-24-16-7-6-12-15(23-17-13(20)8-22-9-14(17)21)10-25-18(12)19(16)26-11-4-2-3-5-11/h6-11H,2-5H2,1H3,(H,22,23) | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Patents
Similars
| Article
PubMed
| n/a | n/a | 1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kalypsys, Inc.
Curated by ChEMBL
| Assay Description
Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hr |
Bioorg Med Chem Lett 20: 2928-32 (2010)
Article DOI: 10.1016/j.bmcl.2010.03.023
BindingDB Entry DOI: 10.7270/Q2VD6ZMF |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4B
(Homo sapiens (Human)) | BDBM50317602
(3,5-dichloro-N-(8-(cyclopentyloxy)-7-methoxychroma...)Show InChI InChI=1S/C20H22Cl2N2O3/c1-25-17-7-6-13-16(24-18-14(21)10-23-11-15(18)22)8-9-26-19(13)20(17)27-12-4-2-3-5-12/h6-7,10-12,16H,2-5,8-9H2,1H3,(H,23,24) | PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Patents
| Article
PubMed
| n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kalypsys, Inc.
Curated by ChEMBL
| Assay Description
Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hr |
Bioorg Med Chem Lett 20: 2928-32 (2010)
Article DOI: 10.1016/j.bmcl.2010.03.023
BindingDB Entry DOI: 10.7270/Q2VD6ZMF |
More data for this
Ligand-Target Pair | |
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