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| Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Voltage-dependent T-type calcium channel subunit alpha-1H (Homo sapiens (Human)) | BDBM50117922 ((1S,2S)-2-(2-((3-(1H-benzo[d]imidazol-2-yl)propyl)...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet  | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 32 | n/a | n/a | n/a | n/a | n/a | n/a |
Icagen, Inc. Curated by ChEMBL | Assay Description Antagonist activity against T-type calcium channel subunit alpha-1H assessed as inactivation of channel current by cell based patch clamp assay | Bioorg Med Chem Lett 20: 6375-8 (2010) Article DOI: 10.1016/j.bmcl.2010.09.098 BindingDB Entry DOI: 10.7270/Q2ZW1M5B | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Voltage-dependent N-type calcium channel subunit alpha-1B (Homo sapiens (Human)) | BDBM50117922 ((1S,2S)-2-(2-((3-(1H-benzo[d]imidazol-2-yl)propyl)...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 416 | n/a | n/a | n/a | n/a | n/a | n/a |
Icagen, Inc. Curated by ChEMBL | Assay Description Antagonist activity against L-type calcium channel subunit alpha-1C assessed as inactivation of channel current by cell based patch clamp assay | Bioorg Med Chem Lett 20: 6375-8 (2010) Article DOI: 10.1016/j.bmcl.2010.09.098 BindingDB Entry DOI: 10.7270/Q2ZW1M5B | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
